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2

Total database: 17430
Struktur (SMILES)
2 (100.0%)
Target
2 (100.0%)
Genomik
0 (0%)
Referensi
2 (100.0%)

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Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (2)

Methimazole Approved DB00763
small molecule | CAS: 60-56-0

Methimazole is a thionamide antithyroid agent that inhibits the synthesis of thyroid hormones.[A184559,A184733,A184694] It was first introduced as an antithyroid agent in 1949[A184502] and is now commonly used in the management of hyperthyroidism, particularl…

Kategori:
Antithyroid agentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +30
Target Protein:
Thyroid peroxidase
Waktu ParuhFollowing a single …
Vol. DistribusiThe apparent volume…
KlirensFollowing a single …
Genetik -
Propylthiouracil Approved DB00550
small molecule | CAS: 51-52-5

A thiourea antithyroid agent. Propythiouracil inhibits the synthesis of thyroxine and inhibits the peripheral conversion of throxine to tri-iodothyronine. It is used in the treatment of hyperthyroidism. (From Martindale, The Extra Pharmacopeoia, 30th ed, p534)

Kategori:
Agents Causing Muscle ToxicityAntimetabolitesAntithyroid agents +14
Target Protein:
Type I iodothyronine deiodinaseThyroid peroxidase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -