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33

Total database: 17430
Struktur (SMILES)
33 (100.0%)
Target
31 (93.9%)
Genomik
3 (9.1%)
Referensi
33 (100.0%)

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Hasil Pencarian (33)

Acepromazine DB01614
small molecule | CAS: 61-00-7

Acepromazine is one of the phenothiazine derivative psychotropic drugs, used little in humans, however frequently in animals as a sedative and antiemetic.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +24
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A +3
Waktu Paruh3 hours in horses.
Vol. Distribusi-
Klirens-
Genetik -
Alimemazine Approved DB01246
small molecule | CAS: 84-96-8

A phenothiazine derivative that is used as an antipruritic.

Kategori:
Antihistamines for Systemic UseAntipruriticsAntipsychotic Agents +13
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amoxapine Approved DB00543
small molecule | CAS: 14028-44-5

Amoxapine, the <i>N</i>-demethylated derivative of the antipsychotic agent loxapine, is a dibenzoxazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine subs…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +49
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterD(2) dopamine receptor +22
Waktu Paruh8 hours
Vol. DistribusiWidely distributed …
Klirens-
Genetik -
Biperiden Approved DB00810
small molecule | CAS: 514-65-8

A muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. It has also been used to alleviate extrapyramidal symptoms induc…

Kategori:
Agents producing tachycardiaAnti-Dyskinesia AgentsAnti-Parkinson Drugs +18
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorpromazine Approved DB00477
small molecule | CAS: 50-53-3

The prototypical phenothiazine antipsychotic drug. Like the other drugs in this class, chlorpromazine's antipsychotic actions are thought to be due to long-term adaptation by the brain to blocking dopamine receptors. Chlorpromazine has several other actions a…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +63
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 1A +21
Waktu Paruh~ 30 hours
Vol. Distribusi* 20 L/kg
Klirens-
Genetik -
Clomipramine Approved DB01242
small molecule | CAS: 303-49-1

Clomipramine, the 3-chloro analog of imipramine, is a dibenzazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-de…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +45
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2B +3
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhFollowing oral admi…
Vol. Distribusi~ 17 L/kg (range: 9…
Klirens-
Genetik 9 Varian
Clopenthixol DB13841
small molecule | CAS: 982-24-1

Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyamemazine DB09000
small molecule | CAS: 3546-03-0

Cyamemazine (Tercian), also known as cyamepromazine, is a typical antipsychotic drug of the phenothiazine class used primarily in the treatment of schizophrenia and psychosis-associated anxiety. Cyamemazine actually behaves like an atypical antipsychotic, due…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntipsychotic Agents +16
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desipramine Approved DB01151
small molecule | CAS: 50-47-5

Desipramine hydrochloride is a dibenzazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individuals, de…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +52
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +14
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu Paruh7-60+ hours; 70% el…
Vol. Distribusi-
Klirens-
Genetik 7 Varian
small molecule | CAS: 63834-04-8

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal DisordersSynthetic Antispasmodics, Amides With Tertiary Amines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluphenazine Approved DB00623
small molecule | CAS: 69-23-8

A phenothiazine used in the treatment of psychoses. Its properties and uses are generally similar to those of chlorpromazine.

Kategori:
Agents that reduce seizure thresholdAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +24
Target Protein:
5-hydroxytryptamine receptor 1BD(2) dopamine receptorD(1A) dopamine receptor +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imipramine Approved DB00458
small molecule | CAS: 50-49-7

Imipramine, the prototypical tricyclic antidepressant (TCA), is a dibenzazepine-derivative TCA. TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +70
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +21
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhImipramine has a me…
Vol. DistribusiImipramine has a hi…
KlirensImipramine has a me…
Genetik 9 Varian
Mesoridazine Approved DB00933
small molecule | CAS: 5588-33-0

A phenothiazine antipsychotic with effects similar to chlorpromazine.

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +23
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh24 to 48 hours
Vol. Distribusi-
Klirens-
Genetik -
Methdilazine Approved DB00902
small molecule | CAS: 1982-37-2

Methdilazine is a phenothiazine compound with antihistaminic activity. It is used in the treatment of various dermatoses to relieve pruritus.

Kategori:
Agents that reduce seizure thresholdAntihistamines for Systemic UseHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methotrimeprazine Approved DB01403
small molecule | CAS: 60-99-1

A phenothiazine with pharmacological activity similar to that of both chlorpromazine and promethazine. It has the histamine-antagonist properties of the antihistamines together with central nervous system effects resembling those of chlorpromazine. (From Mart…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +46
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor +16
Waktu ParuhApproximately 20 ho…
Vol. Distribusi-
Klirens-
Genetik -
Moricizine Approved DB00680
small molecule | CAS: 31883-05-3

An antiarrhythmia agent used primarily for ventricular rhythm disturbances.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +15
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh2 hours (range 1.5-…
Vol. Distribusi* 300 L
Klirens-
Genetik -
Periciazine Approved DB01608
small molecule | CAS: 2622-26-6

Periciazine is a phenothiazine of the piperidine group. It has been shown to reduce pathologic arousal and affective tension in some psychotic patients, while the symptoms of abnormal mental integration are relatively unaffected. It is a sedative phenothiazin…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +12
Target Protein:
D(1A) dopamine receptorAlpha-2A adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perphenazine Approved DB00850
small molecule | CAS: 58-39-9

An antipsychotic phenothiazine derivative with actions and uses similar to those of chlorpromazine.

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Central Nervous System Agents +28
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorCalmodulin
Waktu Paruh8-12 hours, but ran…
Vol. Distribusi-
Klirens-
Genetik -
Phenothiazine DB11447
small molecule | CAS: 92-84-2

Phenothiazine (PTZ) is an organic thiazine compound.

Kategori:
Agents that reduce seizure thresholdAnti-Infective AgentsAntiparasitic Agents +3
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipotiazine Approved DB01621
small molecule | CAS: 39860-99-6

Pipotiazine has actions similar to those of other phenothiazines. Among the different phenothiazine derivatives, it appears to be less sedating and to have a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetic…

Kategori:
Antidepressive AgentsAntipsychotic AgentsCentral Nervous System Depressants +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prochlorperazine Approved DB00433
small molecule | CAS: 58-38-8

Prochlorperazine, also known as compazine, is a piperazine phenothiazine and first-generation antipsychotic drug that is used for the treatment of severe nausea and vomiting, as well as short-term management of psychotic disorders such as generalized non-psyc…

Kategori:
AntiemeticsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +28
Target Protein:
D(2) dopamine receptorHistamine H1 receptorAlpha-1 adrenergic receptors +1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn a preliminary ph…
KlirensThe mean plasma cle…
Genetik -
Profenamine Approved DB00392
small molecule | CAS: 522-00-9

Profenamine (also known as ethopropazine) is a medication derived from phenothiazine. It is primarily used as an antidyskinetic to treat Parkinsonism. It is sold under the trade name Parsitan in Canada.[L46812] In the US, the marketing of profenamine has been…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAgents producing tachycardia +12
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M1Glutamate receptor ionotropic, NMDA 3A +1
Waktu Paruh1 to 2 hours
Vol. Distribusi-
Klirens-
Genetik -
Promazine Approved DB00420
small molecule | CAS: 58-40-2

A phenothiazine with actions similar to chlorpromazine but with less antipsychotic activity. It is primarily used in short-term treatment of disturbed behavior and as an antiemetic. It is currently not approved for use in the United States.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +49
Target Protein:
D(2) dopamine receptorMuscarinic acetylcholine receptor M55-hydroxytryptamine receptor 2A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promethazine Approved DB01069
small molecule | CAS: 60-87-7

Promethazine, originally known as 3,277 R.P., is an N-dimethylaminopropyl derivative of [phenothiazine] that was developed in France in 1946.[A189901] Promethazine antagonizes a variety of receptors, allowing it to be used for a number of indications includin…

Kategori:
Acid ReducersAgents producing tachycardiaAgents that reduce seizure threshold +44
Target Protein:
Histamine H1 receptorD(2) dopamine receptorMuscarinic acetylcholine receptor M1 +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe intravenous cle…
Genetik -
Propiomazine Approved DB00777
small molecule | CAS: 362-29-8

Propiomazine, an atypical antipsychotic agent, is used to treat both negative and positive symptoms of schizophrenia, acute mania with bipolar disorder, agitation, and psychotic symptoms in dementia. Future uses may include the treatment of obsessive-compulsi…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +20
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protriptyline Approved DB00344
small molecule | CAS: 438-60-8

Protriptyline hydrochloride is a dibenzocycloheptene-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents that produce hypertension +24
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiethylperazine Approved DB00372
small molecule | CAS: 1420-55-9

A dopamine antagonist that is particularly useful in treating the nausea and vomiting associated with anesthesia, mildly emetic cancer chemotherapy agents, radiation therapy, and toxins. This piperazine phenothiazine does not prevent vertigo or motion sicknes…

Kategori:
AntiemeticsAntihistamines for Systemic UseAntipsychotic Agents +16
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thioproperazine DB01622
small molecule | CAS: 316-81-4

Thioproperazine is a potent neuroleptic with antipsychotic properties. Thioproperazine has a marked cataleptic and antiapomorphine activity associated with relatively slight sedative, hypothermic and spasmolytic effects. It is virtually without antiserotonin …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +18
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thioridazine Approved DB00679
small molecule | CAS: 50-52-2

A phenothiazine antipsychotic used in the management of psychoses, including schizophrenia, and in the control of severely disturbed or agitated behavior. It has little antiemetic activity. Thioridazine has a higher incidence of antimuscarinic effects, but a …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh21-25 hours
Vol. Distribusi-
Klirens-
Genetik -
Thiothixene Approved DB01623
small molecule | CAS: 3313-26-6

A thioxanthine used as an antipsychotic agent. Its effects are similar to the phenothiazine antipsychotics.

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +29
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh10-20 hours
Vol. Distribusi-
Klirens-
Genetik -
Trifluoperazine Approved DB00831
small molecule | CAS: 117-89-5

A phenothiazine with actions similar to chlorpromazine. It is used as an antipsychotic and an antiemetic.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptorCalmodulin-1Calmodulin-3 +6
Waktu Paruh10-20 hours
Vol. Distribusi-
Klirens-
Genetik -
Triflupromazine Approved DB00508
small molecule | CAS: 146-54-3

A phenothiazine used as an antipsychotic agent and as an antiemetic.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntidepressive Agents +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2B +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zuclopenthixol Approved DB01624
small molecule | CAS: 53772-83-1

Zuclopenthixol, also known as Zuclopentixol or Zuclopenthixolum, is an antipsychotic agent. Zuclopenthixol is a thioxanthene-based neuroleptic with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine rece…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +34
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +4
Waktu Paruh20 hours (range 12-…
Vol. Distribusi20 L/kg.
Klirensapproximately 0.9 L…
Genetik -