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39

Total database: 17430
Struktur (SMILES)
38 (97.4%)
Target
34 (87.2%)
Genomik
0 (0%)
Referensi
39 (100.0%)

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Hasil Pencarian (39)

Amdinocillin DB01163
small molecule | CAS: 32887-01-7

Amidinopenicillanic acid derivative with broad spectrum antibacterial action. It is poorly absorbed if given orally and is used in urinary infections and typhus. Amdinocillin is not available in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 2Penicillin-binding protein 3 +3
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Amoxicillin Approved DB01060
small molecule | CAS: 26787-78-0

Amoxicillin, or BRL-2333, is a penicillin G derivative first described in the literature in 1972.[A190648] Amoxicillin has similar activity to [penicillin] and [ampicillin], but leads to higher serum concentrations than ampicillin.[A190648] Amoxicillin was…

Kategori:
Alimentary Tract and MetabolismAmidesAminopenicillins +19
Target Protein:
Penicillin binding protein
Waktu ParuhThe half life of am…
Vol. DistribusiThe central volume …
KlirensThe mean clearance …
Genetik -
Ampicillin Approved DB00415
small molecule | CAS: 69-53-4

Ampicillin is a semi-synthetic derivative of penicillin that functions as an orally active broad-spectrum antibiotic.

Kategori:
AmidesAminopenicillinsAnti-Bacterial Agents +14
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 1bPenicillin-binding protein 3 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azidocillin DB08795
small molecule | CAS: 17243-38-8

Azidocillin is a penicillin antibiotic similir to ampicillin.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +8
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 1bPenicillin-binding protein 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azlocillin Approved DB01061
small molecule | CAS: 37091-66-0

Azlocillin is a semisynthetic ampicillin-derived acylureido penicillin.

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +11
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhMean elimination ha…
Vol. Distribusi-
Klirens-
Genetik -
Benzylpenicillin Approved DB01053
small molecule | CAS: 61-33-6

Benzylpenicillin (Penicillin G) is narrow spectrum antibiotic used to treat infections caused by susceptible bacteria. It is a natural penicillin antibiotic that is administered intravenously or intramuscularly due to poor oral absorption. Penicillin G may al…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +5
Waktu ParuhIn adults with norm…
Vol. Distribusi0.53–0.67 L/kg in a…
Klirens560ml/min in health…
Genetik -
Benzylpenicilloyl polylysine Approved DB00895
small molecule | CAS: 31855-75-1

Benzylpenicilloyl polylysine is used as a skin-testing reagent to detect immunoglobulin E antibodies in people with a history of penicillin allergy. The quantitation of in vitro IgE antibodies to the benzylpenicilloyl determinant is a useful tool for evaluati…

Kategori:
AcetamidesAmidesAnti-Bacterial Agents +9
Target Protein:
High affinity immunoglobulin epsilon receptor subunit gammaHigh affinity immunoglobulin epsilon receptor subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carbenicillin Approved DB00578
small molecule | CAS: 4697-36-3

Broad-spectrum semisynthetic penicillin derivative used parenterally. It is susceptible to gastric juice and penicillinase and may damage platelet function.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding proteinBeta-lactamase Toho-1
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Carindacillin Approved DB09319
small molecule | CAS: 35531-88-5

Carindacillin or Carbenicillin isdanyl was an oral penicillin prodrug of [carbenicillin] marketed by Pfizer as Geocillin. It is no longer marketed in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefixime Approved DB00671
small molecule | CAS: 79350-37-1

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding proteinPenicillin-binding protein 2
Waktu ParuhCefixime has a seru…
Vol. DistribusiCefixime has a volu…
KlirensCefixime administer…
Genetik -
Ceftazidime Approved DB00438
small molecule | CAS: 72558-82-8

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +2
Waktu ParuhCeftazidime has an …
Vol. DistribusiCeftazidime has a v…
KlirensThe mean renal clea…
Genetik -
Cloxacillin Approved DB01147
small molecule | CAS: 61-72-3

A semi-synthetic penicillin antibiotic which is a chlorinated derivative of [oxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacAPenicillin-binding protein 2XPenicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclacillin Approved DB01000
small molecule | CAS: 3485-14-1

A cyclohexylamido analog of penicillanic acid.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 3Penicillin binding protein 2a +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dicloxacillin Approved DB00485
small molecule | CAS: 3116-76-5

One of the penicillins which is resistant to penicillinase.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1bPenicillin-binding protein 2a +3
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Flucloxacillin Approved DB00301
small molecule | CAS: 5250-39-5

Antibiotic analog of [cloxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +17
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh0.75–1 hour
Vol. Distribusi-
Klirens-
Genetik -
Fosfomycin Approved DB00828
small molecule | CAS: 23155-02-4

Fosfomycin was discovered in 1969 by scientists at the Spanish Penicillin and Antibiotics Company and is produced by _Streptomyces fradiae_.[A229338,A230348] It may also be produced synthetically and is commercially available as the disodium salt for intraven…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Urinary +7
Target Protein:
UDP-N-acetylglucosamine 1-carboxyvinyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn healthy subjects…
KlirensIn one study, the r…
Genetik -
Hetacillin Approved DB00739
small molecule | CAS: 3511-16-8

Hetacillin is a penicillin beta-lactam antibiotic used in the treatment of bacterial infections caused by susceptible, usually gram-positive, organisms. The name "penicillin" can either refer to several variants of penicillin available, or to the group of ant…

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +8
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 1bPenicillin-binding protein 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isopenicillin N DB03550
small molecule | CAS: 58678-43-6

Deskripsi belum tersedia.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metampicillin DB13836
small molecule | CAS: 6489-97-0

Metampicillin is a penicillin antibiotic prepared by the reaction of ampicillin with formaldehyde. It is hydrolysed in aqueous solution to form ampicillin. Hydrolysis is rapid under acid conditions like the stomach.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meticillin Approved DB01603
small molecule | CAS: 61-32-5

One of the penicillins which is resistant to penicillinase but susceptible to a penicillin-binding protein. It is inactivated by gastric acid so administered by injection.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
MecA PBP2' (penicillin binding protein 2')Penicillin-binding protein 2aPenicillin-binding protein 1b +3
Waktu Paruh25-60 minutes
Vol. Distribusi-
Klirens-
Genetik -
Mezlocillin Approved DB00948
small molecule | CAS: 51481-65-3

Semisynthetic ampicillin-derived acylureido penicillin. It has been proposed for infections with certain anaerobes and may be useful in inner ear, bile, and CNS infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 3 +1
Waktu Paruh1.3 to 4.4 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

N-[(2S,4S,6R)-2-(dihydroxymethyl)-4-hydroxy-3,3-dimethyl-7-oxo-4lambda~4~-thia-1-azabicyclo[3.2.0]hept-6-yl]-2-phenylacetamide is a solid. This compound belongs to the penicillins. These are organic compounds containing the penicillin core structure, which is…

Target Protein:
Penicillin G acylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nafcillin Approved DB00607
small molecule | CAS: 147-52-4

A semi-synthetic antibiotic related to penicillin, Naficillin is a narrow-spectrum beta-lactam antibiotic drug. It is a beta-lactamase-resistant penicillin that is indicated for the treatment of Staphylococcal infections caused by strains that are resistant t…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +17
Target Protein:
Penicillin-binding protein 1bPenicillin-binding protein 2BPenicillin-binding protein 2a +2
Waktu ParuhThe serum half-life…
Vol. DistribusiNafcillin is report…
Klirens-
Genetik -
Oxacillin Approved DB00713
small molecule | CAS: 66-79-5

An antibiotic similar to [flucloxacillin] used in resistant staphylococci infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1A +7
Waktu Paruh20 to 30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Penamecillin DB13739
small molecule | CAS: 983-85-7

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillamine Approved DB00859
small molecule | CAS: 52-67-5

Penicillamine is a pharmaceutical of the chelator class. The pharmaceutical form is D-penicillamine, as L-penicillamine is toxic (it inhibits the action of pyridoxine). It is an ?-amino acid metabolite of penicillin, although it has no antibiotic properties.

Kategori:
Agents Causing Muscle ToxicityAmino AcidsAmino Acids, Peptides, and Proteins +16
Target Protein:
Copper
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemia
Target Protein:
Regulatory protein BlaR1Beta-lactam-inducible penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penimepicycline DB13264
small molecule | CAS: 4599-60-4

Penimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients [L2791]. In the classification of the active ingredients included on this li…

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pheneticillin Approved DB13337
small molecule | CAS: 147-55-7

Pheneticillin (or phenethicillin) is a penicillin antibiotic which is approved for use internationally.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenoxymethylpenicillin Approved DB00417
small molecule | CAS: 87-08-1

Phenoxymethylpenicillin is a narrow spectrum antibiotic also commonly referred to as Penicillin V or Penicillin VK.[A178609] It is a phenoxymethyl analog of Penicillin G, or [benzylpenicillin]. An orally active naturally penicillin, phenoxymethylpenicillin is…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
MecA PBP2' (penicillin binding protein 2')Penicillin-binding protein 1AD-alanyl-D-alanine carboxypeptidase DacB +2
Waktu ParuhUpon oral administr…
Vol. DistribusiFollowing intraveno…
Klirens-
Genetik -
Piperacillin Approved DB00319
small molecule | CAS: 66258-76-2

Semisynthetic, broad-spectrum, ampicillin derived ureidopenicillin antibiotic proposed for pseudomonas infections. It is also used in combination with other antibiotics.

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +15
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2BPenicillin-binding protein 2a +1
Waktu Paruh36-72 minutes
Vol. Distribusi* 101 mL/kg [intrav…
Klirens* 32 - 41 mL/min/1.…
Genetik -
Procaine benzylpenicillin Approved DB09320
small molecule | CAS: 54-35-3

Procaine benzylpenicillin (INN), also known as procaine G penicillin, is an injectable antiobiotic. It is a poorly soluble salt form of penicillin which is a combination of naturally occuring benzylpenicillin (penicillin G) and the local anaesthetic agent pro…

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +16
Target Protein:
Penicillin-binding protein
Waktu ParuhIntramuscular injec…
Vol. DistribusiThe drug is distrib…
Klirens-
Genetik -
Rosoxacin Approved DB00817
small molecule | CAS: 40034-42-2

Rosoxacin is a quinolone derivative antibiotic for the treatment of bacterial infection of respiratory tract, urinary tract, GI, CNS and immuno compromised patients. Rosoxacin is known to be effective against penicillin resistant strains and is a single dose …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sulbactam Approved DB09324
small molecule | CAS: 68373-14-8

Sulbactam is a beta (?)-lactamase inhibitor and a derivative of the basic penicillin nucleus.[L50131] When given in combination with ?-lactam antibiotics, sulbactam produces a synergistic effect as it blocks the enzyme responsible for drug resistance by hydro…

Kategori:
AmidesAnti-Infective AgentsAntibacterials for Systemic Use +10
Target Protein:
Beta-lactamase
Waktu ParuhIn healthy voluntee…
Vol. DistribusiThe steady-state vo…
KlirensEenal clearance is …
Genetik -
Tedizolid Approved DB14569
small molecule | CAS: 856866-72-3

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Tedizolid phosphate Approved DB09042
small molecule | CAS: 856867-55-5

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntidepressive Agents +10
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Ticarcillin Approved DB01607
small molecule | CAS: 34787-01-4

An antibiotic derived from penicillin similar to carbenicillin in action.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Penicillin binding protein 2a
Waktu Paruh1.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Valine Approved DB00161
small molecule | CAS: 72-18-4

Valine is a branched-chain essential amino acid that has stimulant activity. It promotes muscle growth and tissue repair. It is a precursor in the penicillin biosynthetic pathway.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Propionyl-CoA carboxylase beta chain, mitochondrialBranched-chain-amino-acid aminotransferase, cytosolicValine--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -