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Total database: 17430
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Target
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Hasil Pencarian (20)

ABX-196 DB16339
small molecule | CAS: 1161877-58-2

ABX-196 is under investigation in clinical trial NCT03897543 (ABX196 in Combination With Nivolumab in Patients With Hepatocellular Carcinoma).

Kategori:
AmidesCarbohydratesCeramides +8
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Alintegimod DB18879
small molecule | CAS: 1378535-08-0

Alintegimod is under investigation in clinical trial NCT06362369 (A Study of Oral 7HP349 (Alintegimod) in Combination With Ipilimumab Followed by Nivolumab Monotherapy).

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biotech | CAS: 1939126-74-5

Bempegaldesleukin is under investigation in clinical trial NCT03729245 (A Study of NKTR-214 in Combination With Nivolumab Compared With the Investigator's Choice of a Tyrosine Kinase Inhibitor (TKI) Therapy (Either Sunitinib or Cabozantinib Monotherapy) for A…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
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BMS-813160 DB16240
small molecule | CAS: 1286279-29-5

BMS-813160 is under investigation in clinical trial NCT03496662 (BMS-813160 With Nivolumab and Gemcitabine and Nab-paclitaxel in Borderline Resectable and Locally Advanced Pancreatic Ductal Adenocarcinoma (PDAC)).

Kategori:
Cardiovascular Agents
Target Protein:
C-C chemokine receptor type 2C-C chemokine receptor type 5
Waktu Paruh-
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Cabiralizumab DB15082
biotech | CAS: 1613144-80-1

Cabiralizumab is under investigation in clinical trial NCT03502330 (APX005M With Nivolumab and Cabiralizumab in Advanced Melanoma, Non-small Cell Lung Cancer or Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Dostarlimab Approved DB15627
biotech | CAS: 2022215-59-2

Dostarlimab is an IgG<sub>4</sub> humanized monoclonal antibody targeted against the human programmed death receptor-1 (PD-1).[L33320] PD-1 receptors are found on T-cells and, when activated, serve to inhibit immune responses - some cancers leverage this syst…

Kategori:
Amino Acids, Peptides, and ProteinsAnionsAntibodies +21
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAt steady-state, th…
KlirensAt steady-state, th…
Genetik -
Etigilimab DB18854
biotech | CAS: 2044984-83-8

Etigilimab is under investigation in clinical trial NCT04761198 (A Study of Etigilimab and Nivolumab in Subjects With Locally Advanced or Metastatic Tumors.).

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Lomvastomig DB19060
biotech | CAS: 2648840-52-0

Lomvastomig is under investigation in clinical trial NCT04785820 (A Study of Lomvastomig (RO7121661) and Tobemstomig (RO7247669) Compared With Nivolumab in Participants With Advanced or Metastatic Squamous Cell Carcinoma of the Esophagus).

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Nivolumab Approved DB09035
biotech | CAS: 946414-94-4

Nivolumab is a fully human IgG4 antibody targeting the immune checkpoint programmed death receptor-1 (PD-1).[L12129] This antibody was produced entirely in mice and grafted onto human kappa and IgG4 Fc region with the mutation _S228P_ for additional stability…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe serum half life…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
Pegilodecakin DB15162
biotech | CAS: 1966111-35-2

Pegilodecakin is under investigation in clinical trial NCT03382912 (Study of Pegilodecakin (LY3500518) With Nivolumab Compared to Nivolumab Alone Second-line Tx in Participants With Metastatic Non-Small Cell Lung Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Pemlimogene merolisbac is under investigation in clinical trial NCT03371381 (An Efficacy and Safety Study of JNJ-64041757, a Live Attenuated Listeria Monocytogenes Immunotherapy, in Combination With Nivolumab Versus Nivolumab Monotherapy in Participants With …

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Pepinemab DB15155
biotech | CAS: 2097151-87-4

Pepinemab is under investigation in clinical trial NCT03769155 (VX15/2503 With or Without Ipilimumab and/or Nivolumab in Patients With Resectable Stage IIIB-D Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Pexmetinib DB16294
small molecule | CAS: 945614-12-0

Pexmetinib is under investigation in clinical trial NCT04074967 (Study of ARRY-614 Plus Either Nivolumab or Ipilimumab).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Angiopoietin-1 receptor
Waktu Paruh-
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Genetik -
Pixatimod DB19166
small molecule | CAS: 1144617-49-1

Pixatimod is under investigation in clinical trial NCT05061017 (Pixatimod (PG545) Plus Nivolumab in PD-1 Relapsed/refractory Metastatic Melanoma and NSCLC and With Nivolumab and Low-dose Cyclophosphamide in MSS Metastatic Colorectal Carcinoma (Mcrc)).

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Relatlimab Approved DB14851
biotech | CAS: 1673516-98-7

Relatlimab is a human IgG4 monoclonal antibody and novel immune checkpoint inhibitor that targets lymphocyte activation gene-3 (LAG-3).[A246165,L41265] It was the first commercially developed anti-LAG-3 antibody, entering clinical trials in 2013,[A246155] and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Lymphocyte activation gene 3 protein
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensAt steady-state, th…
Genetik -
Renvistobart DB19065
biotech | CAS: 2725062-35-9

Renvistobart is under investigation in clinical trial NCT02913313 (A Study of BMS-986207 Given Alone and in Combination With Nivolumab or With Nivolumab and Ipilimumab in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
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Retifanlimab Approved DB15766
biotech | CAS: 2079108-44-2

Retifanlimab is a humanized IgG4 kappa monoclonal antibody that binds to the programmed death receptor-1 (PD-1), blocking PD-1 interaction with its ligands, programmed death-ligand 1 (PD-L1) and programmed death-ligand 2 (PD-L2). By blocking the PD-1/PD-L1/2 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +11
Target Protein:
Programmed cell death protein 1
Waktu ParuhAt steady-state, re…
Vol. DistribusiAt steady-state, re…
KlirensFollowing the first…
Genetik -
Sitravatinib DB15036
small molecule | CAS: 1123837-84-2

Sitravatinib is under investigation in clinical trial NCT03680521 (Neoadjuvant Sitravatinib in Combination With Nivolumab in Patients With Clear Cell Renal Cell Carcinoma).

Kategori:
AmidesAminesAniline Compounds +3
Target Protein:
Hepatocyte growth factor receptorVascular endothelial growth factor receptor 3Vascular endothelial growth factor receptor 2 +1
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Sotigalimab DB16413
biotech | CAS: 2305607-45-6

Sotigalimab is under investigation in clinical trial NCT03123783 (CD40 Agonistic Antibody APX005M in Combination With Nivolumab).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Tilsotolimod DB16341
biotech | CAS: 1948266-37-2

Tilsotolimod is under investigation in clinical trial NCT03865082 (Study of Tilsotolimod in Combination With Nivolumab and Ipilimumab for the Treatment of Solid Tumors (ILLUMINATE-206)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Toll-like receptor 9
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