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Total database: 17430
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7 (22.6%)
Target
16 (51.6%)
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Hasil Pencarian (31)

small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Genetik -
Antithrombin III human Approved DB11598
biotech | CAS: 9000-94-6

A plasma alpha 2 glycoprotein that accounts for the major antithrombin activity of normal plasma and also inhibits several other enzymes. It is a member of the serpin superfamily.

Kategori:
Alpha-GlobulinsAmino Acids, Peptides, and ProteinsAnticoagulants +18
Target Protein:
Antithrombin-III
Waktu Paruh2.5 - 3.8 hs
Vol. DistribusiDistributed into pl…
Klirens-
Genetik -
Ardeparin Approved DB00407
small molecule | CAS: 9005-49-6

Ardeparin, marketed under the US trade name Normiflo, is a low molecular weight heparin (LMWH) anticoagulant used for the prevention of postoperative venous thrombosis. Ardeparin is derived via peroxide degradation of heparin extracted from porcine intestinal…

Kategori:
Agents causing hyperkalemiaAnticoagulantsCarbohydrates +7
Target Protein:
Antithrombin-IIIHeparin cofactor 2
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Argatroban Approved DB00278
small molecule | CAS: 74863-84-6

Argatroban is a direct, selective thrombin inhibitor. The American College of Cardiologists (ACC) recommend using bivalirudin or argatroban in patients who have had, or at risk for, heparin induced thrombocytopenia (HIT) and are undergoing percutaneous corona…

Kategori:
AmidesAmino AcidsAmino Acids, Basic +22
Target Protein:
Prothrombin
Waktu Paruh39 and 51 minutes
Vol. Distribusi* 174 mL/kg * 12.1…
Klirens* 5.1 L/kg/hr [infu…
Genetik -
biotech | CAS: 106096-93-9

Basic Fibroblast Growth Factor (bFGF) is a single-chain polypeptide growth factor that plays a significant role in the process of wound healing and is a potent inducer of physiologic angiogenesis. Several different forms of the human protein exist ranging fro…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factor 2, antagonists & inhibitors +4
Waktu Paruh-
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Bemiparin Approved DB09258
small molecule | CAS: 91449-79-5

Bemiparin is an antithrombotic and belongs to the group of drugs known as the low molecular weight heparins (LMWH). Like semuloparin, bemiparin is classified as an ultra-LMH because of its low mean molecular mass of 3600 daltons, which is a unique property of…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +6
Target Protein:
Coagulation factor XAntithrombin-IIIHeparin cofactor 2
Waktu ParuhBemiparin, when adm…
Vol. Distribusi5.1 L [A32018].
KlirensElimination occurs …
Genetik -
Certoparin Approved DB09261
small molecule

Certoparin is part of the heparins of low molecular weight that presents high activity against the coagulation factor Xa. It is normally used to prevent deep venous thrombosis.

Kategori:
Agents causing hyperkalemiaAnticoagulantsCarbohydrates +5
Waktu Paruh-
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Dalteparin Approved DB06779
small molecule | CAS: 9005-49-6

Dalteparin, a low molecular weight heparin (LMWH) prepared by nitrous acid degradation of unfractionated heparin of porcine intestinal mucosa origin, is an anticoagulant. It is composed of strongly acidic sulphated polysaccharide chains with an average molecu…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIVascular endothelial growth factor A, long formP-selectin
Waktu ParuhTerminal Half life:…
Vol. Distribusi3 litres
KlirensExcreted via kidney…
Genetik -
Danaparoid Approved DB06754
small molecule | CAS: 308068-55-5

Danaparoid is a low-molecular-weight heparinoid with an average molecular weight of 5500 Daltons consisting of a mixture of glycosaminoglycans [A32565]. The active constituents are heparan, dermatan and [DB09301] [T28], and they are isolated from the porcine …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +9
Target Protein:
Antithrombin-III
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
small molecule | CAS: 24967-94-0

Deskripsi belum tersedia.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansCarbohydrates +5
Waktu Paruh-
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Genetik -
small molecule | CAS: 177021-00-0

Deskripsi belum tersedia.

Kategori:
AnticoagulantsCarbohydratesExperimental Unapproved Treatments for COVID-19 +3
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Genetik -
Enoxaparin Approved DB01225
small molecule | CAS: 9005-49-6

Enoxaparin is a common low-molecular-weight heparin (LMWH) used in the prevention and management of various thromboembolic disorders. Initially approved by the FDA in 1993, it is administered by a subcutaneous or intravenous injection and marketed by several …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +7
Target Protein:
Antithrombin-IIICoagulation factor XProthrombin
Waktu ParuhThe half-life of en…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Factor IX Complex (Human) Approved DB11330
biotech | CAS: 37224-63-8

Factor IX Complex is a sterile, lyophilized concentrate composed of a number of Vitamin K-dependent clotting factors found in functioning human plasma. Also known as prothrombin complex concentrate, products containing this complex often include Factor IX (an…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Waktu Paruh-
Vol. Distribusi-
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Fondaparinux Approved DB00569
small molecule | CAS: 104993-28-4

Fondaparinux (Arixtra) is a synthetic anticoagulant agent consisting of five monomeric sugar units and a O-methyl group at the reducing end of the molecule. It is structurally similar to polymeric glycosaminoglycan heparin and heparan sulfate (HS) when they a…

Kategori:
AnticoagulantsAntithrombinsBlood and Blood Forming Organs +13
Target Protein:
Coagulation factor XAntithrombin-III
Waktu Paruh17-21 hours
Vol. Distribusi* 7 - 11 L (healthy…
Klirens-
Genetik -
Heparin Approved DB01109
small molecule | CAS: 9005-49-6

Unfractionated heparin (UH) is a heterogenous preparation of anionic, sulfated glycosaminoglycan polymers with weights ranging from 3000 to 30,000 Da. It is a naturally occurring anticoagulant released from mast cells. It binds reversibly to antithrombin III …

Kategori:
Agents causing hyperkalemiaAnticoagulantsAntivaricose Therapy +16
Target Protein:
Antithrombin-IIICoagulation factor XP-selectin +9
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensThe clearance in ad…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
C-C motif chemokine 5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
C-C motif chemokine 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Heparin, bovine DB15404
small molecule | CAS: 9005-49-6

Heparin, bovine is under investigation in clinical trial NCT01072747 (Efficacy And Safety Of Unfractionated Heparin In Patients With Cardiovascular Surgery Using Cardiopulmonary Bypass).

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Lepirudin Approved DB00001
biotech | CAS: 138068-37-8

Lepirudin is a recombinant hirudin formed by 65 amino acids that acts as a highly specific and direct thrombin inhibitor.[L41539,L41569] Natural hirudin is an endogenous anticoagulant found in _Hirudo medicinalis_ leeches.[L41539] Lepirudin is produced in yea…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Target Protein:
Prothrombin
Waktu ParuhLepirudin has an in…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of le…
Genetik -
Nadroparin Approved DB08813
small molecule

Nadroparin is a low molecular weight heparin (LMWH) which, when bound to antithrombin III (ATIII), accelerates the inactivation of factor II and factor Xa. Nadroparin halts the coagulation pathway by inhibiting the activation of thrombin (factor IIa) by facto…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIP-selectinProtein c-Fos +1
Waktu ParuhIn healthy patients…
Vol. Distribusi3.59L
KlirensThe clearance of na…
Genetik -
NDX-3315 DB18671
small molecule

NDX-3315 is an investigational radiopharmaceutical agent for the diagnosis, treatment monitoring, and management of eosinophilic esophagitis. It is a technetium-99m radiolabeled [heparin].

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Parnaparin Approved DB09260
small molecule | CAS: 9005-49-6

Parnaparin is an heparin of low molecular weight with antithrombotic effects.

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegmusirudin DB19220
biotech | CAS: 8001-27-2

Pegmusirudin is under investigation in clinical trial NCT00074620 (A Clinical Study to Assess the Safety of Peg-hirudin (SPP200) Compared to Heparin in Patients Who Are on Haemodialysis).

Kategori:
Amino Acids, Peptides, and ProteinsAntithrombin ProteinsEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pentosan polysulfate Approved DB00686
small molecule | CAS: 37300-21-3

Pentosan polysulfate is a sulfated pentosyl polysaccharide with heparin-like properties.

Kategori:
AnticoagulantsAntivaricose TherapyCarbohydrates +12
Target Protein:
Fibroblast growth factor 2Fibroblast growth factor 1Fibroblast growth factor 4
Waktu Paruh4.8 hours
Vol. Distribusi-
Klirens-
Genetik -
PGX-100 DB06114
small molecule

PGX-100 is an intravenous dosage form of modified heparin. It is developed for treatment of exacerbation of obstructive pulmonary disease (COPD) and for the prevention and treatment of cardiac ischemia reperfusion injury (following acute myocardial infarction…

Waktu Paruh-
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Protamine sulfate Approved DB09141
biotech | CAS: 9009-65-8

Since it's earliest discovery in salmon rine sperm heads in the late 1800's to its formal introduction via US FDA approval in 1939, protamine sulfate has occupied an important therapeutic niche as perhaps the only viable option for reversing the anticoagulant…

Kategori:
Amino Acids, Peptides, and ProteinsAntiheparin AgentsHematologic Agents +5
Waktu ParuhThe half-life of pr…
Vol. DistribusiIn a study group of…
KlirensIn a study group of…
Genetik -
Reviparin Approved DB09259
small molecule | CAS: 9041-08-1

Reviparin is a low molecular weight heparin which seems to have a better safety profile than unfractionated heparin.[A32019] It is prepared from porcine intestinal mucosa by nitrous acid depolymerization. Reviparin has a molecular weight of 3.9 kDa.[A32021] I…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sulodexide Approved DB06271
biotech | CAS: 57821-29-1

Sulodexide is a mixture of glycosaminoglycans (GAGs) composed of dermatan sulfate (DS) and fast moving heparin (FMH).

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Heparin cofactor 2Antithrombin-III
Waktu ParuhThe elimination hal…
Vol. DistribusiCmax=516+/-77.54ng/…
Klirens2.70+/-0.58L/h
Genetik -
Taurolidine Approved DB12473
small molecule | CAS: 19388-87-5

Taurolidine is an antimicrobial used for the prevention of catheter-related infections. It is a derivative of the amino acid [taurine]. It was first synthesized in the 1970s and was originally used as a prophylactic against intraperitoneal bacterial infect…

Kategori:
AlkanesAlkanesulfonic AcidsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tinzaparin Approved DB06822
small molecule | CAS: 9041-08-1

Tinzaparin is a low molecular weight heparin (LMWH), produced by enzymatic depolymerization of unfractionated heparin from porcine intestinal mucosa. It is a heterogeneous mixture of with an average molecular weight between 5500 and 7500 daltons. Tinzaparin i…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIIntegrin alpha-4Stromal cell-derived factor 1
Waktu ParuhAnti-Xa activity is…
Vol. DistribusiAnti-Xa activity is…
KlirensClearance is dose-d…
Genetik -