Hasil Pencarian (2)
small molecule | CAS: 740028-90-4
Glycopyrronium, also known as NVA237 or glycopyrrolate, is a racemic mixture of two enantiomers.[L33110] They are both quaternary ammonium compounds and long acting muscarinic antagonists.[L33110] It is one of the most commonly prescribed anticholinergic medi…
Kategori:
Adjuvants, AnesthesiaAdrenergics, InhalantsAgents producing tachycardia
+30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2
+2
Waktu ParuhThe half life after…
Vol. DistribusiThe mean volume of …
KlirensA 6 µg/kg intraveno…
Genetik
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small molecule | CAS: 1628251-49-9
Sofpironium is a "soft" anticholinergic analog of [glycopyrronium] that has been modified with a readily hydrolyzable ester moiety.[L51109] Soft drugs are designed to reduce systemic toxicity while enhancing local efficacy by employing retrometabolic drug des…
Kategori:
Anticholinergic AgentsCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown)
+13
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor
Waktu ParuhThe _in vitro_ half…
Vol. Distribusi-
Klirens-
Genetik
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