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Total database: 17430
Struktur (SMILES)
2 (100.0%)
Target
1 (50.0%)
Genomik
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Hasil Pencarian (2)

Fosinopril Approved DB00492
small molecule | CAS: 98048-97-6

Fosinopril is a phosphinic acid-containing ester prodrug that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is rapidly hydrolyzed to fosinoprilat, its principle active metabolite. Fosinoprilat inhibits ACE, the enzyme r…

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +17
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh12 hours
Vol. Distribusi-
Klirens* 26 - 39 mL/min [h…
Genetik -
Fosinoprilat DB14207
small molecule | CAS: 95399-71-6

Fosinoprilat is the active phosphinic acid metabolite of prodrug [fosinopril], which is activated by esterases in vivo. It binds zinc with phosphinic acid group.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -