Hasil Pencarian (2)
small molecule | CAS: 133099-04-4
Darifenacin (Enablex®, Novartis) is a medication used to treat urinary incontinence. Darifenacin blocks M3 muscarinic acetylcholine receptors, which mediate bladder muscle contractions. This block reduces the urgency to urinate and so it should not be used…
Kategori:
Agents producing tachycardiaAnticholinergic AgentsCholinergic Agents
+15
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2
+2
Waktu ParuhThe elimination hal…
Vol. Distribusi* 163 L
Klirens* 40 L/h [extensive…
Genetik
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small molecule | CAS: 223673-61-8
Mirabegron is a sympathomimetic beta-3 adrenergic receptor agonist used to relax the smooth muscle of the bladder in the treatment of urinary frequency and incontinence. It is unique amongst overactive bladder treatment options in that, unlike other treatment…
Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-3 Receptor Agonists
+32
Target Protein:
Beta-3 adrenergic receptorBeta-1 adrenergic receptor
Waktu ParuhThe mean terminal e…
Vol. DistribusiFollowing intraveno…
KlirensTotal plasma cleara…
Genetik
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