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Total database: 17430
Struktur (SMILES)
3 (60.0%)
Target
3 (60.0%)
Genomik
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Referensi
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Hasil Pencarian (5)

Dabigatran Approved DB14726
small molecule | CAS: 211914-51-1

Dabigatran is the active form of the orally bioavailable prodrug [dabigatran etexilate].

Kategori:
AnticoagulantsAntithrombinsBenzimidazoles +9
Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dabigatran etexilate Approved DB06695
small molecule | CAS: 211915-06-9

Dabigatran etexilate is an oral prodrug that is hydrolyzed to the competitive and reversible direct thrombin inhibitor [dabigatran].[A177463, A6970, L34675, L34680] Dabigatran etexilate may be used to decrease the risk of venous thromboembolic events in patie…

Kategori:
AnticoagulantsAntithrombinsBenzimidazoles +11
Target Protein:
Prothrombin
Waktu ParuhDabigatran has a ha…
Vol. DistribusiDabigatran has a vo…
KlirensFollowing intraveno…
Genetik -
Edoxaban Approved DB09075
small molecule | CAS: 480449-70-5

Edoxaban is a member of the Novel Oral Anti-Coagulants (NOACs) class of drugs, and is a rapidly acting, oral, selective factor Xa inhibitor. By inhibiting factor Xa, a key protein in the coagulation cascade, edoxaban prevents the stepwise amplification of pro…

Kategori:
AnticoagulantsAntithrombinsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
Klirens22 L/hr
Genetik -
Idarucizumab Approved DB09264
biotech | CAS: 1362509-93-0

Idarucizumab is a humanized monoclonal antibody fragment (Fab) derived from an immunoglobulin G1 isotype molecule that binds to and inactivates the oral anticoagulant dabigatran, thereby reversing its anticoagulant effect. As a direct acting oral anticoagulan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruhinitial half-life: …
Vol. Distribusi8.9 L
Klirens47.0 mL/min
Genetik -
Protamine sulfate Approved DB09141
biotech | CAS: 9009-65-8

Since it's earliest discovery in salmon rine sperm heads in the late 1800's to its formal introduction via US FDA approval in 1939, protamine sulfate has occupied an important therapeutic niche as perhaps the only viable option for reversing the anticoagulant…

Kategori:
Amino Acids, Peptides, and ProteinsAntiheparin AgentsHematologic Agents +5
Waktu ParuhThe half-life of pr…
Vol. DistribusiIn a study group of…
KlirensIn a study group of…
Genetik -