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Total database: 17430
Struktur (SMILES)
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Target
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Hasil Pencarian (4)

Cetirizine Approved DB00341
small molecule | CAS: 83881-51-0

Cetirizine, also commonly known as _Zyrtec_, is an orally active second-generation histamine H1 antagonist proven effective in the treatment of various allergic symptoms, such as sneezing, coughing, nasal congestion, hives, and other symptoms [A175051], [A175…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +14
Target Protein:
Histamine H1 receptor
Waktu ParuhPlasma elimination …
Vol. DistribusiApparent volume of …
KlirensApparent total body…
Genetik -
Hydroxyzine Approved DB00557
small molecule | CAS: 68-88-2

Hydroxyzine is a first-generation histamine H<sub>1</sub>-receptor antagonist of the dephenylmethane and piperazine classes that exhibits sedative, anxiolytic, and antiemetic properties.[A1257,A187589] It was first developed in 1955,[A189726] and has since re…

Kategori:
Anti-Anxiety AgentsAntipruriticsCentral Nervous System Depressants +21
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe half-life of hy…
Vol. DistribusiThe mean volume of …
KlirensClearance of hydrox…
Genetik -
Levocetirizine Approved DB06282
small molecule | CAS: 130018-77-8

Levocetirizine is a selective histamine H<sub>1</sub> antagonist used to treat a variety of allergic symptoms.[A181748,A181790,L7694] It is the R enantiomer of [cetirizine].[L7694] Levocetirizine has greater affinity for the histamine H<sub>1</sub> receptor t…

Kategori:
Antihistamines for Systemic UseCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Histamine H1 receptor
Waktu ParuhThe average half li…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Pheniramine Approved DB01620
small molecule | CAS: 86-21-5

Pheniramine is a first-generation antihistamine in the alkylamine class, similar to [brompheniramine] and [chlorpheniramine].[A181628] It is used in some over-the-counter allergy as well as cold & flu products in combination with other drugs. Pheniramine's …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseAntihistamines for Topical Use +10
Target Protein:
Histamine H4 receptorHistamine H1 receptorNuclear receptor subfamily 1 group I member 3
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
Klirens-
Genetik -