Hasil Pencarian (2)
small molecule | CAS: 59803-98-4
Brimonidine is an alpha-adrenergic agonist and 2-imidazoline derivative that was first introduced in 1996.[A178951] It is considered to be a third generation alpha-2 aadrenergic receptor agonist, since it displays preferential binding at alpha-2 adrenoceptors…
Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists
+14
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor
Waktu ParuhFollowing ocular ad…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik
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small molecule | CAS: 138890-62-7
Brinzolamide is a highly specific, non-competitive, reversible carbonic anhydrase II (CA-II) inhibitor indicated to reduce ocular pressure in patients with ocular hypertension or open-angle glaucoma.[L35310] Although the exact pathophysiology of glaucoma is s…
Kategori:
AmidesAntiglaucoma Preparations and MioticsCarbonic Anhydrase Inhibitors
+17
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1Carbonic anhydrase 4
+2
Waktu ParuhDue to its affinity…
Vol. Distribusi-
Klirens-
Genetik
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