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Total database: 17430
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Target
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Hasil Pencarian (2)

Atogepant Approved DB16098
small molecule | CAS: 1374248-81-3

Atogepant is an oral antagonist of calcitonin gene-related peptide (CGRP) receptors indicated for the prevention of episodic migraine headaches. It was developed by AbbVie and received FDA approval under the brand name Qulipta in September 2021.[L38814] While…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Rimegepant Approved DB12457
small molecule | CAS: 1289023-67-1

Rimegepant is an oral antagonist of the CGRP receptor developed by Biohaven Pharmaceuticals.[L11028] It received FDA approval on February 27, 2020 for the acute treatment migraine headache,[L11974] and was subsequently approved by the European Commission in A…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +19
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady state, th…
Klirens-
Genetik -