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Total database: 17430
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Target
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Hasil Pencarian (4)

Andexanet alfa Approved DB14562
biotech | CAS: 1262449-58-0

Andexanet alfa is a recombinant human coagulation Factor Xa that promotes blood coagulation. It was developed by Portola Pharmaceuticals and was approved in in May 2018. It is marketed as Andexxa for intravenous injection or infusion and is indicated for the …

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesBiological Factors +12
Target Protein:
Tissue factor pathway inhibitor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensClearance for andex…
Genetik -
Apixaban Approved DB06605
small molecule | CAS: 503612-47-3

Apixaban is an oral, direct, and highly selective factor Xa (FXa) inhibitor of both free and bound FXa, as well as prothrombinase, independent of antithrombin III for the prevention and treatment of thromboembolic diseases[Label,A6897]. It is marketed under t…

Kategori:
AnticoagulantsAntithrombinsBCRP/ABCG2 Substrates +17
Target Protein:
Coagulation factor X
Waktu Paruh12.7±8.55h[Label,A1…
Vol. DistribusiApproximately 21L[L…
Klirens3.3L/h[Label] thoug…
Genetik -
Edoxaban Approved DB09075
small molecule | CAS: 480449-70-5

Edoxaban is a member of the Novel Oral Anti-Coagulants (NOACs) class of drugs, and is a rapidly acting, oral, selective factor Xa inhibitor. By inhibiting factor Xa, a key protein in the coagulation cascade, edoxaban prevents the stepwise amplification of pro…

Kategori:
AnticoagulantsAntithrombinsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
Klirens22 L/hr
Genetik -
Ichorcumab DB18930
biotech | CAS: 2589583-20-8

Ichorcumab is under investigation in clinical trial NCT03251482 (A Study to Evaluate the Safety and Efficacy of Intravenous JNJ-64179375 Versus Oral Apixaban in Participants Undergoing Elective Total Knee Replacement Surgery).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -