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Total database: 17430
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Target
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Hasil Pencarian (2)

Amrinone Approved DB01427
small molecule | CAS: 60719-84-8

Amrinone (or inamrinone) is a type 3 pyridine phosphodiesterase inhibitor. It is used in the treatment of congestive heart failure.

Kategori:
AminesAminopyridinesCalcium-Regulating Hormones and Agents +14
Target Protein:
cAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)cGMP-inhibited 3',5'-cyclic phosphodiesterase 3AcGMP-inhibited 3',5'-cyclic phosphodiesterase 3B +1
Waktu Paruh5 to 8 hours
Vol. Distribusi* 1.2 L/kg [normal …
Klirens-
Genetik -
Milrinone Approved DB00235
small molecule | CAS: 78415-72-2

Heart failure is a multifactorial condition that affects roughly 1-2% of the adult population. Often the result of long-term myocardial ischemia, cardiomyopathy, or other cardiac insults, heart failure results from an inability of the heart to perfuse periphe…

Kategori:
AminesAminopyridinesCardiac Stimulants Excl. Cardiac Glycosides +12
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhMilrinone administe…
Vol. DistribusiMilrinone administe…
KlirensMilrinone administe…
Genetik -