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Total database: 17430
Struktur (SMILES)
2 (100.0%)
Target
2 (100.0%)
Genomik
0 (0%)
Referensi
2 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (2)

Almorexant DB06673
small molecule | CAS: 871224-64-5

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Orexin/Hypocretin receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Daridorexant Approved DB15031
small molecule | CAS: 1505484-82-1

Daridorexant, formerly known as nemorexant, is a selective dual orexin receptor antagonist used to treat insomnia. Insomnia is characterized by difficulties with sleep onset and/or sleep maintenance and impairment of daytime functioning. It chronically affect…

Kategori:
Central Nervous System DepressantsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +6
Target Protein:
Orexin/Hypocretin receptor type 1Orexin receptor type 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiDaridorexant has a …
KlirensThere is limited in…
Genetik -