Hasil Filter

2

Total database: 17430
Struktur (SMILES)
2 (100.0%)
Target
1 (50.0%)
Genomik
0 (0%)
Referensi
2 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (2)

Bamocaftor DB15177
small molecule | CAS: 2204245-48-5

Bamocaftor (VX-659) is under investigation in clinical trial NCT03224351 (A Study Evaluating the Safety and Efficacy of VX-659 Combination Therapy in Subjects With Cystic Fibrosis).

Kategori:
Chloride Channel AgonistsMembrane Transport Modulators
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elexacaftor Approved DB15444
small molecule | CAS: 2216712-66-0

Elexacaftor (previously VX-445) is a small molecule, next-generation corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) protein.[A187361] It received FDA approval in October 2019 in combination with [tezacaftor] and [ivacaftor] as the…

Kategori:
Cystic Fibrosis Transmembrane Conductance Regulator CorrectorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -