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3

Total database: 17430
Struktur (SMILES)
3 (100.0%)
Target
2 (66.7%)
Genomik
0 (0%)
Referensi
3 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (3)

Rocuronium Approved DB00728
small molecule | CAS: 143558-00-3

Rocuronium (rapid onset-curonium) is a desacetoxy analogue of vecuronium with a more rapid onset of action. It is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and t…

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +16
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M25-hydroxytryptamine receptor 3A
Waktu ParuhThe rapid distribut…
Vol. Distribusi* 0.3 L/kg [3 to <1…
Klirens* 0.25 L/kg/hr [Adu…
Genetik -
Sugammadex Approved DB06206
small molecule | CAS: 343306-71-8

Sugammadex is a selective relaxant binding agent indicated for reversal of neuromuscular blockade induced by rocuronium bromide and vecuronium bromide during surgery. Rocuronium bromide and vecuronium bromide are neuromuscular blocking medications that cause …

Kategori:
AntidotesCarbohydratesCompounds used in a research, industrial, or household setting +6
Waktu ParuhAbout 2 hours
Vol. DistribusiAt steady state, th…
Klirens88L/min
Genetik -
Tubocurarine Approved DB01199
small molecule | CAS: 57-95-4

Tubocurarine is a non-depolarizing neuromuscular blocking agent and the first identified curare alkaloid.[A216008] Curare is one of the names used to describe plant-derived poisons used by indigenous South Americans to coat the tips of hunting arrows and dart…

Kategori:
AlkaloidsAminesAnticholinergic Agents +23
Target Protein:
Neuronal acetylcholine receptor subunit alpha-25-hydroxytryptamine receptor 3AAcetylcholinesterase +1
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -