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Total database: 17430
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Target
24 (49.0%)
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Hasil Pencarian (49)

ADU-S100 DB14722
small molecule | CAS: 1638241-89-0

ADU-S100 (MIW815) is a synthetic cyclic dinucleotide (CDN) agonist (activator) of Stimulator of Interferon Genes (STING), a receptor crucial to activate the innate (endogenous) immune system. ADU-S100 (MIW815) activates all known human and mouse STINGs, and e…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotides
Target Protein:
Stimulator of interferon genes protein
Waktu Paruh-
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Amatuximab DB12845
biotech | CAS: 931402-35-6

Amatuximab has been used in trials studying the treatment and basic science of Mesothelioma, Ovarian Cancer, Ovarian Neoplasms, Pancreatic Cancer, and Mesothelioma, Malignant, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Mesothelin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Anti-GD2 monoclonal antibody 3F8 is under investigation in clinical trial NCT00089258 (Biological Therapy in Treating Patients With Neuroblastoma That Has Not Responded to Previous Treatment).

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Apolizumab DB06467
biotech | CAS: 267227-08-7

Apolizumab is a humanized monoclonal antibody that is being studied as a treatment for hematologic cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Arcitumomab DB17201
biotech | CAS: 154361-48-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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ASI402 DB06373
biotech | CAS: 372075-37-1

ASI402 is a monoclonal antibody that targets an aberrantly glycosylated antigen Mucin 1. It is being investigated in cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mucin-1
Waktu Paruh-
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Basiliximab Approved DB00074
biotech | CAS: 179045-86-4

A recombinant chimeric (murine/human) monoclonal antibody (IgG1k) that functions as an immunosuppressive agent, specifically binding to and blocking the interleukin-2 receptor a-chain (IL-2R alpha, also known as CD25 antigen) on the surface of activated T-lym…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu Paruh7.2 +/- 3.2 days (a…
Vol. Distribusi* 7.8 ± 5.1 L [Pedi…
Klirens* 41 +/- 19 mL/h [A…
Genetik -
Bectumomab DB04962
biotech | CAS: 158318-63-9

Bectumomab (marketed under the trade name LymphoScan®) is a mouse monoclonal antibody and which it's used to treat non-Hodgkin's lymphoma. It has a radioisotope, technetium (99m TC) which it's added.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Besilesomab Approved DB13979
biotech | CAS: 537694-98-7

Besilesomab is a mouse monoclonal antibody labelled with the radioactive isotope technetium-99m for determining the location of inflammation/infection in peripheral bone in adults with suspected osteomyelitis [FDA Label]. Utilised only as a diagnostic agent, …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Carcinoembryonic antigen
Waktu ParuhWhole blood concent…
Vol. DistribusiIn the besilesomab …
KlirensOnce administered i…
Genetik -
biotech | CAS: 400010-39-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +19
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Carotuximab DB06322
biotech | CAS: 1268714-50-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Endoglin
Waktu Paruh-
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CCR5 mAb DB05906
biotech

CCR5 mAb is a fully human monoclonal antibody that specifically recognizes and binds the chemokine receptor CCR5, which is known to be a key facilitator of infection with human immunodeficiency virus (HIV-1). It was generated by HGS using the Abgenix XenoMous…

Target Protein:
C-C chemokine receptor type 5
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Cetuximab Approved DB00002
biotech | CAS: 205923-56-4

Cetuximab is a recombinant chimeric human/mouse IgG1 monoclonal antibody that competitively binds to epidermal growth factor receptor (EGFR) and competitively inhibits the binding of epidermal growth factor (EGF).[A227973] EGFR is a member of the ErbB family …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptorLow affinity immunoglobulin gamma Fc region receptor III-BComplement C1q subcomponent subunit A +5
Gen Terkait:
FCGR2A FCGR3A
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of the d…
KlirensIn patients with re…
Genetik 2 Varian
CPGJ602 DB17485
biotech

CPGJ602 is a recombinant anti-EGFR human-mouse chimeric monoclonal antibody.

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Difelikefalin Approved DB11938
small molecule | CAS: 1024828-77-0

Difelikefalin (CR845) is an agonist of kappa opioid receptors (KORs) useful in the treatment of pruritus secondary to chronic kidney disease. KORs were first associated with itching in 1984.[A237610] Further investigations revealed that dynorphins, endogenous…

Kategori:
Kappa Opioid Receptor Agonist
Target Protein:
Kappa-type opioid receptor
Waktu ParuhThe half-life of di…
Vol. DistribusiThe mean volume of …
KlirensOne cycle of hemodi…
Genetik -
Dinutuximab Approved DB09077
biotech | CAS: 1363687-32-4

Dinutuximab is an IgG1 monoclonal human/mouse chimeric antibody against GD2, a disialoganglioside expressed on tumors of neuroectodermal origin, including human neuroblastoma and melanoma, with highly restricted expression on normal tissues. It is composed of…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
GD2 disialoganglioside
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe mean volume of …
KlirensThe clearance is 0.…
Genetik -
Edobacomab DB17779
biotech | CAS: 141410-98-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Elotuzumab Approved DB06317
biotech | CAS: 915296-00-3

Elotuzumab is a humanized IgG1 (Immunoglobulin G) monoclonal antibody indicated in combination with lenalidomide and dexamethasone for the treatment of patients with multiple myeloma who have received one to three prior therapies. Elotuzumab targets SLAMF7, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
SLAM family member 7
Waktu Paruh-
Vol. Distribusi-
KlirensThe clearance of el…
Genetik -
Emrusolmin DB13927
small molecule | CAS: 882697-00-9

Emrusolmin restores hippocampal synaptic and transcriptional plasticity as well as spatial memory in a mouse model for Alzheimer's disease, when given orally before or after the onset of pathology. [A31409]

Kategori:
DioxolesHeterocyclic Compounds, Fused-Ring
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EP-1043 DB06118
biotech

EP-1043 is an epitope-based recombinant protein vaccine designed to induce HIV-1 specific helper T-lymphocyte (HTL) responses. The vaccine consists of a string of 18 HIV-derived major histocompatibility complex (MHC) Class II restricted epitopes, each separat…

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Etigilimab DB18854
biotech | CAS: 2044984-83-8

Etigilimab is under investigation in clinical trial NCT04761198 (A Study of Etigilimab and Nivolumab in Subjects With Locally Advanced or Metastatic Tumors.).

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Girentuximab DB05304
biotech | CAS: 916138-87-9

Girentuximab is a monoclonal chimeric (mouse/human) antibody directed against carbonic anhydrase IX, an antigen expressed in 95% of clear cell renal cell carcinomas (RCC).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Carbonic anhydrase 9Interleukin-2
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Ibritumomab tiuxetan Approved DB00078
biotech | CAS: 206181-63-7

Indium or yttrium conjugated murine IgG1 kappa monoclonal antibody directed against the CD20 antigen, which is found on the surface of normal and malignant B lymphocytes. Ibritumomab is produced in Chinese hamster ovary cells and is composed of two murine gam…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
B-lymphocyte antigen CD20
Waktu Paruh0.8 hours (mammalia…
Vol. DistribusiBinding observed on…
KlirensApproximately 7.2% …
Genetik -
biotech | CAS: 138660-99-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
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Genetik -
biotech | CAS: 138661-00-4

Indium In-111 imciromab pentetate is a mouse monoclonal antibody labelled with the radioisotope Indium-111 which was used for cardiac imaging under the trade name Myoscint, but was withdrawn in 1993.

Kategori:
Diagnostic Radiopharmaceuticals
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Infliximab Approved DB00065
biotech | CAS: 170277-31-3

Infliximab is a tumor necrosis factor (TNF-alpha or TNF-?) blocker and a chimeric monoclonal IgG1 antibody composed of human constant (75%) and murine variable (25%) regions [A31469]. Infliximab is produced by a recombinant cell line cultured by continuous pe…

Kategori:
Agents Causing Muscle ToxicityAgents reducing cytokine levelsAmino Acids, Peptides, and Proteins +21
Target Protein:
Tumor necrosis factor
Gen Terkait:
FCGR3A
Waktu ParuhThe median terminal…
Vol. DistribusiBased on a pharmaco…
KlirensIn patients with Cr…
Genetik 1 Varian
Inolimomab DB15628
biotech | CAS: 152981-31-2

Inolimomab is under investigation as an agent to treat steroid-resistant graft vs host disease. It has thus far offered similar efficacy to other monoclonal antibody options, though it may carry a higher risk of infections.[A241385]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +9
Target Protein:
Interleukin-2 receptor subunit alpha
Waktu Paruh-
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J147 DB13957
small molecule | CAS: 1146963-51-0

J147 is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging. [A31606,A31607,A31608] It is a curcumin derivative and a potent neurogenic and neuroprotective drug candidate initially develo…

Kategori:
AlkanesBenzene DerivativesCatechols +4
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KT-253 DB18487
small molecule

KT-253 is a selective heterobifunctional small molecule degrader of mouse double minute 2 (MDM2).

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Lirentelimab DB16728
biotech | CAS: 2283348-97-8

Lirentelimab is under investigation in clinical trial NCT04856891 (A Study of Lirentelimab (AK002) in Patients With Active Eosinophilic Duodenitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Margetuximab Approved DB14967
biotech | CAS: 1350624-75-7

The HER2 oncoprotein, the product of the human _ERBB2_/mouse _neu_ genes, is a member of the HER family of receptor tyrosine kinases that includes the epidermal growth factor receptor (EGFR). Of the various subtypes of breast cancer, HER2-positive breast canc…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhMargetuximab has a …
Vol. DistribusiMargetuximab has a …
KlirensMargetuximab has a …
Genetik -
Merimepodib DB04862
small molecule | CAS: 198821-22-6

Merimepodib (VX-497) is a novel noncompetitive inhibitor of IMPDH. Merimepodib is orally bioavailable and inhibits the proliferation of primary human, mouse, rat, and dog lymphocytes at concentrations of approximately 100 nM.

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor +1
Waktu Paruh-
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Molnupiravir DB15661
small molecule | CAS: 2349386-89-4

Molnupiravir (EIDD-2801, MK-4482) is the isopropylester prodrug of [N4-hydroxycytidine].[A193014,A193026] With improved oral bioavailability in non-human primates, it is hydrolyzed _in vivo_, and distributes into tissues where it becomes the active 5’-triphos…

Kategori:
AminesAnti-Infective AgentsAntiinfectives for Systemic Use +13
Waktu ParuhThe half life of th…
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Muromonab Approved DB00075
biotech | CAS: 140608-64-6

Murine monoclonal antibody specific to CD3 T-cell lymphocyte antigens. More specifically it is a purified murine (mouse) monoclonal antibody, directed against the CD3 (T3) receptor on the surface of human T-cells (T-lymphocytes) cultured using the murine asci…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
T-cell surface glycoprotein CD3 delta chainT-cell surface glycoprotein CD3 epsilon chainT-cell surface glycoprotein CD3 gamma chain +2
Waktu Paruh0.8 hours (mammalia…
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Genetik -
Mus musculus skin Approved DB10412
biotech

Mus musculus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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small molecule | CAS: 3258-02-4

N4-Hydroxyctidine, or EIDD-1931, is a ribonucleoside analog which induces mutations in RNA virions.[A193008,A193011] N4-hydroxycytidine was first described in the literature in 1980 as a potent mutagen of bacteria and phage.[A193023] It has shown antiviral ac…

Kategori:
CarbohydratesCytosine NucleotidesExperimental Unapproved Treatments for COVID-19 +6
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Natalizumab Approved DB00108
biotech | CAS: 189261-10-7

Natalizumab is a recombinant humanized IgG4? monoclonal antibody that binds to ?4-integrin.[L48041] While natalizumab was originally approved by the FDA to treat multiple sclerosis in 2004, it was withdrawn from the market following multiple reports of fatal …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Integrin alpha-4Low affinity immunoglobulin gamma Fc region receptor III-BHigh affinity immunoglobulin gamma Fc receptor I +1
Waktu ParuhFollowing the repea…
Vol. DistribusiFollowing the repea…
KlirensFollowing the repea…
Genetik -
Ofatumumab Approved DB06650
biotech | CAS: 679818-59-8

Ofatumumab is a novel anti-CD20 monoclonal antibody that targets B-cells. It is an IgG1? human monoclonal antibody produced from a recombinant murine cell line (NS0) via transgenic mouse and hybridoma technology.[L12612] Ofatumumab works by recognizing antige…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhIn patients with CL…
Vol. DistribusiIn patients with CL…
KlirensIn patients with CL…
Genetik -
Pagibaximab DB17786
biotech | CAS: 595566-61-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Palivizumab Approved DB00110
biotech | CAS: 188039-54-5

Humanized monoclonal antibody (IgG1k) produced by recombinant DNA technology, directed to an epitope in the A antigenic site of the F protein of respiratory syncytial virus (RSV). Synagis is a composite of human (95%) and murine (5%) antibody sequences. The h…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +15
Target Protein:
Fusion glycoprotein F0Low affinity immunoglobulin gamma Fc region receptor III-BComplement C1r subcomponent +6
Waktu Paruh18-20 days (in adul…
Vol. Distribusi-
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Genetik -
Pembrolizumab Approved DB09037
biotech | CAS: 1374853-91-4

Pembrolizumab is a highly selective IgG4-kappa humanized monoclonal antibody against PD-1 receptors. It was generated by grafting the variable sequences of a very high-affinity mouse antihuman PD-1 antibody onto a human IgG4-kappa isotype containing a stabili…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensClearance is modera…
Genetik -
Siltuximab Approved DB09036
biotech | CAS: 541502-14-1

Siltuximab is a chimeric (human-mouse) monoclonal immunoglobulin G1-kappa antibody produced in a Chinese hamster ovary (CHO) cell line by recombinant DNA technology. Siltuximab prevents the binding of IL-6 to soluble and membrane-bound IL-6 receptors by formi…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Interleukin-6
Waktu ParuhThe mean terminal h…
Vol. DistribusiBased on population…
KlirensBody weight was ide…
Genetik -
Sulesomab Approved DB13976
biotech | CAS: 167747-19-5

Market product is Tc99m-labeled murine antibody fragment for nuclear imaging of activated granulocytes.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
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Genetik -
biotech

Tick-borne encephalitis (TBE) is a disease caused by the TBE virus (TBEV), transmitted by ticks from the genus _Ixodes_. The disease course is variable. Some patients will be asymptomatic or experience a mild febrile illness, while others will experience the …

Kategori:
VaccinesViral Vaccines
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Toralizumab DB16384
biotech | CAS: 252662-47-8

Toralizumab is under investigation in clinical trial NCT03605927 (CD40-L Blockade for Prevention of Acute Graft-versus-host Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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UB-612 DB16444
biotech

The UB-612 COVID-19 vaccine was developed by United Biomedical Inc Asia in Taipei as the first COVID-19 “multi-tope” protein-peptide vaccine made up of eight rationally designed components[L30653]. The vaccine incorporates a strong S1-RBD component linked to …

Kategori:
Biological ProductsComplex MixturesVaccines +1
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Urtoxazumab DB17806
biotech | CAS: 502496-16-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Vilobelimab DB16416
biotech | CAS: 2250440-41-4

Vilobelimab is a chimeric monoclonal immunoglobulin G4 (IgG4) antibody that binds to the soluble form of human C5a with high affinity. It consists of mouse anti-human complement factor 5a (C5a) monoclonal binding sites (variable regions of heavy and light cha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Complement C5
Waktu ParuhThe elimination hal…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Vonlerolizumab DB16352
biotech | CAS: 1638935-72-4

Vonlerolizumab is under investigation in clinical trial NCT03029832 (A Study of MOXR0916 in Combination With Atezolizumab Versus Atezolizumab Alone in Participants With Untreated Locally Advanced or Metastatic Urothelial Carcinoma Who Are Ineligible for Cispl…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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