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Total database: 17430
Struktur (SMILES)
2 (100.0%)
Target
2 (100.0%)
Genomik
1 (50.0%)
Referensi
2 (100.0%)

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Hasil Pencarian (2)

Donepezil Approved DB00843
small molecule | CAS: 120014-06-4

In 2016, the global burden of dementia was estimated to be 43.8 million, demonstrating a significant increase from a global prevalence of 20.2 million in 1990.[A182411] Donepezil, also known as Aricept, is a piperidine derivative acetylcholinesterase inhibito…

Kategori:
Anti-Dementia DrugsBCRP/ABCG2 SubstratesBradycardia-Causing Agents +20
Target Protein:
Acetylcholinesterase5-hydroxytryptamine receptor 2ACholinesterase +5
Gen Terkait:
CYP2D6
Waktu ParuhThe average elimina…
Vol. DistribusiThe volume of distr…
KlirensAccording to the FD…
Genetik 1 Varian
Memantine Approved DB01043
small molecule | CAS: 19982-08-2

Initially approved by the FDA in 2013, memantine is an N-methyl-D-aspartate (NMDA) receptor antagonist used in the management of Alzheimer's Disease (AD). It is different from many other Alzheimer's Disease medications, as it works by a different mechanism t…

Kategori:
Anti-Dementia DrugsAnti-Dyskinesia AgentsAnti-Parkinson Drugs +20
Target Protein:
Glutamate (NMDA) receptor5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThis drug is cleare…
Genetik -