Hasil Pencarian (2)
MK-0752
DB12852
small molecule | CAS: 471905-41-6
Mk 0752 is under investigation in clinical trial NCT00572182 (MK0752 in Treating Young Patients With Recurrent or Refractory CNS Cancer).
Kategori:
Acids, AcyclicAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors
+5
Target Protein:
Gamma-secretase subunit PEN-2NicastrinGamma-secretase subunit APH-1B
+2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik
-
MRK-003
DB17015
small molecule | CAS: 623165-93-5
MRK-003 is a potent and selective ?-secretase inhibitor developed by Merck. It is the preclinical analog of [MK-0752], a drug in clinical development.[A252682]
Kategori:
Amyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme InhibitorsGamma Secretase Inhibitors and Modulators
+2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik
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