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Sotalol Approved DB00489
small molecule | CAS: 3930-20-9

Sotalol is a methanesulfonanilide developed in 1960.[A178579] It was the first of the class III anti arrhythmic drugs.[A178579] Sotalol was first approved as an oral tablet on 30 October 1992.[L6334] A racemic mixture of sotalol is currently formulated as a t…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensIn patients with a …
Genetik -