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Carvedilol Approved DB01136
small molecule | CAS: 72956-09-3

Carvedilol is a racemic mixture where the S(-) enantiomer is both a beta and alpha-1 adrenoceptor blocker, and the R(+) enantiomer is an alpha-1 adrenoceptor blocker.[L7889,L7892] It is currently used to treat heart failure, left ventricular dysfunction, and …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +40
Target Protein:
Beta-1 adrenergic receptorAlpha-1A adrenergic receptorAlpha-1 adrenergic receptors +16
Gen Terkait:
ADRB1
Waktu ParuhThe half life of ca…
Vol. DistribusiCarvedilol has a vo…
KlirensThe plasma clearanc…
Genetik 1 Varian