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Sofpironium Approved DB19325
small molecule | CAS: 1628251-49-9

Sofpironium is a "soft" anticholinergic analog of [glycopyrronium] that has been modified with a readily hydrolyzable ester moiety.[L51109] Soft drugs are designed to reduce systemic toxicity while enhancing local efficacy by employing retrometabolic drug des…

Kategori:
Anticholinergic AgentsCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +13
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor
Waktu ParuhThe _in vitro_ half…
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