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Talazoparib Approved DB11760
small molecule | CAS: 1207456-01-6

Talazoparib is an inhibitor of mammalian polyadenosine 5’-diphosphoribose polymerases (PARPs), enzymes responsible for regulating essential cellular functions, such as DNA transcription and DNA repair.[L47236] Developed by Pfizer, talazoparib was first app…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +7
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2
Waktu ParuhThe mean terminal p…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -