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Acetylcarnitine Approved DB08842
small molecule | CAS: 3040-38-8

Acetylcarnitine is an investigational drug in the United states, Italy, United Kingdom, China, Israel, and Norway, and it is approved in Italy, Portugal, Argentina, Chile, Philippines, Australia, and India. Acetylcarnitine can be synthesized, but it is also n…

Kategori:
AminesCentral Nervous System AgentsMicronutrients +6
Waktu Paruh-
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Adagrasib Approved DB15568
small molecule | CAS: 2326521-71-3

Adagrasib (MRTX849) is an oral, small-molecule KRAS inhibitor developed by Mirati Therapeutics. KRAS mutations are highly common in cancer and account for approximately 85% of all RAS family mutations.[A254941] However, the development of KRAS inhibitors has …

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalAntineoplastic and Immunomodulating Agents +21
Target Protein:
GTPase KRas
Waktu ParuhAdagrasib has a ter…
Vol. DistribusiAdagrasib has an ap…
KlirensAdagrasib has an ap…
Genetik -
Alclofenac Approved DB13167
small molecule | CAS: 22131-79-9

Alclofenac is a non-steroidal anti-inflammatory drug. It was withdrawn from the market in the United Kingdom in 1979.

Kategori:
Acetic Acid Derivatives and Related SubstancesAcids, CarbocyclicAgents causing hyperkalemia +14
Target Protein:
Prostaglandin G/H synthase 2
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensFor oral dose of 50…
Genetik -
biotech

Allogeneic processed thymus tissue is used for immune reconstitution in immune disorders where the patients are severely immunocompromised due to the absence of a functional thymus, such as congenital athymia. As part of the immune system, the thymus is an or…

Waktu ParuhThe pharmacokinetic…
Vol. DistribusiThe pharmacokinetic…
KlirensThe pharmacokinetic…
Genetik -
biotech

Anti-GD2 monoclonal antibody 3F8 is under investigation in clinical trial NCT00089258 (Biological Therapy in Treating Patients With Neuroblastoma That Has Not Responded to Previous Treatment).

Waktu Paruh-
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APD668 DB05166
small molecule

APD668 is a novel, highly potent and orally active glucose-dependent insulinotropic receptor (GDIR) agonist intended to more efficiently stimulate insulin release by beta cells in response to elevated blood glucose levels, and to also avoid hypoglycemia.

Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
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ATN-161 DB05491
small molecule | CAS: 262438-43-7

ATN-161 is a non-RGD based integrin binding peptide targeting alpha-5 beta-1 and alpha-v beta-3. It inhibits the migration and adhesion of particular integrins on activated endothelial cells that play a critical role in tumor angiogenesis. This approach targe…

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Besilesomab Approved DB13979
biotech | CAS: 537694-98-7

Besilesomab is a mouse monoclonal antibody labelled with the radioactive isotope technetium-99m for determining the location of inflammation/infection in peripheral bone in adults with suspected osteomyelitis [FDA Label]. Utilised only as a diagnostic agent, …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Carcinoembryonic antigen
Waktu ParuhWhole blood concent…
Vol. DistribusiIn the besilesomab …
KlirensOnce administered i…
Genetik -
Bromopride DB09018
small molecule | CAS: 4093-35-0

Bromopride is a dopamine antagonist used as an antiemetic. Its prokinetic properties are similar to those of metoclopramide. It is unavailable in America or the United Kingdom.

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +22
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
KlirensRenal, 10-14% as or…
Genetik -
Cannabidiol Approved DB09061
small molecule | CAS: 13956-29-1

Cannabidiol, or CBD, is one of at least 85 active cannabinoids identified within the Cannabis plant. It is a major phytocannabinoid, accounting for up to 40% of the Cannabis plant's extract, that binds to a wide variety of physiological targets of the endocan…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnticonvulsants +56
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +36
Waktu ParuhThe CBD component o…
Vol. DistribusiCannabinoids are di…
Klirens-
Genetik -
Cyclandelate Approved DB04838
small molecule | CAS: 456-59-7

A direct-acting smooth muscle relaxant used to dilate blood vessels. It may cause gastrointestinal distress and tachycardia. Cyclandelate is not approved for use in the U.S. or Canada, but is approved in various European countries.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAntiarrhythmic agents +10
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Liver carboxylesterase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Diamorphine Approved DB01452
small molecule | CAS: 561-27-3

Diamorphine (heroin) is a narcotic analgesic that may be habit-forming. It is a controlled substance (opium derivative) listed in the U.S. Code of Federal Regulations, Title 21 Parts 329.1, 1308.11 (1987). Sale is forbidden in the United States by Federal sta…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +16
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhIn humans, administ…
Vol. DistribusiData regarding the …
KlirensSome studies have d…
Genetik -
small molecule

Deskripsi belum tersedia.

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Dinutuximab Approved DB09077
biotech | CAS: 1363687-32-4

Dinutuximab is an IgG1 monoclonal human/mouse chimeric antibody against GD2, a disialoganglioside expressed on tumors of neuroectodermal origin, including human neuroblastoma and melanoma, with highly restricted expression on normal tissues. It is composed of…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
GD2 disialoganglioside
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe mean volume of …
KlirensThe clearance is 0.…
Genetik -
Dronabinol Approved DB00470
small molecule | CAS: 1972-08-3

Dronabinol (marketed as Marinol) is a synthetic form of delta-9-tetrahydrocannabinol (??-THC), the primary psychoactive component of cannabis (marijuana). THC demonstrates its effects through weak partial agonist activity at Cannabinoid-1 (CB1R) and Cannabino…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnalgesics +47
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2
Waktu ParuhThe elimination pha…
Vol. DistribusiDronabinol has a la…
KlirensThe value for clear…
Genetik -
Efepoetin alfa DB19197
biotech | CAS: 1905452-78-9

Efepoetin alfa is under investigation in clinical trial NCT04155125 (A Study of Efepoetin Alfa in Treating Anaemia Associated With Chronic Kidney Diseases Patient).

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Efinopegdutide DB15077
biotech | CAS: 2055640-93-0

Efinopegdutide is under investigation in clinical trial NCT03606057 (A Study to Investigate the Effect of JNJ-64565111 on Cardiac Repolarization (Corrected QT Interval) Compared With Placebo in Healthy Adults: a Thorough ECG Study Employing Placebo, JNJ-64565…

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Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1644543-31-6

Efmitermant alfa, a locally-acting GDF/activin ligand trap, is under investigation in clinical trial NCT03124459 (Study of ACE-083 in Patients With Charcot-marie-tooth Disease).

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Ergidina DB18565
biotech

Ergidina is a recombinant human minibody against complement component C5 fused with RGD-motif.

Waktu Paruh-
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Fenebrutinib DB14785
small molecule | CAS: 1434048-34-6

Fenebrutinib is under investigation in clinical trial NCT03174041 (A Drug-Drug Interaction Study Between GDC-0853 and Midazolam, Itraconazole, Rosuvastatin, and Simvastatin).

Kategori:
Pyridines
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
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Genetik -
Flotetuzumab DB15223
biotech | CAS: 1664355-28-5

Flotetuzumab is under investigation in clinical trial NCT02152956 (Safety Study of MGD006 in Relapsed/Refractory Acute Myeloid Leukemia (AML) or Intermediate-2/High Risk MDS).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Foreskin fibroblast-like stromal cells (FDSCs) are progenitors isolated from human tissue that can differentiate into various cell types [A32660]. Also known as Dermagraft, this device is a cryopreserved human fibroblast-derived dermal substitute. Composed…

Kategori:
Allogeneic Cultured Cell Scaffold
Target Protein:
Vascular endothelial growth factor receptor 1Interleukin-6Interleukin-1 receptor type 1 +8
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gadoteric acid Approved DB09132
small molecule | CAS: 72573-82-1

Gadoteric acid, commonly used in the salt form gadoterate meglumine, is a macrocyclic, ionic gadolinium-based contrast agent (GBCA).[A263131] It is composed of the organic acid DOTA (1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid) used for its chel…

Kategori:
AlcoholsAmino SugarsCarbohydrates +12
Waktu ParuhFollowing an intrav…
Vol. DistribusiThe volume of distr…
KlirensIn healthy subjects…
Genetik -
Gadoteridol Approved DB00597
small molecule | CAS: 120066-54-8

Gadoteridol is a macrocyclic nonionic gadolinium that provides contrast enhancement of the brain, spine, and surrounding tissues, resulting in improved visualization (compared with unenhanced MRI) of lesions with abnormal vascularity or those thought to disru…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe plasma distribu…
KlirensThe renal and plasm…
Genetik -
Gadoxetic acid Approved DB08884
small molecule | CAS: 135326-11-3

Gadoxetic acid (gadoxetate) is a paramagnetic gadolinium-containing ionic linear contrast agent in which its salt form, gadoxetate disodium, is used for intravenous injection. Ethoxybenzyl diethylenetriaminepentaacetic acid is the moiety that chelates with a …

Kategori:
AcetatesAcids, AcyclicAmines +13
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe total volume of…
KlirensA total serum clear…
Genetik -
small molecule | CAS: 17465-86-0

Gamma cyclodextrin is under investigation in clinical trial NCT03931057 (The use of ADV6209 for Premedication in Pediatric Anesthesia).

Kategori:
CarbohydratesCyclodextrinsDextrins +4
Waktu Paruh-
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Genetik -
GDC-0134 DB17079
small molecule | CAS: 1637394-01-4

Deskripsi belum tersedia.

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GDC-0152 DB12380
small molecule | CAS: 873652-48-3

GDC-0152 has been used in trials studying the treatment of Solid Cancers.

Kategori:
Cycloparaffins
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
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GDC-0349 DB13072
small molecule | CAS: 1207360-89-1

GDC-0349 has been used in trials studying the treatment of Non-Hodgkin's Lymphoma, Solid Tumor.

Kategori:
AmidesBenzene Derivatives
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GDC-0425 DB14791
small molecule | CAS: 1627539-18-7

GDC-0425 is under investigation in clinical trial NCT01359696 (A Study Evaluating the Safety, Tolerability, and Pharmacokinetics of GDC-0425 Administered With and Without Gemcitabine in Patients With Refractory Solid Tumors or Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0623 DB11982
small molecule | CAS: 1168091-68-6

GDC-0623 has been used in trials studying the treatment of Solid Cancers.

Kategori:
Nicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
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GDC-0810 DB12253
small molecule | CAS: 1365888-06-7

ARN-810 has been used in trials studying the basic science and treatment of Breast Cancer.

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0917 DB12336
small molecule | CAS: 1446182-94-0

CUDC-427 has been used in trials studying the treatment of LYMPHOMA and Solid Cancers.

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GDC-0927 DB14934
small molecule | CAS: 2100830-77-9

GDC-0927 is under investigation in clinical trial NCT02316509 (A Study of GDC-0927 in Postmenopausal Women With Locally Advanced or Metastatic Estrogen Receptor Positive Breast Cancer).

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GDC-1971 DB17487
small molecule | CAS: 2377352-49-1

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GDP-mannose 6-dehydrogenase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GDP-L-fucose DB18689
small molecule | CAS: 15839-70-0

Deskripsi belum tersedia.

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Vol. Distribusi-
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Genetik -
GDX012 DB18448
biotech

Deskripsi belum tersedia.

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Gluconolactone Approved DB04564
small molecule | CAS: 90-80-2

Gluconolactone is a naturally-occurring food additive used as a sequestrant, an acidifier, or a curing, pickling, or leavening agent. It is a cyclic ester of D-gluconic acid. Pure gluconolactone is a white odorless crystalline powder.

Kategori:
Acids, AcyclicCalculi Dissolution AgentCarbohydrates +3
Target Protein:
Lactase/phlorizin hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanosine DB02857
small molecule | CAS: 118-00-3

Guanosine is a nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a ?-N9-glycosidic bond. Guanosine can be phosphorylated to become GMP (guanosine monophosphate), cGMP (cyclic guanosine monophosphate), GDP (guanosine diphosphate) and G…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunitPurine nucleoside phosphorylase +2
Waktu Paruh-
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Genetik -
Hexobendine Approved DB13265
small molecule | CAS: 54-03-5

Hexobendine is a medication used to cause vasodilation, to treat several conditions including angina pectoris. It has not been approved in the United States or the United Kingdom, but has been used widely in Austria and Germany [T478].

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

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Vol. Distribusi-
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Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

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Lanreotide Approved DB06791
small molecule | CAS: 108736-35-2

Lanreotide is a drug employed in the management of acromegaly (a hormonal condition caused by excess growth hormone) in addition to symptoms caused by neuroendocrine tumors, especially carcinoid syndrome. This drug is a long-acting analog of the drug somatost…

Kategori:
AcromegalyAmino Acids, Peptides, and ProteinsAntineoplastic Agents +22
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5
Waktu ParuhHalf-life is approx…
Vol. DistribusiEstimated Volume of…
KlirensEstimated Clearance…
Genetik -
LGD-1550 DB05785
small molecule | CAS: 178600-20-9

LGD-1550 is an orally-active synthetic aromatic retinoic acid agent with potential antineoplastic and chemopreventive activities.

Kategori:
AlkenesBiological FactorsCarotenoids +8
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor betaRetinoic acid receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-2226 DB08089
small molecule | CAS: 328947-93-9

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-3303 DB13937
small molecule | CAS: 917891-35-1

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
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LGD-6972 DB14779
small molecule | CAS: 1207989-09-0

LGD-6972 is under investigation in clinical trial NCT01919684 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of LGD-6972 in Healthy Subjects and Subjects With Type 2 Diabetes Mellitus).

Kategori:
Acids, CarbocyclicAlkanesAlkanesulfonic Acids +7
Target Protein:
Glucagon receptor
Waktu Paruh-
Vol. Distribusi-
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LGD2941 DB05234
small molecule

LGD2941 is a non-steroidal, selective androgen receptor modulator (SARM) developed jointly by Ligand and TAP.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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