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Raloxifene Approved DB00481
small molecule | CAS: 84449-90-1

Raloxifene is a second generation selective estrogen receptor modulator (SERM) that mediates anti-estrogenic effects on breast and uterine tissues, and estrogenic effects on bone, lipid metabolism, and blood coagulation.[A4979,T28] Exhibiting tissue-specific …

Kategori:
BCRP/ABCG2 SubstratesBenzene DerivativesBenzylidene Compounds +23
Target Protein:
Estrogen receptorEstrogen receptor betaSerpin B9 +1
Waktu ParuhThe average plasma …
Vol. DistribusiFollowing oral admi…
KlirensFollowing intraveno…
Genetik -