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Binimetinib Approved DB11967
small molecule | CAS: 606143-89-9

Binimetinib, also known as _Mektovi_, is a potent and selective oral mitogen-activated protein kinase 1/2 (MEK 1/2) inhibitor which is combined with [Encorafenib].[A34275,L3335] On June 27, 2018, the Food and Drug Administration approved the combination of…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +16
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 2Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensThe apparent cleara…
Genetik -