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Imatinib Approved DB00619
small molecule | CAS: 152459-95-5

Imatinib is a small molecule kinase inhibitor that revolutionized the treatment of cancer, particularly chronic myeloid leukemia, in 2001.[A249305] It was deemed a "miracle drug" due to its clinical success, as oncologist Dr. Brian noted that "complete hemato…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Breakpoint cluster region proteinInduced myeloid leukemia cell differentiation protein Mcl-1Mast/stem cell growth factor receptor Kit +8
Waktu ParuhFollowing oral admi…
Vol. DistribusiPopulation pharmaco…
KlirensTypically, clearanc…
Genetik -