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Ertugliflozin Approved DB11827
small molecule | CAS: 1210344-57-2

Ertugliflozin is a sodium-dependent glucose cotransporter-2 (SGLT2) inhibitor used to treat type II diabetes mellitus. It works to block glucose reabsorption from the glomerulus.[A31581] Ertugliflozin was first approved by the FDA in December 2017.[A26195…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 SubstratesBlood Glucose Lowering Agents +9
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensIn one clinical inv…
Genetik -