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Elacestrant Approved DB06374
small molecule | CAS: 722533-56-4

Elacestrant is a non-steroidal small molecule and an estrogen receptor (ER) antagonist.[A256838,L44918] In January 2023, it was approved by the FDA for the treatment of ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer.[L44918,L449…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiElacestrant has an …
KlirensElacestrant has an …
Genetik -