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Elexacaftor Approved DB15444
small molecule | CAS: 2216712-66-0

Elexacaftor (previously VX-445) is a small molecule, next-generation corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) protein.[A187361] It received FDA approval in October 2019 in combination with [tezacaftor] and [ivacaftor] as the…

Kategori:
Cystic Fibrosis Transmembrane Conductance Regulator CorrectorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -