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small molecule | CAS: 157-03-9

6-diazo-5-oxo-L-norleucine is a broad-acting glutamine antagonist.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAminocaproates +7
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Genetik -
Sirpiglenastat DB17536
small molecule | CAS: 2079939-05-0

Sirpiglenastat, also known as DRP-104, is a prodrug of [6-diazo-5-oxo-L-norleucine] (DON), which is a broad-acting glutamine antagonist. It is under investigation in clinical trial NCT04471415 (Study to Investigate DRP-104 in Adults With Advanced Solid Tumors…

Kategori:
AcetatesAcids, AcyclicAmides +1
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