Hasil Filter

13

Total database: 17430
Struktur (SMILES)
13 (100.0%)
Target
10 (76.9%)
Genomik
0 (0%)
Referensi
13 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (13)

small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase SHV-1Beta-lactamaseBeta-lactamase SHV-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase pim-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6051-87-2

?-Naphthoflavone, also known as 5,6-benzoflavone, is a potent agonist of the aryl hydrocarbon receptor and induces cytochromes P450 (CYPs) and uridine 5'-diphospho-glucuronosyltransferases (UGTs). It may be a chemopreventive agent.

Kategori:
BenzoflavonesBenzopyransChromones +7
Target Protein:
Estrogen receptorSteroid hormone receptor ERR1COUP transcription factor 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BI-187004 DB18897
small molecule | CAS: 1303515-32-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CP-271485 DB02118
small molecule | CAS: 35580-46-2

Deskripsi belum tersedia.

Target Protein:
Macrophage metalloelastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Delamanid Approved DB11637
small molecule | CAS: 681492-22-8

Delamanid is an anti-tuberculosis agent derived from the nitro-dihydro-imidazooxazole class of compounds that inhibits mycolic acid synthesis of bacterial cell wall [A31965]. It is used in the treatment of multidrug-resistant and extensively drug-resistant tu…

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsCytochrome P-450 CYP3A Substrates +7
Waktu ParuhThe half life range…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omacetaxine mepesuccinate Approved DB04865
small molecule | CAS: 26833-87-4

Omacetaxine mepesuccinate (formerly known as HHT or Homoharringtonine), is a cephalotaxine ester and protein synthesis inhibitor with established clinical activity as a single agent in hematological malignancies. Omacetaxine mepesuccinate is synthesized from…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic Agents, Phytogenic +7
Target Protein:
50S ribosomal protein L2Large ribosomal subunit protein uL3
Waktu ParuhHomoharringtonine h…
Vol. DistribusiHomoharringtonine h…
KlirensClearance for homoh…
Genetik -
Quizartinib Approved DB12874
small molecule | CAS: 950769-58-1

Quizartinib is an oral and potent fms-like tyrosine kinase 3 (FLT3) inhibitor and it is the first drug developed specifically targeting FLT3, as other agents with FLT3 inhibition activities were investigated with other targets in mind.[A260641] Additionally, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean (SD) effec…
Vol. DistribusiVolume of distribut…
KlirensTotal body clearanc…
Genetik -
Rifampin Approved DB01045
small molecule | CAS: 13292-46-1

Rifampin, also known as rifampicin, is a broad-spectrum antimicrobial [A263748] that was first discovered in 1965 [A263753] and clinically used in 1968.[A263768] Rifampin is used to treat tuberculosis and works by inhibiting the microbial DNA-dependent RNA po…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +55
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhIn healthy adults, …
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
SRT-1720 DB17057
small molecule | CAS: 925434-55-5

SRT-1720 is an activator of NAD(+)-dependent histone deacetylase SIRT1.[A253147]

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tavaborole Approved DB09041
small molecule | CAS: 174671-46-6

Tavaborale is a novel, boron-based topical antifungal medication for the treatment of onychomycosis, a fungal infection of the nail and nail bed due to *Trichophyton rubrum* or *Trichophyton mentagrophytes* infection. Tavaborole functions by inhibiting Leucyl…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
leucine--tRNA ligase
Waktu Paruh28.5 hr
Vol. Distribusi-
Klirens-
Genetik -