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6694

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4518 (67.5%)
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3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 99 / 134
Pegilodecakin DB15162
biotech | CAS: 1966111-35-2

Pegilodecakin is under investigation in clinical trial NCT03382912 (Study of Pegilodecakin (LY3500518) With Nivolumab Compared to Nivolumab Alone Second-line Tx in Participants With Metastatic Non-Small Cell Lung Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peginesatide Approved DB08894
biotech | CAS: 913976-27-9

Peginesatide is a synthetic peptide attached to polyethylene glycol for the treatment of anemia. The polyethylene glycol moiety helps make the drug less immunogenic and prolongs its plasma half-life. Chemically, peginesatide is designed to mimic the pharmacol…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntianemic Preparations +10
Target Protein:
Erythropoietin receptor
Waktu ParuhIV dose, healthy su…
Vol. DistribusiIV dose, dialysis p…
KlirensSystemic clearance,…
Genetik -
Peginterferon alfa-2a Approved DB00008
biotech | CAS: 198153-51-4

Peginterferon alfa-2a is a form of recombinant interferon used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Adjuvants, ImmunologicAlcoholsAlfa Interferons +29
Target Protein:
Interferon alpha/beta receptor 2Interferon alpha/beta receptor 1
Gen Terkait:
IFNL3
Waktu ParuhThe mean terminal h…
Vol. Distribusi-
KlirensThe mean systemic c…
Genetik 1 Varian
Peginterferon alfa-2b Approved DB00022
biotech | CAS: 215647-85-1

Peginterferon alfa-2b is a form of recombinant interferon used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Adjuvants, ImmunologicAlcoholsAlfa Interferons +34
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Gen Terkait:
IFNL3
Waktu ParuhThe mean half-life …
Vol. Distribusi-
KlirensThe estimated appar…
Genetik 1 Varian
Pegloticase Approved DB09208
biotech | CAS: 885051-90-1

Pegloticase is a porcine recombinant PEGylated uricase indicated for the treatment of chronic gout in adult patients that do not respond to other types of therapies.[L42425] Pegloticase has a similar activity to rasburicase, an enzyme that metabolizes uric ac…

Kategori:
Antigout PreparationsCompounds used in a research, industrial, or household settingEnzymes +6
Target Protein:
Uric acid
Waktu ParuhIn patients with sy…
Vol. DistribusiThe volume of distr…
KlirensIn gout patients gi…
Genetik -
Pegsitacianine DB19098
small molecule | CAS: 2396651-85-5

Pegsitacianine is under investigation in clinical trial NCT05576974 (A Phase 2a, Single-dose, Open-label Study to Evaluate Diagnostic Performance and Safety of Pegsitacianine, an Intraoperative Fluorescence Imaging Agent for the Detection of Cancer, in Patien…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegtarviliase DB18999
biotech | CAS: 2649372-23-4

Pegtarviliase is under investigation in clinical trial NCT05154890 (A Multiple Ascending Dose Study of ACN00177 (Pegtarviliase) in Subjects With CBS Deficiency).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegulicianine Approved DB18731
small molecule | CAS: 2230217-17-9

Pegulicianine is an optical imaging agent indicated for fluorescence imaging in patients with breast cancer. It is used following surgical resection of the primary tumor to detect areas of remaining cancer. Pegulicianine itself is a prodrug comprising three m…

Kategori:
Contrast MediaFluorescent Dyes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegunigalsidase alfa Approved DB14992
biotech | CAS: 1644392-61-9

Pegunigalsidase alfa (PRX-102) is a recombinant form of human ?-galactosidase-A indicated for long-term enzyme replacement therapy in patients with Fabry disease, a rare genetic disorder characterized by the deficiency of alpha-galactosidase A.[A259352,L46342…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Alpha-galactosidase AGlobotriaosylceramide
Waktu ParuhPegunigalsidase alf…
Vol. DistribusiIn enzyme replaceme…
KlirensPatients treated wi…
Genetik -
Pegvaliase Approved DB12839
biotech | CAS: 1585984-95-7

Pegvaliase is a recombinant phenylalanine ammonia lyase (PAL) enzyme derived from _Anabaena variabilis_ that converts phenylalanine to ammonia and _trans_-cinnamic acid [A33284]. Both the U.S. Food and Drug Administration and European Medicines Agency approve…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAmmonia-Lyases +7
Target Protein:
Phenylalanine-4-hydroxylase
Waktu ParuhFollowing once-dail…
Vol. DistribusiThe mean ± SD (rang…
KlirensAt steady state fol…
Genetik -
biotech | CAS: 1620390-06-8

Pegvorhyaluronidase alfa is under investigation in clinical trial NCT02241187 (Two Stage Study Of Single Dose PEGPH20 And Cetuximab In Patients With Pancreatic Adenocarcinoma Prior To Surgical Resection).

Kategori:
Carbon-Oxygen LyasesEnzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegzilarginase Approved DB14780
biotech | CAS: 1659310-95-8

Pegzilarginase is under investigation in clinical trial NCT02488044 (A Phase 1/2 Study of AEB1102 in Patients With Arginase I Deficiency).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelacarsen DB16284
biotech | CAS: 1637637-70-7

Pelacarsen is under investigation in clinical trial NCT03070782 (Phase 2 Study of ISIS 681257 (Akcea-apo(a)-lrx) in Participants With Hyperlipoproteinemia(a) and Cardiovascular Disease).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelcitoclax DB16285
small molecule | CAS: 1619923-36-2

Pelcitoclax is under investigation in clinical trial NCT04210037 (Study of Combination APG-1252 Plus Paclitaxel in Patients With Relapsed/refractory Small Cell Lung Cancer).

Kategori:
Amines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peldesine DB02568
small molecule | CAS: 133432-71-0

Peldesine is a potent inhibitor of human CCRF-CEM T-cell proliferation. It has undergone phase I trials for the treatment of Human Immunodeficiency Virus (HIV) infections.

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 SubstratesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelitrexol DB12757
small molecule | CAS: 446022-33-9

Pelitrexol has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Sulfur Compounds
Target Protein:
Trifunctional purine biosynthetic protein adenosine-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemetrexed Approved DB00642
small molecule | CAS: 137281-23-3

Pemetrexed is a chemotherapy drug that is manufactured and marketed by Eli Lilly and Company under the brand name Alimta. It is indicated for use in combination with cisplatin for the treatment of patients with malignant pleural mesothelioma whose disease is …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +19
Target Protein:
Thymidylate synthaseThymidylate synthaseBifunctional purine biosynthesis protein ATIC +2
Waktu ParuhThe elimination hal…
Vol. DistribusiPemetrexed has a st…
KlirensThe total systemic …
Genetik -
Pemigatinib Approved DB15102
small molecule | CAS: 1513857-77-6

Pemigatinib is a small molecule kinase inhibitor with antitumour activity. It works by inhibiting fibroblast growth factor receptors (FGFRs), which are receptor tyrosine kinases that activate signalling pathways in tumour cells.[A193719] FGFRs gained attentio…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +16
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhFollowing administr…
Vol. DistribusiThe apparent volume…
KlirensFollowing administr…
Genetik -
Pemivibart DB18720
biotech | CAS: 2858673-18-2

Pemivibart (Pemgarda) is a human IgG1 monoclonal antibody targeting the SARS-CoV-2 spike protein receptor binding domain.[L50326] It received emergency use authorization (EUA) from the FDA in March 2024 for pre-exposure prophylaxis (PrEP) of COVID-19 in certa…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalApproved Treatments for COVID-19 +4
Target Protein:
Spike glycoprotein
Waktu ParuhPemivibart has an e…
Vol. DistribusiFollowing the admin…
KlirensFollowing the admin…
Genetik -
biotech

Pemlimogene merolisbac is under investigation in clinical trial NCT03371381 (An Efficacy and Safety Study of JNJ-64041757, a Live Attenuated Listeria Monocytogenes Immunotherapy, in Combination With Nivolumab Versus Nivolumab Monotherapy in Participants With …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemtumomab DB18563
biotech

Pemtumomab is a murine monoclonal antibody radiolabeled with Yttrium-90. It targets the mucin 1 (MUC1) protein.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PEN-866 DB16186
small molecule | CAS: 1472614-83-7

PEN-866 is under investigation in clinical trial NCT03221400 (PEN-866 in Patients With Advanced Solid Malignancies).

Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penamecillin DB13739
small molecule | CAS: 983-85-7

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penciclovir Approved DB00299
small molecule | CAS: 39809-25-1

Penciclovir is a synthetic acyclic guanine derivative with antiviral activity used for the treatment of various herpes simplex virus (HSV) infections. Displaying low toxicity and good selectivity, penciclovir is a nucleoside analogue.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
Thymidine kinase, cytosolicDNA polymerase catalytic subunitThymidine kinase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Penclomedine DB12987
small molecule | CAS: 108030-77-9

Penclomedine has been used in trials studying the treatment of Lymphoma and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Antineoplastic AgentsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillamine Approved DB00859
small molecule | CAS: 52-67-5

Penicillamine is a pharmaceutical of the chelator class. The pharmaceutical form is D-penicillamine, as L-penicillamine is toxic (it inhibits the action of pyridoxine). It is an ?-amino acid metabolite of penicillin, although it has no antibiotic properties.

Kategori:
Agents Causing Muscle ToxicityAmino AcidsAmino Acids, Peptides, and Proteins +16
Target Protein:
Copper
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemia
Target Protein:
Regulatory protein BlaR1Beta-lactam-inducible penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium camemberti Approved DB10809
biotech

Penicillium camemberti is a fungus which can provoke allergic reactions. Penicillium camemberti extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Penicillium chrysogenum var. chrysogenum is a fungus which can provoke allergic reactions. Penicillium chrysogenum var. chrysogenum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium digitatum Approved DB11023
biotech

Penicillium digitatum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium expansum Approved DB10810
biotech

Penicillium expansum is a fungus which can provoke allergic reactions. Penicillium expansum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium glaucum Approved DB14171
biotech

Penicillium glaucum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium italicum Approved DB10811
biotech

Penicillium italicum is a fungus which can provoke allergic reactions. Penicillium italicum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium roqueforti Approved DB10812
biotech

Penicillium roqueforti is a fungus which can provoke allergic reactions. Penicillium roqueforti extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penimepicycline DB13264
small molecule | CAS: 4599-60-4

Penimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients [L2791]. In the classification of the active ingredients included on this li…

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaerythritol tetranitrate Approved DB06154
small molecule | CAS: 78-11-5

Pentaerythritol tetranitrate is the nitrate ester of pentaerythritol that possesses explosive properties. When mixed with a plasticizer, this chemical forms a plastic explosive. It is recognized by the FDA to be a coronary vasodilator in the treatment of hear…

Kategori:
AlcoholsAntianginal AgentsCarbohydrates +11
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit betaFree radicals
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensIn a pharmacokineti…
Genetik -
Pentafluoropropane Approved DB13117
small molecule | CAS: 460-73-1

Pentafluoropropane is under investigation in clinical trial NCT01673061 (Vapocoolant Spray for Numbing Small Boils Before Incision and Drainage).

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentagastrin Approved DB00183
small molecule | CAS: 5534-95-2

A synthetic pentapeptide that mimics the actions of endogenous gastrin when given parenterally. It works by stimulating the secretion of gastric acid, pepsin, and intrinsic factor. It has also been used as a diagnostic aid.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGastrins +8
Target Protein:
Gastrin/cholecystokinin type B receptor
Waktu Paruh10 minutes or less
Vol. Distribusi-
Klirens-
Genetik -
Pentamycin DB13571
small molecule | CAS: 6834-98-6

Deskripsi belum tersedia.

Kategori:
AlkenesAntifungal AgentsGenito Urinary System and Sex Hormones +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentastarch Approved DB09111
small molecule | CAS: 9005-27-0

Pentastarch is an artificial colloid (hydroxyethyl starch derivative). Pentastarch is characterized by presenting five hydroxyethyl groups, which signifies an approximate 50% hydroxyethylation. It is sold under the name Pentaspan by Bristol-Myers Squibb and i…

Kategori:
Blood SubstitutesCarbohydratesCompounds used in a research, industrial, or household setting +9
Waktu Paruh~2.5 hours.
Vol. Distribusi-
Klirens-
Genetik -
Pentazocine Approved DB00652
small molecule | CAS: 359-83-1

The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)

Kategori:
Adjuvants, AnesthesiaAgents that reduce seizure thresholdAlkaloids +20
Target Protein:
Sigma non-opioid intracellular receptor 1Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh2 to 3 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentetic acid Approved DB14007
small molecule | CAS: 67-43-6

Pentetic acid, also known as diethylenetriaminepentaacetic acid (DTPA), is a synthetic polyamino carboxylic acid with eight coordinate bond forming sites that can sequester metal ions and form highly stable DTPA-metal ion complexes. DTPA, along with its calci…

Kategori:
AcetatesAcids, AcyclicAmines +10
Target Protein:
Transuranium elements
Waktu ParuhIn preclinical stud…
Vol. DistribusiThe volume of distr…
KlirensPentetic acid prese…
Genetik -
Pentetrazol DB13415
small molecule | CAS: 54-95-5

Pentetrazol, also known as pentylenetetrazole, is a gamma-aminobutyric acid type A (GABA<sub>A</sub>) receptor antagonist that was approved by the FDA until 1982.[A254437]

Kategori:
AzepinesCentral Nervous System AgentsCentral Nervous System Stimulants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentobarbital Approved DB00312
small molecule | CAS: 76-74-4

A short-acting barbiturate that is effective as a sedative and hypnotic (but not as an anti-anxiety) agent and is usually given orally. It is prescribed more frequently for sleep induction than for sedation but, like similar agents, may lose its effectiveness…

Kategori:
Adjuvants, AnesthesiaAnticholinergic AgentsAnticonvulsants +23
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +10
Waktu Paruh5 to 50 hours (dose…
Vol. Distribusi-
Klirens-
Genetik -
Pentostatin Approved DB00552
small molecule | CAS: 53910-25-1

A potent inhibitor of adenosine deaminase. The drug is effective in the treatment of many lymphoproliferative malignancies, particularly hairy-cell leukemia. It is also synergistic with some other antineoplastic agents and has immunosuppressive activity.

Kategori:
Adenosine Deaminase InhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Adenosine deaminase
Waktu Paruh5.7 hours (with a r…
Vol. Distribusi-
Klirens* 68 mL/min/m2
Genetik -
Pentoxifylline Approved DB00806
small molecule | CAS: 6493-05-6

Pentoxifylline (PTX) is a synthetic dimethylxanthine derivative that modulates the rheological properties of blood and also has both anti-oxidant and anti-inflammatory properties.[A226415, L30300] Although originally developed to treat intermittent claudicati…

Kategori:
AlkaloidsAntioxidantsAntiplatelet agents +23
Target Protein:
Adenosine receptor A2aTumor necrosis factorPhosphodiesterase enzymes +2
Waktu ParuhOverall, pentoxifyl…
Vol. DistribusiPentoxifylline has …
KlirensPentoxifylline give…
Genetik -
Pentoxyverine Approved DB11186
small molecule | CAS: 77-23-6

Pentoxyverine, also referred to as carbetapentane, is a non-opioid central acting antitussive with antimuscarinic, anticonvulsant [A32717], and local anesthetic properties. It is an active ingredient in over-the-counter cough suppressants in combination with …

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +2
Target Protein:
Sigma non-opioid intracellular receptor 1Voltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated sodium channel alpha subunit +2
Waktu ParuhThe half-life is 2.…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Peppermint oil Approved DB11198
biotech | CAS: 8006-90-4

Extracted from the stem, leaves, and flowers of _Mentha piperita_ L. plant, peppermint oil (Mentha piperita) is a popular essential oil used in aromatherapy for both external and internal use. Mentha piperita is a hybrid of spearmint (Mentha spicata) and wate…

Kategori:
Alimentary Tract and MetabolismAngiospermsAntiemetics +31
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Pepsin Approved DB13198
biotech | CAS: 9001-75-6

Pepsin is a potent enzyme in gastric juice that digests proteins such as those in meat, eggs, seeds, and dairy products [L2358]. Studies on gastric digestion from 1820-1840 led to the discovery of pepsin as the substance which, in the presence of stomach a…

Kategori:
Alimentary Tract and MetabolismAspartic Acid EndopeptidasesAspartic Acid Proteases +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peracetic acid DB14556
small molecule | CAS: 79-21-0

A liquid that functions as a strong oxidizing agent. It has an acrid odor and is used as a disinfectant.

Kategori:
AcetatesAcids, AcyclicAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4901–4950 dari 6694
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