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11793

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11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 99 / 236
Everolimus Approved DB01590
small molecule | CAS: 159351-69-6

Everolimus is a derivative of Rapamycin (sirolimus), and works similarly to Rapamycin as an mTOR (mammalian target of rapamycin) inhibitor. It is currently used as an immunosuppressant to prevent rejection of organ transplants. In a similar fashion to other m…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +32
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh~30 hours.
Vol. DistribusiThe blood-to-plasma…
KlirensFollowing a 3 mg ra…
Genetik -
Evexomostat DB19140
small molecule | CAS: 2416263-67-5

Evexomostat is under investigation in clinical trial NCT05570253 (A Study of SDX-7320 in Combination With Eribulin for People With Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evinacumab Approved DB15354
biotech | CAS: 1446419-85-7

Evinacumab is a recombinant human IgG4 monoclonal antibody targeted against angiopoietin-like protein 3 (ANGPTL3) and the first drug of its kind. The ANGPTL family of proteins serve a number of physiologic functions - including involvement in the regulation o…

Kategori:
Amino Acids, Peptides, and ProteinsAngiopoietin-like 3 InhibitorAngiopoietin-like 3 Inhibitors +8
Target Protein:
Angiopoietin-related protein 3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Evocalcet DB12388
small molecule | CAS: 870964-67-3

Evocalcet has been used in trials studying the treatment of Hyperparathyroidism and Secondary Hyperparathyroidism.

Kategori:
Anti-Parathyroid AgentsCalcium HomeostasisSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evofosfamide DB06091
small molecule | CAS: 918633-87-1

TH-302 is a novel cancer therapeutic specifically activated under the low oxygen or "hypoxic" conditions typical of solid tumor cancer cells. TH-302 is a nitroimidazole-linked prodrug of a brominated derivative of an isophosphoramide mustard previously used i…

Kategori:
Hydrocarbons, HalogenatedImidazolesMustard Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evogliptin DB12625
small molecule | CAS: 1222102-29-5

Evogliptin has been used in trials studying the treatment and screening of Osteoporosis, Renal Impairment, Type 2 Diabetes Mellitus, Diabetes Mellitis Type 2, and Diabetes Mellitus, Type 2.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +4
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evolocumab Approved DB09303
biotech | CAS: 1256937-27-5

Evolocumab is a monoclonal antibody designed for the treatment of hyperlipidemia by Amgen. It is a subcutaneous injection approved by the FDA for individuals on maximum statin therapy who still require additional LDL-cholesterol lowering. It is approved for b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu Paruh-
Vol. Distribusi-
KlirensEvolocumab showed n…
Genetik -
EVT 201 DB05721
small molecule | CAS: 308239-86-3

EVT 201 is a novel partial positive allosteric modulator of the GABAA receptor complex which is being developed as a treatment for insomnia. It is being developed by Evotec Inc.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT 302 DB06057
small molecule

EVT 302 is an orally active, potent, highly selective and reversible inhibitor of MAO-B. It is in the development for smoking cessation, and potential for disease modification in Alzheimer's disease.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT-101 DB05956
small molecule | CAS: 1189088-41-2

Deskripsi belum tersedia.

Target Protein:
Glutamate receptor ionotropic, NMDA 2BRetinoic acid receptor RXR-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Holoclar (_ex vivo_ expanded autologous human corneal epithelial cells containing stem cells) is a stem cell therapy used to treat limbal stem cell deficiencies.[L48375]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exagamglogene autotemcel Approved DB15572
biotech

Sickle cell disease (SCD) is a genetic disorder characterized by the production of abnormal sickle-shaped red blood cells (called hemoglobin S, HbS) that initiate a pathophysiology resulting in severe pain, progressive multi-organ damage, and premature death.…

Kategori:
Autologous Cultured CellBlood and Blood Forming Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exaluren DB17631
small molecule | CAS: 1375073-93-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exametazime Approved DB11179
small molecule | CAS: 105613-48-7

Exametazime is a diagnostic radiopharmaceutical agent commonly used for the preparation of Tc99m Exametazime injection. It acts as a chelating agent for the radioisotope technetium-99m to form a cationic complex. It is used in the detection of altered regiona…

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exarafenib DB17582
small molecule | CAS: 2639957-39-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exbivirumab DB17747
biotech | CAS: 569658-80-6

Exbivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exebacase DB16161
biotech | CAS: 1404122-92-4

Exebacase is under investigation in clinical trial NCT03163446 (Safety, Efficacy and Pharmacokinetics of CF-301 vs. Placebo in Addition to Antibacterial Therapy for Treatment of S. Aureus Bacteremia).

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exemestane Approved DB00990
small molecule | CAS: 107868-30-4

Exemestane is an oral steroidal aromatase inhibitor used in the adjuvant treatment of hormonally-responsive (also called hormone-receptor-positive, estrogen-responsive) breast cancer in postmenopausal women. It irreversibly binds to the active site of the enz…

Kategori:
AndrostanesAndrostenesAntineoplastic Agents +14
Target Protein:
Aromatase
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
Exenatide Approved DB01276
biotech | CAS: 141758-74-9

Exenatide is a glucagon-like peptide-1 (GLP-1) analog[L42690]. It activates the GLP-1 receptor and increases insulin secretion, decreases glucagon secretion, and slows gastric emptying to improve glycemic control[L42690]. Exenatide was given FDA approval on A…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Obesity Agents +16
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh2.4 hours[Label]
Vol. Distribusi28.3L[Label].
Klirens9.1 L/hour[Label].
Genetik -
Exicorilant DB16162
small molecule | CAS: 1781244-77-6

Exicorilant is under investigation in clinical trial NCT03437941 (Study to Evaluate CORT125281 in Combination With Enzalutamide in Patients With Mcrpc).

Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exidavnemab DB19452
biotech | CAS: 2438229-02-6

Exidavnemab is under investigation in clinical trial NCT06671938 (Safety, Tolerability, and Pharmacokinetics of Exidavnemab in Patients With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exisulind DB06246
small molecule | CAS: 59973-80-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +10
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseGlutathione S-transferase PAldo-keto reductase family 1 member B1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exlinkibart DB17474
biotech | CAS: 2642171-64-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EXT608 DB18453
biotech

EXT608 is a long-acting PTH derivative under investigation for the treatment of hyperparathyroidism.[L48270]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2226647-27-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezatiostat DB05460
small molecule | CAS: 168682-53-9

Ezatiostat is investigated in clinical trials for treating myelodysplastic syndrome. This compound belongs to the peptides. These are compounds containing an amide derived from two or more amino carboxylic acid molecules (the same or different) by formation o…

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Glutathione S-transferase P
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezeprogind DB16954
small molecule | CAS: 615539-20-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezetimibe Approved DB00973
small molecule | CAS: 163222-33-1

Ezetimibe is a lipid-lowering compound that inhibits intestinal cholesterol and phytosterol absorption. The discovery and research of this drug began in the early 1990s, after the intravenous administration of radiolabelled ezetimibe in rats revealed that it …

Kategori:
Anticholesteremic AgentsAzetinesBCRP/ABCG2 Substrates +20
Target Protein:
NPC1-like intracellular cholesterol transporter 1Sterol O-acyltransferase 1Aminopeptidase N
Waktu ParuhBoth ezetimibe and …
Vol. DistribusiThe relative volume…
KlirensThere are no pharma…
Genetik -
Ezurpimtrostat DB16458
small molecule | CAS: 1914148-72-3

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
F-15599 DB16936
small molecule | CAS: 635323-95-4

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +3
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 78-96-6

Deskripsi belum tersedia.

Target Protein:
Glutamate mutase sigma subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
F6-734 DB17444
biotech

F6-734 is a bispecific monoclonal antibody with affinity for anticarcinoembryonic antigen (CEA) and anti-diethylenetriamine pentaacetic acid (DTPA) (hMN-14 × m734).[A255217,A255222]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fabomotizole DB13623
small molecule | CAS: 173352-21-1

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsNervous System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Facinicline DB05586
small molecule | CAS: 677306-35-3

Deskripsi belum tersedia.

Kategori:
Bridged-Ring CompoundsHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Factor IX Complex (Human) Approved DB11330
biotech | CAS: 37224-63-8

Factor IX Complex is a sterile, lyophilized concentrate composed of a number of Vitamin K-dependent clotting factors found in functioning human plasma. Also known as prothrombin complex concentrate, products containing this complex often include Factor IX (an…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Factor XIII (human) Approved DB12909
biotech | CAS: 9013-56-3

Factor XIII (human) is a heat-treated, lyophilized concentrate of coagulation factor XIII, an endogenous enzyme responsible for the crosslinking of fibrin and an essential component of the coagulation cascade [FDA Label]. For people with congenital deficiency…

Kategori:
AcyltransferasesAmino Acids, Peptides, and ProteinsAminoacyltransferases +14
Waktu Paruh6.6 ±2.29 days [FDA…
Vol. DistribusiVss = 51.1 mL/kg (v…
Klirens0.25 ±0.09 mL/hr/kg…
Genetik -
Fadrozole DB16832
small molecule | CAS: 102676-47-1

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalAromatase Inhibitors +7
Target Protein:
AromataseCytochrome P450 11B1, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fagrocorat DB14676
small molecule | CAS: 1044535-52-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Falimarev DB17333
biotech | CAS: 685563-14-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fallypride DB15167
small molecule | CAS: 166173-78-0

Fallypride is under investigation in clinical trial NCT02310360 (Striatal and Extra-striatal Dopamine Release in Response to Food in Healthy Humans).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fallypride F-18 DB19254
small molecule | CAS: 166173-82-6

Fallypride F-18 is under investigation in clinical trial NCT00846040 (Reduced Carbohydrate Versus Fat in Obese Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Falnidamol DB12966
small molecule | CAS: 196612-93-8

Falnidamol has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Famciclovir Approved DB00426
small molecule | CAS: 104227-87-4

Famciclovir, marketed as Famvir by Novartis, is a guanine analogue used to treat herpes virus infections. It is most commonly used to treat herpes zoster (shingles). Famciclovir is a prodrug of penciclovir with higher oral bioavailability.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh10 hours
Vol. Distribusi* 1.08±0.17 L/kg [h…
Klirens* 36.6 +/- 6.3 L/hr…
Genetik -
Famitinib DB11741
small molecule | CAS: 1044040-56-3

Famitinib has been used in trials studying the treatment of Colorectal Cancer, Renal Cell Cancer, Colorectal Cancer Recurrent, Colorectal Cancer Metastatic, and Metastatic Renal Cell Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-RingReceptor Protein-Tyrosine Kinases, antagonists & inhibitors
Target Protein:
Platelet-derived growth factor receptor alphaReceptor-type tyrosine-protein kinase FLT3Mast/stem cell growth factor receptor Kit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Famotidine Approved DB00927
small molecule | CAS: 76824-35-6

Famotidine is a competitive histamine-2 (H<sub>2</sub>) receptor antagonist that works to inhibit gastric acid secretion. It is commonly used in gastrointestinal conditions related to acid secretion, such as gastric ulcers and gastroesophageal reflux disease …

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +20
Target Protein:
Histamine H2 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensRenal clearance is …
Genetik -
Famprofazone DB16702
small molecule | CAS: 22881-35-2

Famprofazone is a nonsteroidal anti-inflammatory agent found in combination products such as ‘Gewodin’ which is marketed in Taiwan.[L34724] It is important to note that the drug is metabolized to [methamphetamine] and [amphetamine] in the body and can lead to…

Kategori:
AminesAmphetaminesAnalgesics +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fanapanel DB12393
small molecule | CAS: 161605-73-8

Fanapanel has been investigated for the treatment of Visual Acuity.

Kategori:
Heterocyclic Compounds, Fused-RingOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FAPi-46 GA-68 DB18827
small molecule | CAS: 2374784-98-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Farampator DB15012
small molecule | CAS: 211735-76-1

Farampator is under investigation in clinical trial NCT00113022 (Org 24448 to Treat Major Depression).

Kategori:
Oxazoles
Target Protein:
Glutamate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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