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12560

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Halaman 97 / 252
Dolcanatide DB13112
biotech | CAS: 1092457-65-2

Dolcanatide has been investigated in Exposure.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme ActivatorsGastrointestinal Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Dolichovespula arenaria venom protein is an extract of Dolichovespula arenaria venom. Dolichovespula arenaria venom protein is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Dolichovespula maculata venom protein is an extract of Dolichovespula maculata venom. Dolichovespula maculata venom protein is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dolutegravir Approved DB08930
small molecule | CAS: 1051375-16-6

Dolutegravir is an HIV-1 integrase inhibitor that blocks the strand transfer step of the integration of the viral genome into the host cell (INSTI).[A7514] The effect of this drug has no homology in human host cells, which gives it excellent tolerability and …

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinIntegrase
Gen Terkait:
UGT1A1 UGT1A1 UGT1A1
Waktu ParuhThe half-life of do…
Vol. DistribusiThe administration …
KlirensThe apparent cleara…
Genetik 3 Varian
Domagrozumab DB15083
biotech | CAS: 1629605-31-7

Domagrozumab is under investigation in clinical trial NCT01616277 (A Phase 1 Study To Evaluate The Safety And Tolerability Of PF-06252616 In Healthy Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domatinostat DB17521
small molecule | CAS: 910462-43-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domiphen Approved DB11594
small molecule | CAS: 13900-14-6

Domiphen bromide is a quaternary ammonium compound that is predominantly employed as a topically administered antiseptic agent.

Kategori:
Alimentary Tract and MetabolismAminesAmmonium Compounds +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2382896-04-8

Domofenogene zalfaparvovec, formerly known as BMN-307, is an investigational AAV5-phenylalanine hydroxylase (PAH) gene therapy developed by BioMarin Pharmaceutical.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domoic Acid DB02852
small molecule | CAS: 14277-97-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsNeuromuscular AgentsNeurotoxins +2
Target Protein:
Glutamate receptor ionotropic, kainate 1Glutamate receptor ionotropic, kainate 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domperidone Approved DB01184
small molecule | CAS: 57808-66-9

A specific blocker of dopamine receptors. It speeds gastrointestinal peristalsis, causes prolactin release, and is used as antiemetic and tool in the study of dopaminergic mechanisms.

Kategori:
Alimentary Tract and MetabolismAntiemeticsAutonomic Agents +25
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
Waktu Paruh7 hours
Vol. Distribusi-
Klirens-
Genetik -
Domvanalimab DB18848
biotech | CAS: 2368219-35-4

Domvanalimab is under investigation in clinical trial NCT05502237 (Zimberelimab and Domvanalimab in Combination With Chemotherapy Versus Pembrolizumab With Chemotherapy in Patients With Untreated Metastatic Non-small Cell Lung Cancer).

Waktu Paruh-
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Genetik -
Donanemab Approved DB16647
biotech | CAS: 1931944-80-7

Donanemab is a humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against insoluble N-truncated pyroglutamate amyloid beta (A?), [L50978] which is found in the brain amyloid plaques that contribute to the pathophysiology of Alzheimer's Disea…

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAmyloid Beta-directed Antibodies +11
Target Protein:
Beta amyloid plaque
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe central volume …
KlirensThe clearance is ab…
Genetik -
Donepezil Approved DB00843
small molecule | CAS: 120014-06-4

In 2016, the global burden of dementia was estimated to be 43.8 million, demonstrating a significant increase from a global prevalence of 20.2 million in 1990.[A182411] Donepezil, also known as Aricept, is a piperidine derivative acetylcholinesterase inhibito…

Kategori:
Anti-Dementia DrugsBCRP/ABCG2 SubstratesBradycardia-Causing Agents +20
Target Protein:
Acetylcholinesterase5-hydroxytryptamine receptor 2ACholinesterase +5
Gen Terkait:
CYP2D6
Waktu ParuhThe average elimina…
Vol. DistribusiThe volume of distr…
KlirensAccording to the FD…
Genetik 1 Varian
Donidalorsen DB18751
biotech | CAS: 2304692-48-4

Donidalorsen is under investigation in clinical trial NCT05392114 to assess the long-term safety and efficacy of donidalorsen in the prophylactic treatment of hereditary angioedema (HAE)

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Donislecel Approved DB17961
biotech

Donislecel is the first allogeneic pancreatic islet cellular from deceased donor pancreatic cells used for the treatment of adult type 1 diabetes with unsuccessful control of glycated hemoglobin, despite intensive diabetes management and treatments.[L47166,L4…

Kategori:
Cellular and Gene TherapyDrugs Used in Diabetes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DONU DB12968
small molecule | CAS: 58484-17-6

Donu has been used in trials studying the treatment of Psychosis.

Kategori:
AmidesNitroso Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dopamine Approved DB00988
small molecule | CAS: 51-61-6

One of the catecholamine neurotransmitters in the brain. It is derived from tyrosine and is the precursor to norepinephrine and epinephrine. Dopamine is a major transmitter in the extrapyramidal system of the brain, and important in regulating movement. A fa…

Kategori:
Adrenergic and Dopaminergic AgentsAgents producing tachycardiaAgents that produce hypertension +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor +13
Waktu Paruh2 minutes
Vol. Distribusi-
Klirens-
Genetik -
Dopastatin DB16144
small molecule | CAS: 868562-36-1

Dopastatin is under investigation in clinical trial NCT04335357 (TBR-760 in Adult Patients With Non-functioning Pituitary Adenomas).

Kategori:
AminesAmino Acids, Peptides, and ProteinsBenzene Derivatives +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doramapimod DB03044
small molecule | CAS: 285983-48-4

Doramapimod is a P38 MAP kinase inhibitor.

Kategori:
AmidesBenzene DerivativesProtein Kinase Inhibitors
Target Protein:
Tyrosine-protein kinase HCKMitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doramectin DB11400
small molecule | CAS: 117704-25-3

Doramectin is a veterinary drug approved by the Food and Drug Administration for the treatment of parasites such as gastrointestinal roundworms, lungworms, eyeworms, grubs, sucking lice and mange mites in cattle.

Kategori:
AgrochemicalsAnthelminticsAnti-Anxiety Agents +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doravirine Approved DB12301
small molecule | CAS: 1338225-97-0

Doravirine is an HIV-1 non-nucleoside reverse transcriptase inhibitor (NNRTI) intended to be administered in combination with other antiretroviral medicines.[L12729,L4562] Doravirine is available by itself or as a combination product of doravirine (100 mg), l…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +10
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensThe oral and renal …
Genetik -
Dordaviprone DB14844
small molecule | CAS: 1616632-77-9

Dordaviprone (ONC-201) is under investigation in clinical trial NCT03394027 (ONC201 in Recurrent/Refractory Metastatic Breast Cancer and Advanced Endometrial Carcinoma).

Kategori:
Antineoplastic Agents
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dornase alfa Approved DB00003
biotech | CAS: 143831-71-4

Dornase alfa is a biosynthetic form of human deoxyribunuclease I (DNase I) enzyme. It is produced in genetically modified Chinese hamster ovary (CHO) cells using recombinant DNA technology. The 260-amino acid sequence of dornase alfa is identical to the endog…

Kategori:
Amino Acids, Peptides, and ProteinsCough and Cold PreparationsDecreased Respiratory Secretion Viscosity +10
Target Protein:
Deoxyribonuclease-1
Waktu Paruh-
Vol. DistribusiIn studies in rats …
KlirensStudies in rats ind…
Genetik -
Dorsomorphin DB08597
small molecule | CAS: 866405-64-3

Deskripsi belum tersedia.

Kategori:
AMP-Activated Protein Kinases, antagonists & inhibitorsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
5'-AMP-activated protein kinase catalytic subunit alpha-15'-AMP-activated protein kinase subunit beta-15'-AMP-activated protein kinase subunit gamma-1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dorzagliatin DB15123
small molecule | CAS: 1191995-00-2

Dorzagliatin is under investigation in clinical trial NCT03173391 (Long-term Efficacy and Safety of HMS5552 in T2DM).

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes
Target Protein:
Hexokinase-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dorzolamide Approved DB00869
small molecule | CAS: 120279-96-1

Dorzolamide is a non-bacteriostatic sulfonamide derivative [A1304] and topical carbonic anhydrase (CA) inhibitor that treats elevated intraocular pressure (IOP) associated with open-angle glaucoma and ocular hypertension.[L11377] It works by blocking an enzym…

Kategori:
AmidesAntiglaucoma Preparations and MioticsAntihypertensive Agents +16
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 4Carbonic anhydrase 1 +1
Waktu ParuhAs the drug adminis…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
Dostarlimab Approved DB15627
biotech | CAS: 2022215-59-2

Dostarlimab is an IgG<sub>4</sub> humanized monoclonal antibody targeted against the human programmed death receptor-1 (PD-1).[L33320] PD-1 receptors are found on T-cells and, when activated, serve to inhibit immune responses - some cancers leverage this syst…

Kategori:
Amino Acids, Peptides, and ProteinsAnionsAntibodies +21
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAt steady-state, th…
KlirensAt steady-state, th…
Genetik -
Dosulepin Approved DB09167
small molecule | CAS: 113-53-1

Dosulepin (INN, BAN) formerly known as dothiepin (USAN), is a tricyclic antidepressant with anxiolytic properties that is used in several European and South Asian countries, as well as Australia, South Africa, and New Zealand. It is not FDA-approved due to lo…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +45
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2AHistamine H1 receptor +9
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent V…
KlirensOral clearance is a…
Genetik -
small molecule | CAS: 2230254-48-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dotarizine DB06446
small molecule | CAS: 84625-59-2

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntidepressive Agents +14
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1AVoltage-dependent P/Q-type calcium channel subunit alpha-1A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dotatate Approved DB14554
small molecule | CAS: 177943-88-3

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic Agent
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dotatate gallium Ga-68 Approved DB13925
small molecule | CAS: 1027785-90-5

Dotatate gallium (Ga-68) is a somatostatin-2 receptor analog which is radiolabeled with gallium 68 as a positron-emitting radioisotope. Ga-68 dotatate has a high affinity for somatostatin-2 receptor and it is rapidly excreted from the nontarget sites which gi…

Kategori:
Amino Acids, Peptides, and ProteinsGallium RadioisotopesPeptides +3
Target Protein:
Somatostatin receptor type 2
Waktu ParuhThe half-life of ga…
Vol. DistribusiThe volume of distr…
KlirensThe pharmacokinetic…
Genetik -
Dotinurad DB16145
small molecule | CAS: 1285572-51-1

Dotinurad is under investigation in clinical trial NCT03372200 (Febuxostat-controlled, Double-blind, Comparative Study of FYU-981 in Hyperuricemia With or Without Gout).

Kategori:
Antigout PreparationsAntirheumatic AgentsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Solute carrier family 22 member 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DOTMP HO-166 DB05380
small molecule | CAS: 633308-23-3

DOTMP HO-166 is used in skeletal targeted radiotherapy (STR). SRT is designed to be used in combination with high-dose chemotherapy producing a direct therapeutic effect on the tumor sites in the bone plus a general bone-marrow effect to destroy myeloma cells…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DOTMP SM-153 DB18484
small molecule | CAS: 633308-21-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dovitinib DB05928
small molecule | CAS: 405169-16-6

Dovitinib is an orally active small molecule that exhibits potent inhibitory activity against multiple RTKs involved in tumor growth and angiogenesis. Preclinical data show that dovitinib works to inhibit multiple kinases associated with different cancers, in…

Kategori:
BCRP/ABCG2 InducersBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +17
Target Protein:
Nuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dovramilast DB16242
small molecule | CAS: 340019-69-4

Dovramilast is under investigation in clinical trial NCT01300208 (To Evaluate the Preliminary Safety, Tolerability, Pharmacokinetics, Pharmacodynamics and Efficacy of CC-11050 in Subjects With Discoid Lupus Erythematosus and Subacute Cutaneous Lupus Erythemat…

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doxacurium Approved DB01135
small molecule | CAS: 106791-39-3

Doxacurium chloride is a long-acting, nondepolarizing skeletal muscle relaxant for intravenous administration.

Kategori:
Anticholinergic AgentsCentral Nervous System DepressantsCholinesterase substrates +11
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2
Waktu Paruh99 minutes in norma…
Vol. Distribusi* 0.11-0.43 L/kg [H…
Klirens* 2.66 mL/min/kg [H…
Genetik -
Doxapram Approved DB00561
small molecule | CAS: 309-29-5

A central respiratory stimulant with a brief duration of action. (From Martindale, The Extra Pharmocopoeia, 30th ed, p1225)

Kategori:
Agents that produce hypertensionCentral Nervous System AgentsCentral Nervous System Stimulants +4
Target Protein:
Potassium channel subfamily K member 3Potassium channel subfamily K member 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doxazosin Approved DB00590
small molecule | CAS: 74191-85-8

Doxazosin is an alpha-1 antagonist used for the treatment of benign prostatic hypertrophy (BPH) symptoms and hypertension. Other members of this drug class include [Prazosin], [Terazosin], [Tamsulosin], and [Alfuzosin].[A180661] Because of its long-lasting e…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorHERG human cardiac K+ channel +1
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of do…
Genetik -
Doxefazepam DB13837
small molecule | CAS: 40762-15-0

Deskripsi belum tersedia.

Kategori:
BenzazepinesBenzodiazepines and benzodiazepine derivativesBenzodiazepinones +5
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doxepin Approved DB01142
small molecule | CAS: 1668-19-5

Doxepin is a psychotropic agent with antidepressant and anxiolytic properties.[T559] It is a tertiary amine that can be presented as (E) and (Z) stereoisomers with the (Z) stereoisomer corresponding to [cidoxepin]. Doxepin commonly produces a 5:1 (E):(Z) race…

Kategori:
Acid ReducersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +55
Target Protein:
Histamine H1 receptorHistamine H2 receptorSodium-dependent noradrenaline transporter +16
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +5
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean apparent v…
KlirensThe mean total appa…
Genetik 8 Varian
Doxercalciferol Approved DB06410
small molecule | CAS: 54573-75-0

Doxercalciferol is a synthetic vitamin D2 analog that undergoes metabolic activation in vivo to form 1?,25-dihydroxyvitamin D2 (1?,25-(OH)2D2), a naturally occurring, biologically active form of vitamin D2. Doxercalciferol is indicated for the treatment of se…

Kategori:
Anti-Parathyroid AgentsBone Density Conservation AgentsCalcium Homeostasis +16
Target Protein:
Vitamin D3 receptor
Waktu Paruh32 to 37 hours.
Vol. Distribusi-
Klirens-
Genetik -
Doxifluridine DB12947
small molecule | CAS: 3094-09-5

Doxifluridine has been investigated for the treatment of Stomach Cancer.

Kategori:
AntimetabolitesAntineoplastic AgentsAppetite Stimulants +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doxofylline DB09273
small molecule | CAS: 69975-86-6

Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown similar efficacy to theophylline but with significantly fewer side effects in animal and human st…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +21
Target Protein:
Beta-2 adrenergic receptorcGMP-dependent 3',5'-cyclic phosphodiesteraseAdenosine receptor A2a
Waktu ParuhFollowing administr…
Vol. DistribusiDoxofylline demonst…
KlirensFollowing oral admi…
Genetik -
Doxorubicin Approved DB00997
small molecule | CAS: 23214-92-8

Doxorubicin is a cytotoxic anthracycline antibiotic isolated from cultures of Streptomyces peucetius var. caesius along side with daunorubicin, another cytotoxic agent, in 1970.[A1575,A257709,A257614] Although they both have aglyconic and sugar moieties, doxo…

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +36
Target Protein:
DNA topoisomerase 2-alphaTelomerase reverse transcriptaseDNA +3
Gen Terkait:
RARG SLC28A3 UGT1A6
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state di…
KlirensThe plasma clearanc…
Genetik 3 Varian
Doxycycline Approved DB00254
small molecule | CAS: 564-25-0

Doxycycline is a broad-spectrum antibiotic synthetically derived from [oxytetracycline].[L42880] It is a second-generation tetracycline that was first discovered in 1967.[A19429] Second-generation tetracyclines exhibit lesser toxicity than first-generation te…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAnti-Bacterial Agents +17
Target Protein:
30S ribosomal protein
Waktu ParuhThere is limited in…
Vol. DistribusiThere is limited in…
KlirensPopulation pharmaco…
Genetik -
DP-b99 DB05820
small molecule

DP-b99 is a newly developed lipophilic, cell permeable derivative of BAPTA (1,2-bis(2-aminophenoxy)ethane-N,N,N',N'-tetraacetic acid), that is under development as a neuroprotectant for the potential treatment of stroke, head trauma and neurological damage as…

Kategori:
AcetatesAcids, AcyclicAmines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DP-VPA DB05821
small molecule

DP-VPA is D-Pharm's proprietary lipid modified version of valproic acid (VPA) that demonstrate that DP-VPA is well-tolerated in patients with resistant epilepsy and has a marked effect on reducing seizure frequency.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DPA-714 F-18 DB19189
small molecule | CAS: 958233-09-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4801–4850 dari 12560
Sebelumnya Halaman 97 / 252 Berikutnya