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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 96 / 134
Orotidylic acid DB02957
small molecule | CAS: 2149-82-8

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orthosiphon aristatus leaf Approved DB15838
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osanetant DB04872
small molecule | CAS: 160492-56-8

Developed by Sanofi-Aventis (formerly Sanofi-Synthelabo), osanetant (SR-142801) is an NK3 receptor antagonist which was under development for the treatment of schizophrenia and other Central Nervous System (CNS) disorders. In a review of its R&D portfolio, th…

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Neuromedin-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osbond acid DB14088
small molecule | CAS: 25182-74-5

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSE-2101 DB17122
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oseltamivir Approved DB00198
small molecule | CAS: 196618-13-0

Oseltamivir (marketed as the product Tamiflu?), is an antiviral neuraminidase inhibitor used for the treatment and prophylaxis of infection with influenza viruses A (including pandemic H1N1) and B. Oseltamivir exerts its antiviral activity by inhibiting the a…

Kategori:
AcetamidesAcetatesAmides +8
Target Protein:
NeuraminidaseSialidase-1Sialidase-2
Waktu ParuhPlasma concentratio…
Vol. DistribusiThe mean volume of …
KlirensRenal clearance (18…
Genetik -
small molecule | CAS: 187227-45-8

Deskripsi belum tersedia.

Kategori:
AcetamidesAcetatesAcids, Acyclic +8
Target Protein:
Neuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-027 DB12387
small molecule | CAS: 936890-98-1

OSI-027 has been used in trials studying the treatment of Any Solid Tumor or Lymphoma.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-7836 DB05837
small molecule

OSI-7836 is a member of the nucleoside class of cytotoxic drugs of which gemcitabine is the market leader. OSI Pharmaceuticals develops OSI-7836 as a next-generation gemcitabine. The anti-tumor activity of OSI-7836 appeares to be less schedule dependent than …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-7904L DB05457
small molecule

OSI-7904L is a liposome encapsulated thymidylate synthase inhibitor, which is indicated for use in advanced gastric and/or gastroesophageal adenocarcinoma (A-G/GEJA). Current treatments also inhibit thymidylate synthase but the innovative lipid coating of OSI…

Kategori:
Acids, AcyclicDicarboxylic AcidsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osilodrostat Approved DB11837
small molecule | CAS: 928134-65-0

Osilodrostat is an inhibitor of 11?-hydroxylase (also referred to as CYP11B1), the enzyme that catalyzes the final step in the biosynthesis of endogenous cortisol.[L12123] It is used to lower circulating cortisol levels in the treatment of Cushing's disease, …

Kategori:
Antiadrenal PreparationsAnticorticosteroidsCortisol Synthesis Inhibitors +32
Target Protein:
Cytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial
Waktu ParuhThe elimination hal…
Vol. DistribusiThe median apparent…
KlirensData regarding the …
Genetik -
Osimertinib Approved DB09330
small molecule | CAS: 1421373-65-0

Osimertinib is an oral, third-generation epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) drug developed by AstraZeneca Pharmaceuticals.[A7926,L43453] Its use is indicated for the treatment of metastatic non-small cell lung cancer (NSCL…

Kategori:
Acids, AcyclicAcrylatesAmides +29
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe population esti…
Vol. DistribusiThe mean volume of …
KlirensOral clearance is 1…
Genetik -
Osocimab DB14818
biotech | CAS: 2056878-75-0

Osocimab is under investigation in clinical trial NCT03276143 (Factor XIa inhibition for the prevention of venous Thromboembolism in Patients Undergoing Total Knee Arthroplasty).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osugacestat DB12006
small molecule | CAS: 1401066-79-2

Osugacestat (BMS-906024) has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OT-730 DB16112
small molecule | CAS: 870809-51-1

OT-730 is under investigation in clinical trial NCT00753168 (Phase 1-2 Evaluation of OT-730 Eye Drops in Reducing the Intraocular Pressure in Patients With Ocular Hypertension or Open-angle Glaucoma).

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otelixizumab DB05496
biotech | CAS: 881191-44-2

Otelixizumab is a monoclonal antibody that binds to a receptor found on all T cells called CD3, which is involved in normal T cell signaling. Otelixizumab is believed to inhibit the function of autoreactive T cells, which are important in propagating autoimmu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oteracil Approved DB03209
small molecule | CAS: 937-13-3

Oteracil is an adjunct to antineoplastic therapy, used to reduce the toxic side effects associated with chemotherapy. Approved by the European Medicines Agency (EMA) in March 2011, Oteracil is available in combination with [DB09257] and [DB09256] within the c…

Kategori:
Triazines
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Oteseconazole Approved DB13055
small molecule | CAS: 1340593-59-0

Oteseconazole is an azole metalloenzyme inhibitor that targets fungal CYP51.[L41635] CYP51, also known as 14? demethylase, participates in the formation of ergosterol, a compound that plays a vital role in the integrity of cell membranes.[L41635,A247020] By b…

Kategori:
14-alpha Demethylase InhibitorsAntifungal AgentsAntiinfectives for Systemic Use +5
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe median terminal…
Vol. DistribusiOn average, the vol…
KlirensClinical phase I st…
Genetik -
OTOF-GT DB18129
biotech

OTOF-GT is a dual vector AAV gene therapy being investigated for the restoration of hearing loss associated with otoferlin deficiency.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OTX-2002 DB17246
biotech

OTX-2002 is a bicistronic messenger ribonucleic acid (mRNA) encoding for ZF-DNMT and ZF-KRAB proteins, encapsulated in a lipid nanoparticle (LNP).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ovalicin DB04324
small molecule

Deskripsi belum tersedia.

Kategori:
Terpenes
Target Protein:
Methionine aminopeptidase 1Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ovatodiolide DB19264
small molecule | CAS: 3484-37-5

Ovatodiolide is under investigation in clinical trial NCT04220411 (A Study for AR100DP1 in Mild to Moderate Atopic Dermatitis (AD)).

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ovemotide DB19156
biotech | CAS: 181477-91-8

Ovemotide is under investigation in clinical trial NCT00357461 (Ipilimumab With or Without Vaccine Therapy in Treating Patients With Previously Treated Stage IV Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1254-35-9

Oxabolone cipionate is the C17? cypionate ester and a prodrug of [DB01500]. A synthetic anabolic-androgenic (AAS) steroid, it is a derivative of 19-nortestosterone (nandrolone). It is considered as a performance enhancing drug thus is prohibited from use in s…

Kategori:
Alimentary Tract and MetabolismAnabolic Agents for Systemic UseAnabolic Steroids +11
Waktu Paruh-
Vol. Distribusi-
KlirensThe elimination on …
Genetik -
Oxacillin Approved DB00713
small molecule | CAS: 66-79-5

An antibiotic similar to [flucloxacillin] used in resistant staphylococci infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1A +7
Waktu Paruh20 to 30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Oxalic Acid DB03902
small molecule | CAS: 144-62-7

A strong dicarboxylic acid occurring in many plants and vegetables. It is produced in the body by metabolism of glyoxylic acid or ascorbic acid. It is not metabolized but excreted in the urine. It is used as an analytical reagent and general reducing agent. […

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingDicarboxylic Acids +6
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxaliplatin Approved DB00526
small molecule | CAS: 61825-94-3

Oxaliplatin is a platinum-based chemotherapy drug in the same family as cisplatin and carboplatin. Compared to cisplatin the two amine groups are replaced by diamino cyclohexane (DACH) group to provide a greater antitumor effect.[A797] However, this leads to …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +9
Target Protein:
DNA
Waktu ParuhThe decline of ultr…
Vol. DistribusiAfter a single 2-ho…
KlirensPlatinum was cleare…
Genetik -
small molecule | CAS: 328-42-7

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsKeto Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxametacin DB13308
small molecule | CAS: 27035-30-9

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAntiinflammatory and Antirheumatic ProductsAntiinflammatory and Antirheumatic Products, Non-Steroids +1
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxamic Acid DB03940
small molecule | CAS: 471-47-6

Amino-substituted glyoxylic acid derivative. [PubChem]

Kategori:
Acids, AldehydicAmino AcidsAmino Acids, Peptides, and Proteins +1
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialL-lactate dehydrogenaseL-lactate dehydrogenase +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxamniquine Approved DB01096
small molecule | CAS: 21738-42-1

An anthelmintic with schistosomicidal activity against Schistosoma mansoni, but not against other Schistosoma spp. Oxamniquine causes worms to shift from the mesenteric veins to the liver where the male worms are retained; the female worms return to the mesen…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +15
Target Protein:
DNA
Waktu Paruh1-2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Oxaprozin Approved DB00991
small molecule | CAS: 21256-18-8

Oxaprozin is a non-narcotic, non-steroidal anti-inflammatory drug (NSAID), used to relieve the inflammation, swelling, stiffness, and joint pain associated with osteoarthritis and rheumatoid arthritis.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +22
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh54.9 hours
Vol. Distribusi* 11 to 17 L/70 kg
Klirens-
Genetik -
Oxazepam Approved DB00842
small molecule | CAS: 604-75-1

Oxazepam is an intermediate-acting, 3-hydroxybenzodiazepine used in the treatment of alcohol withdrawal and anxiety disorders. Oxazepam, like related 3-hydroxybenzodiazepine [lorazepam], is considered less susceptible to pharmacokinetic variability based on p…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +16
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
OXB-301 DB19269
biotech

OXB-301 is under investigation in clinical trial NCT00397345 (Trovax Renal Immunotherapy Survival Trial).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxeladin Approved DB04822
small molecule | CAS: 468-61-1

Withdrawn from the Canadian, US, and UK markets in 1976 due to carcinogenicity.

Kategori:
Acids, CarbocyclicAntitussive AgentsCentral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxerutins DB15826
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxetacaine Approved DB12532
small molecule | CAS: 126-27-2

Oxetacaine, also called oxethazaince, is a potent surface analgesic with the molecular formula N, N-bis-(N-methyl-N-phenyl-t-butyl-acetamide)-beta-hydroxyethylamine that conserves its unionized form at low pH levels. Its actions have shown to relieve dysphagi…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAnestheticsAnesthetics, Local +5
Target Protein:
Gastrin
Waktu ParuhOxetacaine presents…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Oxfendazole DB11446
small molecule | CAS: 53716-50-0

Oxfendazole is a sulfoxide metabolite of fenbendazole. This benzimidazole antihelminthic protects livestock from roundworm. strongyles, and pinworn.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxfenicine DB04291
small molecule | CAS: 32462-30-9

Oxfenicine in an inhibitor of myocardial metabolism of nonesterified fatty acids (NEFA).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCarnitine O-Palmitoyltransferase, antagonists & inhibitors +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OXI-4503 DB05143
small molecule | CAS: 288847-35-8

OXI-4503 is investigated in clinical trials for treating cancer/tumors. OXI-4503 is a solid. OXI-4503 blocks and destroys tumor vasculature, resulting in extensive tumor cell death and necrosis. OXI-4503 (combretastatin A1 di-phosphate / CA1P) is a unique and…

Kategori:
AcidsAcids, NoncarboxylicAnions +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxibendazole DB04910
small molecule | CAS: 20559-55-1

Oxibendazole is a polymerase inhibitor in phase III trials for the treatment of helminth intestinal infections.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +1
Target Protein:
Tubulin beta-4B chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxidronic acid Approved DB14159
small molecule | CAS: 15468-10-7

Deskripsi belum tersedia.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxitriptan Approved DB02959
small molecule | CAS: 4350-09-8

5-Hydroxytryptophan (5-HTP), also known as oxitriptan (INN), is a naturally occurring amino acid and metabolic intermediate in the synthesis of serotonin and melatonin. 5-HTP is sold over-the-counter in the United Kingdom, United States and Canada as a dietar…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +8
Target Protein:
Tryptophan--tRNA ligase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxogluric acid DB08845
small molecule | CAS: 328-50-7

Oxogluric acid (?-Ketoglutarate) is not approved for any indication in the world but is an investigational drug in the United States. In the United States a phase I clinical trial is investigating whether oxogluric acid precursors found in nutritional supplem…

Kategori:
Acids, AcyclicDicarboxylic AcidsGlutarates +2
Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxolinic acid DB13627
small molecule | CAS: 14698-29-4

Deskripsi belum tersedia.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 19771-63-2

Procysteine has been used in trials studying the treatment of HIV Infections.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Cyclic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxybuprocaine Approved DB00892
small molecule | CAS: 99-43-4

Oxybuprocaine (also known as Benoxinate) is a local anesthetic, which is used especially in ophthalmology and otolaryngology. Oxybuprocaine binds to sodium channels and reversibly stabilizes the neuronal membrane which decreases its permeability to sodium ion…

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +15
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxybutynin Approved DB01062
small molecule | CAS: 5633-20-5

Overactive bladder (OAB) is a common condition negatively impacting the lives of millions of patients worldwide. Due to its urinary symptoms that include nocturia, urgency, and frequency, this condition causes social embarrassment and a poor quality of life.…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAnticholinergic Agents +23
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1
Waktu ParuhThe plasma eliminat…
Vol. DistribusiOxybutynin has a wi…
Klirens-
Genetik -
Oxycinchophen DB13596
small molecule | CAS: 485-89-2

Deskripsi belum tersedia.

Kategori:
Antiinflammatory and Antirheumatic ProductsMusculo-Skeletal SystemQuinolines +1
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxymetazoline Approved DB00935
small molecule | CAS: 1491-59-4

Oxymetazoline is an imidazole derivative and a potent, direct-acting alpha (?)-adrenergic agonist with affinity to both ?<sub>1</sub>- and ?<sub>2</sub>-adrenoceptors.[A215542] Oxymetazoline is available in various formulations with a wide variety of clinical…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +25
Target Protein:
Alpha-1A adrenergic receptorAlpha-2A adrenergic receptorAlpha-2B adrenergic receptor +7
Waktu ParuhFollowing ocular ad…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
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