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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 96 / 252
Dipotassium phosphate Approved DB09414
small molecule | CAS: 7758-11-4

Dipotassium phosphate (K2HPO4) is a highly water-soluble salt often used as a fertilizer and food additive as a source of phosphorus and potassium as well as a buffering agent.

Kategori:
AcidsAcids, NoncarboxylicAnions +14
Waktu ParuhIn healthy children…
Vol. DistribusiDistribution is lar…
KlirensPhosphates are rapi…
Genetik -
Dipraglurant DB12733
small molecule | CAS: 872363-17-2

Dipraglurant has been used in trials studying the treatment of Parkinson's Disease. It is a metabotropic glutamate receptor 5 (mGluR5) negative allosteric modulator (NAM).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diprenorphine DB01548
small molecule | CAS: 14357-78-9

A narcotic antagonist similar in action to naloxone. It is used to remobilize animals after etorphine neuroleptanalgesia and is considered a specific antagonist to etorphine. [PubChem]

Kategori:
AlkaloidsCentral Nervous System AgentsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 63065-88-3

Dipropyl-4-hydroxytryptamine is the 4-hydroxyl analog of dipropyltryptamine (DPT). Dipropyl-4-hydroxytryptamine was first synthesized by Alexander Shulgin. This agent and its properties haven't been fully elucidated.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25265-71-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipyridamole Approved DB00975
small molecule | CAS: 58-32-2

A phosphodiesterase inhibitor that blocks uptake and metabolism of adenosine by erythrocytes and vascular endothelial cells. Dipyridamole also potentiates the antiaggregating action of prostacyclin. (From AMA Drug Evaluations Annual, 1994, p752)

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +17
Target Protein:
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10AcGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4A +3
Waktu Paruh40 minutes
Vol. Distribusi* 1 to 2.5 L/kg
Klirens* 2.3-3.5 mL/min/kg
Genetik -
Dipyrithione Approved DB11327
small molecule | CAS: 3696-28-4

Dipyrithione, a bactericidal and fungicidal pyrithione derivate, was formulated as Crimanex anti-dandruff shampoo, but is no longer available.[L2611] It is currently used as a pesticide, and not used in any FDA approved drug products.[A32829] Interestingl…

Target Protein:
Nitric oxide synthase, inducibleProstaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CoenzymesEnzymes and Coenzymes
Target Protein:
Porphobilinogen deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diquafosol DB15919
small molecule | CAS: 59985-21-6

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +12
Target Protein:
P2Y purinoceptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diridavumab DB12607
biotech | CAS: 1393659-46-5

Cr6261 is under investigation in clinical trial NCT02016066 (A Study to Assess the Safety, Pharmacokinetics and Immunogenicity of Diridavumab in Japanese Healthy Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dirithromycin DB00954
small molecule | CAS: 62013-04-1

Dirithromycin is a macrolide glycopeptide antibiotic used to treat many different types of bacterial infections, such as bronchitis, pneumonia, tonsillitis, and even skin infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Target Protein:
23S ribosomal RNA
Waktu ParuhThe mean plasma hal…
Vol. Distribusi-
Klirens-
Genetik -
Dirlotapide DB11399
small molecule | CAS: 481658-94-0

Dirlotapide is a drug employed in the treatment of obesity in dogs. It is marketed by Pfizer and Zoetis under the brand name, _Slentrol_, and is not intended for human use.

Kategori:
Acids, AcyclicHeterocyclic Compounds, Fused-Ring
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dirocaftor DB16143
small molecule | CAS: 2137932-23-9

Dirocaftor is under investigation in clinical trial NCT03251092 (Study Designed to Assess the Safety, Tolerability and PK of PTI-808 in Healthy Volunteers and in Adults With Cystic Fibrosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diroximel fumarate Approved DB14783
small molecule | CAS: 1577222-14-0

Multiple Sclerosis (MS) is a chronic, debilitating neurological disease that can lead to profound cognitive and physical symptoms, severely affecting quality of life.[A176474] It is the main cause of neurological disability not caused by trauma in the young a…

Kategori:
Acids, AcyclicAntineoplastic and Immunomodulating AgentsDicarboxylic Acids +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-10
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensNo clearance inform…
Genetik -
Dirucotide DB04921
biotech | CAS: 152074-97-0

Dirucotide is a synthetically prepared peptide. In particular, the sequence prepared is a 17 amino acid chain that is identical to a section of myelin basic protein (MBP) that is found in humans. Dirucotide has been developed for the treatment of multiple scl…

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsMyelin Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130114-83-9

Disaccharide tripeptide glycerol dipalmitoyl is under investigation in clinical trial NCT00003667 (Combination Chemotherapy and Biological Therapy in Treating Patients With High-Risk Ewing's Sarcoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2136633-23-1

Disitamab vedotin is an antibody-drug conjugate drug targeting human epidermal growth factor receptor 2 (HER2). It is currently being investigated for cancers.[A254721]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-drug Conjugates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disitertide DB12953
biotech | CAS: 272105-42-7

Disitertide has been used in trials studying the treatment of Skin Fibrosis.

Target Protein:
Transforming growth factor beta-1 proprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disopyramide Approved DB00280
small molecule | CAS: 3737-09-5

A class I anti-arrhythmic agent (one that interferes directly with the depolarization of the cardiac membrane and thus serves as a membrane-stabilizing agent) with a depressant action on the heart similar to that of guanidine. It also possesses some anticholi…

Kategori:
Agents producing tachycardiaAntiarrhythmic agentsAntiarrhythmics, Class I +21
Target Protein:
Sodium channel protein type 5 subunit alphaMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +5
Waktu Paruh6.7 hours (range 4-…
Vol. Distribusi-
Klirens-
Genetik -
Disperse Blue 106 Approved DB14203
small molecule | CAS: 68516-81-4

Disperse Blue 106 is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distearyldimonium Approved DB14143
small molecule | CAS: 14357-21-2

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAminesAmmonium Compounds +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distigmine DB13694
small molecule | CAS: 17299-00-2

Distigmine is a parasympathomimetic agent with a longer duration of action and enhanced drug accumulation compared to [DB00545] and [DB01400]. It is an anticholinergic drug and long-acting reversible carbamate cholinesterase inhibitor that binds directly and …

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditazole DB08994
small molecule | CAS: 18471-20-0

Ditazole is a non-steroidal anti-inflammatory drug (NSAID). Ditazole's analgesic and antipyretic effects are similar to phenylbutazone. Additionally, ditazole is a platelet aggregation inhibitor marketed in Spain and Portugal with trade name Ageroplas.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansPlatelet Aggregation Inhibitors Excl. Heparin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiazanine DB11516
small molecule | CAS: 7187-55-5

Dithiazanine is a highly potent anthelmintic, introduced in 1959 for the treatment of strongyloid worms and whipworms. However, its use is severely limited due to its toxicity. Dithiazanine iodide was associated with eight fatal cases of severe acidosis and s…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiopyr DB15230
small molecule | CAS: 97886-45-8

Dithiopyr is under investigation in clinical trial NCT01236781 (Comparison of Full-Field Digital Mammography With Digital Breast Tomography for Screening Call-Back Rates).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditiocarb DB02520
small molecule | CAS: 147-84-2

A chelating agent that has been used to mobilize toxic metals from the tissues of man and experimental animals. It is the main metabolite of DISULFIRAM.

Kategori:
Acids, AcyclicAdjuvants, ImmunologicAnti-Infective Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditiocarb zinc Approved DB14193
small molecule | CAS: 14324-55-1

Ditiocarb zinc, also known as Diethyldithiocarbamic acid zinc salt, is a known chelator for copper and zinc. It also a dermatological sensitizer and allergen. Sensitivity to ditiocarb zinc may be identified with a clinical patch test.

Kategori:
Acids, AcyclicAdjuvants, ImmunologicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Divarasib DB17488
small molecule | CAS: 2417987-45-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Divozilimab DB18878
biotech | CAS: 2254061-60-2

Divozilimab is under investigation in clinical trial NCT05730699 (Efficacy and Safety of Divozilimab in Patients With Neuromyelitis Optica Spectrum Disorders (AQUARELLE)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixanthogen DB13712
small molecule | CAS: 502-55-6

Deskripsi belum tersedia.

Kategori:
AnionsAntiparasitic Products, Insecticides and RepellentsEctoparasiticides, Incl. Scabicides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha tocopheryl acetate Approved DB14477
small molecule | CAS: 52225-20-4

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha-Tocopherol Approved DB14476
small molecule | CAS: 10191-41-0

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18656-38-7

A synthetic phospholipid used in liposomes and lipid bilayers for the study of biological membranes. It is used in commercial drug preparations to solubilize drugs for injection [A32711]

Kategori:
Compounds used in a research, industrial, or household settingGlycerophosphatesGlycerophospholipids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-Methylephedrine Approved DB11278
small molecule | CAS: 1201-56-5

Methylephedrine is a sympathomimetic amine that appears in various over-the-counter cough and cold medications throughout the world [L2838], [L2839], [L2840]. The abuse of methylephedrine-containing medications has been reported in Japan. Methylephedrine is n…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Beta-1 adrenergic receptorAlpha-2A adrenergic receptorAlpha adrenergic receptor +1
Waktu Paruh3-6 hours (Ephedrin…
Vol. DistribusiEphedrine: 2.5-3.0 …
Klirens-
Genetik -
DLO6001 DB05178
small molecule

DL6001 is developed by DanioLabs using proprietary zebrafish technology to treat Parkinson’s disease symptoms including sialorrhoea and hyperhidrosis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DLO6002 DB05179
small molecule

DLO6002 is developed by Summit Corporation and is in phase I of clinical trials for the treatment of Parkinson's disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DM-1157 DB18600
small molecule | CAS: 1239953-66-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DMP-777 DB18488
small molecule | CAS: 157341-41-8

DMP-777 is a selective inhibitor of polymorphonuclear leukocyte (PMN) elastase.

Kategori:
AzetinesEnzyme InhibitorsPancreatic Elastase, antagonists & inhibitors
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNB-001 DB05757
small molecule

DNB-001 is a first-in-class oral therapy with dual mechanism of action, which is initially being developed for the treatment of glaucoma. In preclinical animal models, DNB-001 has demonstrated potent IOP- lowering effects as well as neuroprotective effects on…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNL343 DB18678
small molecule | CAS: 2278265-85-1

DNL343 is under investigation in clinical trial NCT05842941 (HEALEY ALS Platform Trial - Regimen G DNL343).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dobesilic acid DB13529
small molecule | CAS: 88-46-0

Deskripsi belum tersedia.

Kategori:
Antivaricose TherapyArylsulfonatesArylsulfonic Acids +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Docetaxel Approved DB01248
small molecule | CAS: 114977-28-5

Docetaxel is a clinically well established anti-mitotic chemotherapy medication used for the treatment of different types of cancer, including breast, ovarian, and non-small cell lung cancer. Docetaxel is a complex diterpenoid molecule and a semisynthetic ana…

Kategori:
Agents Causing Muscle ToxicityAntimitotic AgentsAntineoplastic Agents +32
Target Protein:
Tubulin beta-1 chainApoptosis regulator Bcl-2Nuclear receptor subfamily 1 group I member 2
Gen Terkait:
ABCC2
Waktu ParuhWith plasma samplin…
Vol. DistribusiDocetaxel has a ste…
KlirensAfter the administr…
Genetik 1 Varian
Doconexent Approved DB03756
small molecule | CAS: 6217-54-5

A mixture of fish oil and primrose oil, doconexent is used as a high-docosahexaenoic acid (DHA) supplement. DHA is a 22 carbon chain with 6 cis double bonds with anti-inflammatory effects. It can be biosythesized from alpha-linolenic acid or commercially manu…

Kategori:
Cytochrome P-450 CYP2C9 InhibitorsCytochrome P-450 CYP2C9 Inhibitors (strength unknown)Cytochrome P-450 CYP2C9 Substrates +11
Target Protein:
Peroxisome proliferator-activated receptor alphaProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +6
Waktu ParuhApproximately 20 ho…
Vol. DistribusiDHA is the most abu…
Klirens-
Genetik -
Docusate Approved DB11089
small molecule | CAS: 10041-19-7

Docusate, or dioctyl sulfosuccinate, is a stool softener indicated for the treatment of constipation[A32201]. Docusate acts by increasing the amount of water the stool absorbs in the gut, making the stool softer and easier to pass [L1801]. Docusate can be ora…

Kategori:
Alimentary Tract and MetabolismDrugs for ConstipationEnemas +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1442645-21-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dodecyl sulfate DB03967
small molecule | CAS: 151-41-7

Deskripsi belum tersedia.

Kategori:
AlcoholsAlkanesulfonatesAlkanesulfonic Acids +8
Target Protein:
Lysozyme CLipid A palmitoyltransferase PagP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1643-20-5

Deskripsi belum tersedia.

Kategori:
AminesCompounds used in a research, industrial, or household settingDetergents +3
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialReaction center protein L chainReaction center protein M chain +47
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dofequidar DB14067
small molecule | CAS: 129716-58-1

Dofequidar is an antineoplastic agent.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingP-glycoprotein inhibitors
Target Protein:
ATP-binding cassette sub-family B member 5ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dofetilide Approved DB00204
small molecule | CAS: 115256-11-6

Dofetilide is a class III antiarrhythmic agent that is approved by the Food and Drug Administration (FDA) for the maintenance of sinus rhythm in individuals prone to the formation of atrial fibrillation and flutter, and for the chemical cardioversion to sinus…

Kategori:
AmidesAminesAntiarrhythmic agents +17
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2Potassium channel subfamily K member 2ATP-sensitive inward rectifier potassium channel 12
Waktu Paruh10 hours
Vol. Distribusi* 3 L/kg
Klirens-
Genetik -
Dolasetron Approved DB00757
small molecule | CAS: 115956-12-2

Dolasetron is an antinauseant and antiemetic agent indicated for the prevention of nausea and vomiting associated with moderately-emetogenic cancer chemotherapy and for the prevention of postoperative nausea and vomiting. Dolasetron is a highly specific and s…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +21
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh8.1 hours
Vol. Distribusi* 5.8 L/kg [adults]
Klirens* Apparent cl=9.4 m…
Genetik -
Menampilkan 4751–4800 dari 12560
Sebelumnya Halaman 96 / 252 Berikutnya