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6694

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3751 (56.0%)
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Halaman 95 / 134
OM-301 DB18198
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omacetaxine mepesuccinate Approved DB04865
small molecule | CAS: 26833-87-4

Omacetaxine mepesuccinate (formerly known as HHT or Homoharringtonine), is a cephalotaxine ester and protein synthesis inhibitor with established clinical activity as a single agent in hematological malignancies. Omacetaxine mepesuccinate is synthesized from…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic Agents, Phytogenic +7
Target Protein:
50S ribosomal protein L2Large ribosomal subunit protein uL3
Waktu ParuhHomoharringtonine h…
Vol. DistribusiHomoharringtonine h…
KlirensClearance for homoh…
Genetik -
Omadacycline Approved DB12455
small molecule | CAS: 389139-89-3

Omadacycline has been used in trials studying the treatment of Bacterial Pneumonia, Bacterial Infections, Community-Acquired Infections, and Skin Structures and Soft Tissue Infections. Omadacycline represents a significant advance over the well-known tetracyc…

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Target Protein:
30S ribosomal protein S330S ribosomal protein S730S ribosomal protein S8 +3
Waktu ParuhOmadacycline has a …
Vol. DistribusiOmadacycline has a …
KlirensOmadacycline has a …
Genetik -
Omapatrilat DB00886
small molecule | CAS: 167305-00-2

Omapatrilat is an investigational drug that inhibits both neutral endopeptidase (NEP) and angiotensin converting enzyme (ACE). The inhibition of NEP elevates natriuretic peptide levels, increasing excretion of sodium in urine, dilating blood vessels, and redu…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +11
Target Protein:
NeprilysinAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omarigliptin DB11992
small molecule | CAS: 1226781-44-7

Omarigliptin has been used in trials studying the treatment of Type 2 Diabetes Mellitus and Chronic Renal Insufficiency.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDPP-IV Inhibitors +1
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ombitasvir Approved DB09296
small molecule | CAS: 1258226-87-7

Ombitasvir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
AmidesAminesAmino Acids +18
Target Protein:
Nonstructural protein 5AGenome polyprotein
Waktu ParuhOmbitasvir has a ha…
Vol. DistribusiOmbitasvir has a vo…
KlirensClearance of Ombita…
Genetik -
small molecule | CAS: 873697-71-3

Omecamtiv Mecarbil has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic Heart Failure, and History of Chronic Heart Failure, among others.

Kategori:
AmidesCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Target Protein:
Myosin-binding protein C, cardiac-type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omega-3 fatty acids Approved DB11133
small molecule | CAS: 329042-31-1

Omega-3 fatty acids are polyunsaturated fatty acids (PUFAs) with a double bond at the third carbon atom from the end of the carbon chain. The three types of omega-3 fatty acids involved in human physiology are ?-linolenic acid (ALA) (found in plant oils), eic…

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyDietary Fats +12
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alphaSterol regulatory element-binding protein 1
Waktu ParuhApproximate half-li…
Vol. DistribusiVd of EPA is aproxi…
KlirensClearance of EPA is…
Genetik -
Omega-3-acid ethyl esters Approved DB09539
small molecule | CAS: 308081-97-2

Omega-3-acid ethyl esters are prescription drugs that contain eicosapentaenoic acid-ethyl ester (EPA) and docosahexaenoic acid-ethyl ester (DHA) that are used in combination with changes in diet to lower triglyceride levels in adults with severe (? 500 mg/dL)…

Kategori:
AutacoidsBiological FactorsDiet, Food, and Nutrition +15
Target Protein:
Sterol regulatory element-binding protein 1
Waktu Paruh79 hours ± 47 hours…
Vol. Distribusi82 ± 56L[A18890]
Klirens757 mL/h ± 283mL/h[…
Genetik -
Omega-3-carboxylic acids Approved DB09568
small molecule

The omega-3 carboxylic acid (OM3-CA) is a new formulation of omega-3 fatty acids that present an enhanced bioavailability in the treatment of dyslipidemia. The increased bioavailability is explained because OM3-CA is found in a form of polyunsaturated free f…

Kategori:
Fatty Acids, Omega-3
Target Protein:
Diacylglycerol O-acyltransferase 23-hydroxyacyl-CoA dehydrogenase type-2Enoyl-CoA hydratase, mitochondrial +3
Waktu ParuhThe half-life of OM…
Vol. DistribusiThis pharmacokineti…
KlirensThe registered clea…
Genetik -
small molecule

Omega-6 fatty acids are polyunsaturated fatty acids with a final carbon-carbon double bond in the n-6 position, that is, the sixth bond, counting from the methyl end. They are a family of fatty acid molecules that act as precursors to potent lipid mediator si…

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omeprazole Approved DB00338
small molecule | CAS: 73590-58-6

Originally approved by the FDA in 1989, omeprazole is a _proton-pump inhibitor_, used to treat gastric acid-related disorders. These disorders may include gastroesophageal reflux disease (GERD), peptic ulcer disease, and other diseases characterized by the ov…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +37
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaAryl hydrocarbon receptor
Gen Terkait:
CYP2C19 CYP2C19
Waktu Paruh0.5-1 hour (healthy…
Vol. DistribusiApproximately 0.3 L…
KlirensHealthy subject (de…
Genetik 2 Varian
biotech | CAS: 2249927-58-8

Omfiloctocog alfa is under investigation in clinical trial NCT03947567 (Safety and Efficacy of Long-term Treatment With SCT800 in Previously Treated Hemophilia a Patients.).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Omidenepag isopropyl Approved DB15071
small molecule | CAS: 1187451-19-9

Omidenepag isopropyl is a topical ocular hypotensive agent used to reduce intraocular pressure (IOP) in patients with glaucoma and ocular hypertension.[L43503] Omidenepag isopropyl is quickly metabolized to its active metabolite, omidenepag, a molecule with h…

Kategori:
Antiglaucoma AgentsHypotensive AgentsOphthalmic Solutions +6
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype
Waktu ParuhThe half-life of om…
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Omidubicel Approved DB17132
biotech

Omidubicel is a nicotinamide-modified allogeneic hematopoietic progenitor cell therapy derived from cord blood used as an allogeneic stem cell donor source. Umbilical blood cord cells are expanded _ex-vivo_ and [nicotinamide] (a form of vitamin B3) is used as…

Kategori:
Allogeneic Cord Blood Hematopoietic Progenitor Cell TherapyCells, AllogeneicCells, Cultured, Allogeneic +1
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Omiganan DB06610
small molecule | CAS: 204248-78-2

Omiganan has been investigated for the treatment of Mupirocin-resistant MRSA skin infections.

Kategori:
Amino Acids, Peptides, and ProteinsAntimicrobial PeptidesMembrane Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ompenaclid DB18819
small molecule | CAS: 353-09-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmidinesFatty Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OMS906 DB17722
biotech

OMS906 is a humanized Igg4 monoclonal antibody against mannan-binding lectin-associated serine protease-3 (MASP-3) currently being developed by Omeros.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Onasemnogene abeparvovec Approved DB15528
biotech | CAS: 1922968-73-7

Onasemnogene abeparvovec is an adeno-associated virus vector-based gene therapy that has been approved by the FDA in May 2019 for the treatment of infant patients (less than 2 years of age) with spinal muscular atrophy (SMA) and a specific mutation in the sur…

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsBiological Products +7
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Onatasertib DB12570
small molecule | CAS: 1228013-30-6

Onatasertib (CC-223) has been used in trials studying the treatment and basic science of Multiple Myeloma, Glioblastoma Multiforme, HepatoCellular Carcinoma, Non-small Cell Lung Cancer, and Diffuse Large B-Cell Lymphoma, among others.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ondansetron Approved DB00904
small molecule | CAS: 99614-02-5

A competitive serotonin type 3 receptor antagonist. It is effective in the treatment of nausea and vomiting caused by cytotoxic chemotherapy drugs, including cisplatin, and has reported anxiolytic and neuroleptic properties. Having been developed in the 19…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +29
Target Protein:
5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 4Mu-type opioid receptor +2
Gen Terkait:
CYP2D6 CYP2D6
Waktu ParuhThe half-life of on…
Vol. DistribusiThe volume of distr…
KlirensThe clearance value…
Genetik 2 Varian
Ongericimab DB18949
biotech | CAS: 2145096-91-7

Ongericimab is under investigation in clinical trial NCT05325203 (A Study to Evaluate the Efficacy and Safety of JS002 in Patients With Heterozygous Familial Hypercholesterolemia (Hefh).).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ontamalimab DB15298
biotech | CAS: 2098790-40-8

Ontamalimab is under investigation in clinical trial NCT03627091 (Efficacy and Safety Study of SHP647 as Maintenance Treatment in Participants With Moderate to Severe Crohn's Disease (CARMEN CD 307)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ontuxizumab DB16270
biotech | CAS: 946415-62-9

Ontuxizumab is a humanized monoclonal antibody that targets endosialin or tumour endothelial marker 1 (TEM-1). It is under investigation in clinical trial NCT01574716 (Sarcoma Study of Morab-004 Utilization: Research and Clinical Evaluation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onvansertib DB15110
small molecule | CAS: 1034616-18-6

Onvansertib is under investigation in clinical trial NCT03303339 (Onvansertib in Combination With Either Low-dose Cytarabine or Decitabine in Adult Patients With Acute Myeloid Leukemia (AML).).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase PLK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OP-145 DB05672
biotech | CAS: 732984-79-1

OP-145 is a synthetic antimicrobial peptide developed from human cathelicidin LL-37.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OPC-51803 DB05838
small molecule

OPC-51803 is the first nonpeptide vasopressin (AVP) V(2)-receptor-selective agonist. It is a V(2)-selective agonist that produces a significant antidiuretic action after single and multiple oral dosing in AVP-deficient and normal AVP states. It is useful ther…

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Vasopressin, agonists
Target Protein:
Vasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opebacan DB06161
biotech | CAS: 206254-79-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opicapone Approved DB11632
small molecule | CAS: 923287-50-7

Opicapone is a potent, reversible, and peripherally-acting third-generation inhibitor of catechol-o-methyltransferase (COMT), an enzyme involved in the breakdown of various catecholamines including dopamine.[A36938, A203048] Many patients with Parkinson’s dis…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBCRP/ABCG2 Substrates +25
Target Protein:
Catechol O-methyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing oral admi…
KlirensFollowing oral admi…
Genetik -
Opicinumab DB14959
biotech | CAS: 1422268-07-2

Opicinumab is under investigation in clinical trial NCT02641041 (Safety, Tolerability, and Pharmacokinetics of Single and Multiple Doses of BIIB033 in Healthy Japanese Participants).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opium Approved DB11130
small molecule | CAS: 8008-60-4

Opium is the first substance of the diverse group of the opiates. It has been known for a long time, and the first evidence of a poppy culture dates from 5 thousand years by the Sumerians. During the years, opium was used as a sedative and hypnotic, but it wa…

Kategori:
Alimentary Tract and MetabolismAnalgesicsAntidiarrheals +25
Target Protein:
Delta-type opioid receptorKappa-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half-life of op…
Vol. DistribusiOpium presents a la…
Klirens-
Genetik -
biotech | CAS: 945228-48-8

VB4-845 is studied in the treatment of certain types of head and neck cancer. VB4-845 is made by linking a monoclonal antibody fragment to a toxic protein that may kill cancer cells. VB4-845 is a fusion protein containing humanized scFv specific for the epith…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +8
Target Protein:
Epithelial cell adhesion molecule
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oprelvekin Approved DB00038
biotech | CAS: 145941-26-0

Oprelvekin, the active ingredient in Neumega®, is recombinant Interleukin-11 (IL-11), which is produced in Escherichia coli (E. coli) by recombinant DNA technology. With a molecular mass of approximately 19,000 daltons, the non-glycosylated protein is 177 ami…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-11 receptor subunit alpha
Waktu Paruh6.9 +/- 1.7 hrs
Vol. Distribusi-
Klirens-
Genetik -
Oprozomib DB11991
small molecule | CAS: 935888-69-0

Oprozomib has been used in trials studying the treatment of Solid Tumors, Multiple Myeloma, Waldenstrom Macroglobulinemia, Advanced Hepatocellular Carcinoma, and Advanced Non-Central Nervous System (CNS) Malignancies.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OptPA DB18325
biotech

Optimized tPA (OptPA; W253R/R275S-tPA) is an engineered variant of tPA designed to exhibit reduced neurotoxicity.[A261486]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The oral polio vaccine (OPV) is a live attenuated vaccine containing a mixture of one or more strains of poliovirus serotypes. Strains of the virus are selected based on their reduced incidence of spreading to the central nervous system but still having the a…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orbifloxacin DB11443
small molecule | CAS: 113617-63-3

Orbifloxacin is a fluoroquinolone antibiotic. It is marketed by Schering-Plough Animal Health and approved for certain infections in dogs.

Kategori:
4-QuinolonesAnti-Bacterial AgentsCytochrome P-450 CYP1A2 Inhibitors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORC-13661 DB18903
small molecule | CAS: 1979935-33-5

ORC-13661 is under investigation in clinical trial NCT05730283 (Prevention of Ototoxicity in NTM Patients Treated With IV Amikacin).

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orciprenaline Approved DB00816
small molecule | CAS: 586-06-1

A beta-adrenergic agonist used in the treatment of asthma and bronchospasms. [PubChem]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +26
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh6 hours
Vol. Distribusi-
Klirens-
Genetik -
Oregovomab DB04964
biotech | CAS: 213327-37-8

Oregovomab is a murine monoclonal antibody that attaches to the tumor-associated antigen CA125.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Mucin-16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orellanine DB19263
small molecule | CAS: 37338-80-0

Orellanine is under investigation in clinical trial NCT05287945 (Study of Orellanine in Metastatic Clear-cell or Papillary Renal Cell Carcinoma).

Kategori:
AgaricalesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orforglipron DB18964
small molecule | CAS: 2212020-52-3

Orforglipron is under investigation in clinical trial NCT06010004 (A Long-term Safety Study of Orforglipron (LY3502970) in Participants With Type 2 Diabetes).

Kategori:
Oxazoles
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orgotein DB11444
biotech | CAS: 1569268-91-2

Superoxide is a natural byproduct of oxygen metabolism which, if left unchecked, leads to cell damage. Superoxide dismutase (SOD) is an enzyme that alternately catalyzes the dismutation of the superoxide radical into either the less damaging hydrogen peroxide…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oridonin DB19086
small molecule | CAS: 28957-04-2

Oridonin is under investigation in clinical trial NCT05130892 (Effect of Inflammasome Inhibitor on Hscrp in Patients After PCI).

Kategori:
DiterpenesTerpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
Orlistat Approved DB01083
small molecule | CAS: 96829-58-2

The global prevalence of obesity is increasing rapidly. Obesity-related complications lead to significant personal and economic burden by reducing quality of life and increasing the cost of healthcare. In some individuals, diet and exercise are insufficient …

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAntiobesity Preparations, Excl. Diet Products +11
Target Protein:
Pancreatic triacylglycerol lipaseCannabinoid receptor 1Gastric triacylglycerol lipase +1
Waktu ParuhThe half-life of or…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
ORM-12741 DB12057
small molecule | CAS: 610782-82-6

ORM-12741 has been used in trials studying the basic science and treatment of Alzheimer's Disease.

Kategori:
Adrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +2
Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ornithine Approved DB00129
small molecule | CAS: 70-26-8

Produced during the urea cycle, ornithine is an amino acid produced from the splitting off of urea from arginine. L-Ornithine allows for the disposal of excess nitrogen and acts as a precursor of citrulline and arginine.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +9
Target Protein:
Ornithine aminotransferase, mitochondrialOrnithine transcarbamylase, mitochondrialArginase-1 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orotic acid DB02262
small molecule | CAS: 65-86-1

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialOrotate phosphoribosyltransferaseDihydroorotate dehydrogenase (quinone), mitochondrial +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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