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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 95 / 236
Emicerfont DB12910
small molecule | CAS: 786701-13-1

Emicerfont has been used in trials studying the diagnostic and treatment of Social Anxiety Disorder and Irritable Bowel Syndrome (IBS).

Kategori:
Corticotropin-Releasing Hormone, antagonists & inhibitors
Target Protein:
Corticotropin-releasing factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emicizumab Approved DB13923
biotech | CAS: 1610943-06-0

Emicizumab is a humanized recombinant monoclonal antibody that mimics the function of the coagulation Factor VIII and it has the capacity to bind simultaneously to activated Factor IX and Factor X. The ability of Emicizumab to bind to all these three differen…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Coagulation factor IXCoagulation factor X
Waktu ParuhEmcicizumab present…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Emivirine DB08188
small molecule | CAS: 149950-60-7

Emivirine has been used in trials studying the treatment of HIV Infections.

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiviral Agents +5
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emixustat DB12608
small molecule | CAS: 1141777-14-1

Emixustat has been used in trials studying the treatment of Geographic Atrophy, Age-Related Macular Degeneration, and Dry Age-related Macular Degeneration.

Kategori:
AlcoholsAminesAmino Alcohols +4
Target Protein:
Retinoid isomerohydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emlenoflast DB18304
small molecule | CAS: 1995067-59-8

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Emodin DB07715
small molecule | CAS: 518-82-1

Emodin has been investigated for the treatment of Polycystic Kidney.

Kategori:
AnthracenesAnthraquinonesBiological Products +7
Target Protein:
Casein kinase II subunit alphaPutative ketoacyl reductase3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emopamil DB14064
small molecule | CAS: 78370-13-5

Prevents renal injury after warm & cold ischemia.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +11
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Emoxypine DB19172
small molecule | CAS: 2364-75-2

Emoxypine is under investigation in clinical trial NCT06221826 (MEXIDOL® in the Rehabilitation Treatment of Patients With Acute Cerebral Failure).

Kategori:
Antiarrhythmic agentsAntioxidantsAntiplatelet agents +13
Waktu Paruh-
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Klirens-
Genetik -
Empagliflozin Approved DB09038
small molecule | CAS: 864070-44-0

Empagliflozin is an inhibitor of sodium-glucose co-transporter-2 (SGLT2), the transporters primarily responsible for the reabsorption of glucose in the kidney.[A203453] It is used clinically as an adjunct to diet and exercise, often in combination with other …

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 SubstratesBenzene Derivatives +16
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhThe apparent termin…
Vol. DistribusiThe estimated appar…
KlirensApparent oral clear…
Genetik -
Empasiprubart DB16469
biotech | CAS: 2579031-19-7

Empasiprubart is a humanized sweeping antibody designed to bind to C2, a protein in the complement cascade that leads to cell destruction when activated.[L50783]

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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Empegfilgrastim DB16155
biotech | CAS: 1192706-53-8

Empegfilgrastim is under investigation in clinical trial NCT01569087 (Dose-finding Study of Empegfilgrastim for Neutropenia Prophylaxis in Patients With Breast Cancer).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors
Waktu Paruh-
Vol. Distribusi-
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Emprumapimod DB17603
small molecule | CAS: 765914-60-1

Emprumapimod is a potent, orally active and selective inhibitor of p38? mitogen-activated kinase inhibitor. It was investigated for dilated cardiomyopathy.

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Emraclidine DB18706
small molecule | CAS: 2170722-84-4

Deskripsi belum tersedia.

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Emricasan DB05408
small molecule | CAS: 254750-02-2

Emricasan is the first caspase inhibitor tested in human which has received orphan drug status by FDA. It is developed by Pfizer and made in such a way that it protects liver cells from excessive apoptosis.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Caspase-1Caspase-3Caspase-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emrusolmin DB13927
small molecule | CAS: 882697-00-9

Emrusolmin restores hippocampal synaptic and transcriptional plasticity as well as spatial memory in a mouse model for Alzheimer's disease, when given orally before or after the onset of pathology. [A31409]

Kategori:
DioxolesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emtricitabine Approved DB00879
small molecule | CAS: 143491-57-0

Emtricitabine is a nucleoside reverse transcriptase inhibitor (NRTI) indicated for the treatment of HIV infection in adults[L9019] or combined with [tenofovir alafenamide] for the prevention of HIV-1 infection in high risk adolescents and adults.[L9010] Emtri…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +23
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyprotein
Waktu ParuhThe half life of em…
Vol. DistribusiThe apparent centra…
KlirensEmtricitabine has a…
Genetik -
Emylcamate DB13572
small molecule | CAS: 78-28-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAnti-Anxiety AgentsCarbamates +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EMZ702 DB05021
small molecule

EMZ702, a non-toxic agent that has strong anti-viral synergy with interferon, is an ideal candidate for combination with current standard hepatitis C treatments. EMZ702 has an excellent safety profile and the combination of EMZ702 with interferon and ribaviri…

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Enadenotucirev DB14873
biotech | CAS: 1402042-02-7

Enadenotucirev is under investigation in clinical trial NCT02636036 (Phase I Study of Enadenotucirev and PD-1 Inhibitor in Subjects With Metastatic or Advanced Epithelial Tumors).

Waktu Paruh-
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Enadoline DB16967
small molecule | CAS: 124378-77-4

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCardiovascular AgentsCentral Nervous System Agents +4
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enalapril Approved DB00584
small molecule | CAS: 75847-73-3

Enalapril is a prodrug belonging to the angiotensin-converting enzyme (ACE) inhibitor drug class that works on the renin-angiotensin-aldosterone system, which is responsible for the regulation of blood pressure and fluid and electrolyte homeostasis. Enalapril…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +21
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensFollowing oral admi…
Genetik -
Enalaprilat Approved DB09477
small molecule | CAS: 76420-72-9

Enalaprilat is the active metabolite of the orally available pro-drug, [enalapril]. Used in the treatment of hypertension, enalapril is an ACE inhibitor that prevents Angiotensin Converting Enzyme (ACE) from transforming angiotensin I into angiotensin II. As …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +15
Target Protein:
Angiotensin-converting enzymeB1 bradykinin receptor
Waktu Paruh11 hr
Vol. Distribusi-
KlirensThe disposition of …
Genetik -
Enalkiren DB03395
small molecule | CAS: 113082-98-7

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAmino Acids, Peptides, and ProteinsEnzyme Inhibitors +4
Target Protein:
Renin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1912424-97-5

Enapotamab vedotin is under investigation in clinical trial NCT02988817 (Enapotamab Vedotin (Humax-axl-adc) Safety Study in Patients With Solid Tumors).

Kategori:
Antibody-drug Conjugates
Waktu Paruh-
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Genetik -
Enasidenib Approved DB13874
small molecule | CAS: 1446502-11-9

Enasidenib is an orally available treatment for the treatment of adult patients with relapsed or refractory acute myeloid leukemia (AML) with specific mutations in the isocitrate dehydrogenase 2 (IDH2) gene, which is a recurrent mutation detected in 12-20% of…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +62
Target Protein:
Isocitrate dehydrogenase [NADP] cytoplasmicIsocitrate dehydrogenase [NAD] subunit alpha, mitochondrialIsocitrate dehydrogenase [NAD] subunit beta, mitochondrial +2
Waktu ParuhEnasidenib has a te…
Vol. DistribusiThe mean volume of …
KlirensEnasidenib has a me…
Genetik -
Enavogliflozin DB18970
small molecule | CAS: 1415472-28-4

Enavogliflozin is under investigation in clinical trial NCT06399835 (Enavogliflozin vs. Pioglitazone on Glucose and Atherosclerosis).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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ENB-003 DB17340
small molecule

ENB-003 is a selective and potent inhibitor of the endothelin B receptor (ETBR) being investigated for cancer.

Waktu Paruh-
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Encainide Approved DB01228
small molecule | CAS: 66778-36-7

All drug products containing encainide hydrochloride. Encainide hydrochloride, formerly marketed as Enkaid capsules, was associated with increased death rates in patients who had asymptomatic heart rhythm abnormalities after a recent heart attack. The manufac…

Kategori:
AmidesAminesAnilides +13
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Encaleret DB18096
small molecule | CAS: 787583-71-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlcoholsAmines +3
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Encenicline DB11726
small molecule | CAS: 550999-75-2

Encenicline has been investigated for the treatment of Cognition, Schizophrenia, Alzheimer's Disease, Cardiac Repolarization, and Central Nervous System Diseases.

Kategori:
Nicotinic AgonistsSulfur Compounds
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
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Klirens-
Genetik -
Enclomiphene DB06735
small molecule | CAS: 15690-57-0

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsClomiphene +11
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Encorafenib Approved DB11718
small molecule | CAS: 1269440-17-6

Encorafenib, also known as _BRAFTOVI_, is a kinase inhibitor. Encorafenib inhibits BRAF gene, which encodes for B-raf protein, which is a proto-oncogene involved in various genetic mutations.[L12216] This protein plays a role in regulating the MAP kinase/E…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +47
Target Protein:
Serine/threonine-protein kinase B-rafG1/S-specific cyclin-D1RAF proto-oncogene serine/threonine-protein kinase +7
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe blood-to-plasma…
KlirensThe apparent cleara…
Genetik -
Endostar DB11727
biotech

Endostar is under investigation for the treatment of Nasopharyngeal Carcinoma. Endostar has been investigated for the treatment of Non-small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endostatin DB06423
biotech | CAS: 187888-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
72 kDa type IV collagenaseMatrix metalloproteinase-9Collagenase 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endothelin-1 DB12652
biotech | CAS: 117399-94-7

Endothelin 1 is under investigation in clinical trial NCT00745693 (The Effects of Diesel Exhaust Inhalation on Vascular Function - the Role of Endothelin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsEndothelin-1, antagonists & inhibitors +4
Waktu Paruh-
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Genetik -
Endralazine DB13435
small molecule | CAS: 39715-02-1

Deskripsi belum tersedia.

Kategori:
Antihypertensive AgentsArteriolar Smooth Muscle, Agents Acting OnCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eneboparatide DB18207
biotech | CAS: 1349298-00-5

Deskripsi belum tersedia.

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Enflurane Approved DB00228
small molecule | CAS: 13838-16-9

Enflurane is a halogenated inhalational anesthetic initially approved by the FDA in 1972. Since this date, it has been withdrawn from the US market.[L13646,L13649] Unlike its other inhalational anesthetic counterparts including [isoflurane] and [halothane], e…

Kategori:
Agents that reduce seizure thresholdAnestheticsAnesthetics, General +8
Target Protein:
GABA(A) ReceptorVoltage-dependent calcium channelGlycine receptor subunit alpha-1 +4
Waktu Paruh-
Vol. DistribusiEnflurane distribut…
Klirens-
Genetik -
Enfortumab vedotin Approved DB13007
biotech | CAS: 1346452-25-2

Enfortumab vedotin is an antibody-drug conjugate used in the treatment of patients with advanced, treatment-resistant urothelial cancers.[L10836] It is comprised of a fully human monoclonal antibody targeted against Nectin-4 and a microtubule-disrupting chemo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Nectin-4
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimated stead…
KlirensThe mean clearance …
Genetik -
biotech | CAS: 2567881-77-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Genetik -
Engensis DB17931
biotech

Deskripsi belum tersedia.

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Genetik -
English walnut Approved DB10577
biotech

English walnut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Genetik -
biotech | CAS: 2417199-08-5

Englumafusp alfa is under investigation in clinical trial NCT04077723 (A Study to Evaluate the Safety, Pharmacokinetics and Preliminary Anti-tumor Activity of Englumafusp Alfa in Combination With Obinutuzumab and in Combination With Glofitamab Following a Pre…

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Enibarcimab DB16730
biotech | CAS: 2305638-98-4

Enibarcimab is under investigation in clinical trial NCT03989531 (Adrecizumab in Cardiogenic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enitociclib DB17297
small molecule | CAS: 1610408-97-3

Deskripsi belum tersedia.

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ENMD-1198 DB05959
small molecule | CAS: 864668-87-1

Deskripsi belum tersedia.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Hypoxia-inducible factor 1-alphaTumor necrosis factor receptor superfamily member 11ASignal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-981693 DB16891
small molecule | CAS: 934353-76-1

Deskripsi belum tersedia.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Enoblituzumab DB15017
biotech | CAS: 1353485-38-7

Enoblituzumab is under investigation in clinical trial NCT02982941 (Enoblituzumab (MGA271) in Children With B7-H3-expressing Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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