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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 95 / 252
Diiodohydroxyquinoline Approved DB09115
small molecule | CAS: 83-73-8

Diiodohydroxyquinoline, also known as uidoquinol and iodoquinol, is a quinoline derivative that can be used in the treatment of amoebiasis. The exact mechanism of action is unknown. Iodoquinol is not currently available in any FDA-approved products.

Kategori:
AmebicidesAnti-Infective AgentsAntiparasitic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diisopromine DB13476
small molecule | CAS: 5966-41-6

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1445-75-6

Deskripsi belum tersedia.

Target Protein:
Parathion hydrolaseParathion hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dilazep DB13715
small molecule | CAS: 35898-87-4

Deskripsi belum tersedia.

Kategori:
AzepinesCardiac TherapyCardiovascular Agents +2
Target Protein:
Equilibrative nucleoside transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diloxanide DB08792
small molecule | CAS: 579-38-4

Diloxanide (as [Diloxanide furoate]) is an anti-protozoal drug used in the treatment of Entamoeba histolytica and some other protozoal infections. Although it is not currently approved for use in the United States, it was approved by a CDC study in the treatm…

Kategori:
AmebicidesAnti-Infective AgentsAntiparasitic Agents +4
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Dilpacimab DB16140
biotech | CAS: 1791420-09-1

Dilpacimab is under investigation in clinical trial NCT03368859 (A Study of ABT-165 Plus FOLFIRI vs Bevacizumab Plus FOLFIRI in Subjects With Metastatic Colorectal Cancer Previously Treated With Fluoropyrimidine, Oxaliplatin and Bevacizumab).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diltiazem Approved DB00343
small molecule | CAS: 42399-41-7

Diltiazem is a benzothiazepine derivative with antihypertensive and vasodilating properties. Approved in 1982 by the FDA, it is a member of the non-dihydropyridine calcium channel blockers drug class. It works through various mechanisms of action, but it prim…

Kategori:
Agents causing hyperkalemiaAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAntiarrhythmic agents +44
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent calcium channel gamma-1 subunit
Gen Terkait:
ADRB1
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensFollowing a single …
Genetik 1 Varian
Dimazole Approved DB13858
small molecule | CAS: 95-27-2

Dimazole (diamthazole) is an antifungal. It was withdrawn in Franch in 1972 due to neuropsychiatric reactions.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimefline DB13482
small molecule | CAS: 1165-48-6

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimenhydrinate Approved DB00985
small molecule | CAS: 523-87-5

Dimehydrinate was first described in the literature in 1949,[A233120] and patented in 1950.[L32995] Early research into dimenhydrinate focused on its role as an antihistamine for urticaria; the treatment of motion sickness was an accidental discovery.[A233130…

Kategori:
AlkaloidsAminesAminoalkyl Ethers +21
Target Protein:
Histamine H1 receptor
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Dimenoxadol DB01461
small molecule | CAS: 509-78-4

Dimenoxadol is an opioid analgesic which produces typical opioid effects such as analgesia and sedation. It is structurally similar to methadone and is a benzilic acid derivative. In the United States it is classified as a Schedule I controlled drug.

Kategori:
Acids, CarbocyclicDiphenylacetic AcidsHydroxy Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimepheptanol DB19094
small molecule | CAS: 545-90-4

Dimepheptanol is under investigation in clinical trial NCT00218127 (Treatment of Opioid/heroin Dependence: Comparison of Three Medication Dosing Regimens).

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +5
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimercaprol Approved DB06782
small molecule | CAS: 59-52-9

Dimercaprol is a traditional chelating agent developed by British biochemists at Oxford University during World War II. It was developed as an experimental antidote against the arsenic-based poison gas Lewisite. It has been used clinically since 1949 in arsen…

Kategori:
AntidotesChelating AgentsCompounds used in a research, industrial, or household setting +7
Target Protein:
ArsenicCadmiumMercury +1
Waktu ParuhThe drug has a shor…
Vol. Distribusi-
Klirens-
Genetik -
Dimericine DB17833
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDeoxyribonucleasesEndodeoxyribonucleases +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimetacrine DB08996
small molecule | CAS: 4757-55-5

Dimetacrine is also known as dimethacrine or acripamine. It is marketed under the names Istonil, Istonyl, Linostil, and Miroistonil. Dimetacrine is a tricyclic antidepressant (TCA) with imipramine-like effects used in Europe for the treatment of depression. D…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +9
Target Protein:
Acetylcholinesterase
Waktu ParuhApproximately 10 ho…
Vol. DistribusiThe highest concent…
Klirens-
Genetik -
small molecule | CAS: 366472-45-9

Dimethandrolone Undecanoate is under investigation in clinical trial NCT03455075 (Study of Spermatogenesis Suppression With DMAU Alone or With LNG Versus Placebo Alone in Normal Men).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimethicone 410 Approved DB14005
small molecule | CAS: 9006-65-9

Dimethicone is a silicone-based polymer used as a moisturizer in different skin OTC products.[A32462] It is formed by repeated polymeric units of -(CH3)2SiO- with a terminal trimethyl siloxy unit.[L1769] It is currently recognized by the FDA as a skin protect…

Waktu ParuhAs dimethicone is p…
Vol. DistribusiAs dimethicone is p…
KlirensA very minimal amou…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Estrogen receptorNuclear receptor coactivator 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 39589-98-5

Dimethyl carbate is used as an insect repellant.

Kategori:
Antiparasitic Products, Insecticides and RepellentsEctoparasiticides, Incl. Scabicides, Insecticides and RepellentsInsecticides and Repellents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimethyl fumarate Approved DB08908
small molecule | CAS: 624-49-7

Dimethyl fumarate is an agent indicated for the treatment of relapsing forms of multiple sclerosis.[A253942,L43752] The mechanism of action of dimethyl fumarate in multiple sclerosis is not well understood. It is thought to involve dimethyl fumarate degradati…

Kategori:
Acids, AcyclicAnti-Inflammatory AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
Kelch-like ECH-associated protein 1Transcription factor p65
Waktu ParuhThe dimethyl fumara…
Vol. DistribusiIn healthy people, …
KlirensMonomethyl fumarate…
Genetik -
Dimethyl sulfoxide Approved DB01093
small molecule | CAS: 67-68-5

A highly polar organic liquid, that is used widely as a chemical solvent. Because of its ability to penetrate biological membranes, it is used as a vehicle for topical application of pharmaceuticals. It is also used to protect tissue during cryopreservation. …

Kategori:
AntioxidantsCompounds used in a research, industrial, or household settingCryoprotective Agents +20
Target Protein:
Interleukin-5 receptor subunit alphaMucin-16Myc proto-oncogene protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Dual specificity tyrosine-phosphorylation-regulated kinase 1ADual specificity tyrosine-phosphorylation-regulated kinase 2Casein kinase II subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 358-72-5

Deskripsi belum tersedia.

Kategori:
Terpenes
Target Protein:
Farnesyl pyrophosphate synthaseIsopentenyl-diphosphate Delta-isomerase 14-hydroxy-3-methylbut-2-enyl diphosphate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1403357-81-2

Deskripsi belum tersedia.

Kategori:
CycloheptanesCycloparaffinsPolycyclic Sesquiterpenes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 52328-98-0

Dimethylcurcumin is a synthetic chemical compound that is loosely based on a compound found in curcumin. It is a novel anti-androgen that enhances androgen receptor degradation.

Kategori:
AlkanesBenzene DerivativesCatechols +4
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 524-84-5

Dimethylthiambutene (N,N-Dimethyl-1-methyl-3,3-di-2-thienylallylamine, Dimethibutin, Ohton) is an opioid analgesic drug. It is now under international control under Schedule I of the UN Single Convention On Narcotic Drugs 1961, presumably due to high abuse po…

Target Protein:
Mu-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61-50-7

An N-methylated indoleamine derivative, a serotonergic hallucinogen found in several plants, especially Prestonia amazonica (Apocynaceae) and in mammalian brain, blood, and urine. It apparently acts as an agonist at some types of serotonin receptors and an an…

Kategori:
AminesAntidepressive AgentsBiogenic Amines +13
Target Protein:
5-hydroxytryptamine receptor 6Sigma non-opioid intracellular receptor 15-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimetindene Approved DB08801
small molecule | CAS: 5636-83-9

Dimetindene (Fenistil) is an antihistamine/anticholinergic used orally and locally as an antipruritic.

Kategori:
Agents producing tachycardiaAnti-Allergic AgentsAnticholinergic Agents +13
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimetofrine DB13494
small molecule | CAS: 22950-29-4

Deskripsi belum tersedia.

Kategori:
Adrenergic and Dopaminergic AgentsAlcoholsAmines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimetotiazine Approved DB08967
small molecule | CAS: 7456-24-8

Dimetotiazine has considerable antiemetic & serotonin antagonistic action used mainly in allergic skin conditions.

Kategori:
AnalgesicsAntimigraine PreparationsHeterocyclic Compounds, Fused-Ring +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diminazene DB03608
small molecule | CAS: 536-71-0

Diminazene, also known as Diminazine, 4,4'-(Diazoamino)benzamidine, 4,4'-(1-triazene-1,3-diyl)bis-benzenecarboximidamide, diminazine aceturate, or Diminazene aceturate, is a trypanocidal agent. Major brands of Diminazene are Berenil, Pirocide, Ganasag, and Az…

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +4
Target Protein:
HTH-type transcriptional regulator QacRSerine protease 1Diamine oxidase [copper-containing] +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dinaciclib DB12021
small molecule | CAS: 779353-01-4

Dinaciclib has been used in trials studying the treatment of rrMM, rrCLL, rrDLBCL, Solid Tumors, and Solid Neoplasm, among others.

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingPyridines
Target Protein:
Cyclin-dependent kinase 9Cyclin-dependent kinase 2Cyclin-dependent kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 311768-81-7

Dinalbuphine sebacate is under investigation in clinical trial NCT02468128 (A Study of Intramuscular Sebacoyl Dinalbuphine Ester for Post-Hemorrhoidectomy Pain Management).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dinoprost Approved DB12789
small molecule | CAS: 551-11-1

Dinoprost has been investigated in Headache.

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAutacoids +11
Target Protein:
Prostaglandin F2-alpha receptorThromboxane A2 receptorProstaglandin E2 receptor EP1 subtype +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dinoprost tromethamine Approved DB01160
small molecule | CAS: 38562-01-5

The tromethamine (THAM) salt of the naturally occurring prostaglandin F2 alpha, dinoprost tromethamine occurs as a white to off-white, very hygroscopic, crystalline powder. Dinoprost tromethamine may also be known as dinoprost trometamol, PGF2 alpha THAM, or …

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAngiography +11
Target Protein:
Prostaglandin F2-alpha receptorProstacyclin receptor
Waktu ParuhThe half-life of di…
Vol. Distribusi-
Klirens-
Genetik -
Dinoprostone Approved DB00917
small molecule | CAS: 363-24-6

Dinoprostone is a naturally occurring prostaglandin E2 (PGE2). It has important effects in labour. It also stimulates osteoblasts to release factors which stimualtes bone resorption by osteoclasts. As a prescription drug it is used as a vaginal suppository, t…

Kategori:
AutacoidsBiological FactorsDinoprostone, antagonists & inhibitors +19
Target Protein:
Prostaglandin F2-alpha receptorProstaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype +3
Waktu ParuhLess than 5 minutes.
Vol. Distribusi-
Klirens-
Genetik -
Dioctyldimonium Approved DB13970
small molecule | CAS: 20256-55-7

Deskripsi belum tersedia.

Kategori:
AminesAmmonium CompoundsNitrogen Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diodone DB13568
small molecule | CAS: 300-37-8

Deskripsi belum tersedia.

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diosmetin DB11259
small molecule | CAS: 520-34-3

Diosmetin is an O-methylated flavone and the aglycone part of the flavonoid glycosides diosmin that occurs naturally in citrus fruits [A27231]. Pharmacologically, diosmetin is reported to exhibit anticancer, antimicrobial, antioxidant, oestrogenic and anti-in…

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cytochrome P450 1B1Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diosmin Approved DB08995
small molecule | CAS: 520-27-4

Chronic venous insufficiency is a common condition the western population. Compression and pharmacotherapy are frequently used to manage chronic venous insufficiency, improving circulation and symptoms of venous disease.[A232885] Diosmin is a bioflavonoid …

Kategori:
BenzopyransCapillary Stabilizing AgentsChromones +15
Target Protein:
Aryl hydrocarbon receptor
Waktu ParuhDiosmin half-life r…
Vol. DistribusiA pharmacokinetic s…
Klirens-
Genetik -
small molecule | CAS: 467-86-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dioxybenzone Approved DB11221
small molecule | CAS: 131-53-3

Dioxybenzone, or benzophenone-8, is an organic compound derived from [DB01878] that is used as a sunscreen agent. It absorbed UV-B and UV-AII rays. Dioxybenzone is an approved sunscreen ingredient in concentrations up to 3% [L2525].

Kategori:
Benzene DerivativesKetonesSunscreen Agents
Target Protein:
Sex hormone-binding globulin
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Diperodon DB11513
small molecule | CAS: 101-08-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphemanil Approved DB13720
small molecule | CAS: 15394-62-4

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Asthmatic Agents +9
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphenhydramine Approved DB01075
small molecule | CAS: 58-73-1

Diphenhydramine - perhaps known most commonly as its brand name formulation Benadryl - is a first-generation H1 receptor antihistamine that is used extensively for the treatment of seasonal allergies, insect bites and stings, and rashes [L5263, L5266, L5269, …

Kategori:
Agents producing tachycardiaAminesAminoalkyl Ethers +41
Target Protein:
Histamine N-methyltransferaseHistamine H1 receptorMuscarinic acetylcholine receptor M2
Waktu ParuhThe elimination hal…
Vol. DistribusiDiphenhydramine is …
KlirensValues for plasma c…
Genetik -
Diphenoxylate Approved DB01081
small molecule | CAS: 915-30-0

A meperidine congener used as an antidiarrheal, usually in combination with atropine. At high doses, it acts like morphine. Its unesterified metabolite difenoxin has similar properties and is used similarly. It has little or no analgesic activity. This medica…

Kategori:
Alimentary Tract and MetabolismAnalgesicsAntidiarrheals +11
Target Protein:
Mu-type opioid receptorDelta-type opioid receptor
Waktu Paruh12-14 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117-34-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicPhenylacetates
Target Protein:
Cathepsin B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 244-54-2

An NADPH oxidase 2 (NOX2) inhibitor.[A252987]

Kategori:
Blood Glucose Lowering AgentsEnzyme InhibitorsNitric Oxide Synthase, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphthamide DB03223
small molecule | CAS: 75645-22-6

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins
Target Protein:
Elongation factor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipivefrin Approved DB00449
small molecule | CAS: 52365-63-6

Dipivefrin is a prodrug of adrenaline, which is used to treat glaucoma. It is available as ophthalmic solution (eye drops).

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +24
Target Protein:
Beta-1 adrenergic receptorAlpha-1A adrenergic receptorAlpha-2A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4701–4750 dari 12560
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