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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 95 / 282
CNM-Au8 DB17952
biotech

Deskripsi belum tersedia.

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CNS-5161 DB05824
small molecule

CNS 5161 is a blocker of the NMDA ion channel and has completed Phase IIa proof of concept clinical trials as a novel compound for the treatment of neuropathic pain.

Target Protein:
Glutamate receptor ionotropic, NMDA 1
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CNV-2197944 DB15229
small molecule | CAS: 1204535-44-3

CNV-2197944 is under investigation in clinical trial NCT01893125 (Efficacy and Safety of CNV2197944 Versus Placebo in Patients With Diabetic Peripheral Neuropathy).

Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1B
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small molecule

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serotonin N-acetyltransferase
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Coagulation Factor IX Human Approved DB13152
biotech | CAS: 181054-95-5

Factor IX (or Christmas factor) is one of the serine proteases of the coagulation system; it belongs to peptidase family S1. Deficiency of this protein causes hemophilia B.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours.
Vol. Distribusi-
Klirens8.62 ± 1.7.
Genetik -
biotech | CAS: 102786-61-8

Recombinant human coagulation Factor VIIa (rFVIIa), intended for promoting hemostasis by activating the extrinsic pathway of the coagulation cascade. NovoSeven is a vitamin K-dependent glycoprotein consisting of 406 amino acid residues. Cloned and expressed i…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +15
Target Protein:
Coagulation factor XTissue factor
Waktu Paruh-
Vol. Distribusi* 121 ± 30 mL/kg [a…
Klirens* 33 - 37 mL/h x kg…
Genetik -
Coagulation factor X human Approved DB13148
biotech

Coagulation Factor X (Human), is a plasma-derived human blood coagulation factor is used by adults and children (aged 12 years and above) with hereditary Factor X deficiency. However its use is limited in the perioperative setting for the management of bleedi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
biotech | CAS: 9013-55-2

Coagulation factor XIa is under investigation in clinical trial NCT01701947 (HEMOLEVEN® Expanded Access Program Prevention of Surgical/Postpartum Hemorrhage Severe Inherited Factor XI Deficiency).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +11
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Coagulin-B DB17703
biotech

Coagulin-B is an adeno-associated viral vector expressing human blood-coagulation Factor IX.[A259038, A259043] It was previously investigated for the treatment of hemophilia; however, the manufacturing company discontinued the Phase I trial in 2004, halting i…

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Coal tar Approved DB11082
small molecule | CAS: 8007-45-2

Coal tar is a brown or black liquid of extremely high viscosity. Coal tar is among the by-products when coal is carbonized to make coke or gasified to make coal gas. Coal tars are complex and variable mixtures of phenols, polycyclic aromatic hydrocarbons (PAH…

Kategori:
Complex MixturesDermatologicalsKeratolytic Agents +2
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Cobalt Approved DB14574
small molecule | CAS: 7440-48-4

A trace element that is a component of vitamin B12. It has the atomic symbol Co, atomic number 27, and atomic weight 58.93. It is used in nuclear weapons, alloys, and pigments. Deficiency in animals leads to anemia; its excess in humans can lead to erythrocyt…

Kategori:
Cell-mediated ImmunityDiet, Food, and NutritionElements +9
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Cobalt chloride Approved DB14206
small molecule | CAS: 7646-79-9

Deskripsi belum tersedia.

Kategori:
Antimutagenic AgentsCompounds used in a research, industrial, or household settingElements +4
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Cobalt Co-60 DB15374
small molecule | CAS: 10198-40-0

Cobalt Co-60 is under investigation in clinical trial NCT02891083 (Adjuvant Therapies or Surgery Alone for High Risk pN0 Esophageal Cancer).

Kategori:
Cobalt IsotopesElementsIsotopes +4
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small molecule | CAS: 22541-53-3

Deskripsi belum tersedia.

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small molecule | CAS: 10124-43-3

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Heavy +1
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Cobamamide DB11191
small molecule | CAS: 13870-90-1

Cobamamide is one of the active forms of vitamin B12 that is also known as _adenosylcobalamin_ or _dibencozide_. This drug is available as a nutritional supplement to prevent vitamin B12 deficiency. Vitamin B12 is a collective term for these variously subs…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCoenzymes +6
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Cobicistat Approved DB09065
small molecule | CAS: 1004316-88-4

Cobicistat, marketed under the name Tybost (formerly GS-9350), indicated for treating infection with human immunodeficiency virus (HIV). Although it does not have any anti-HIV activity, cobicistat acts as a pharmacokinetic enhancer by inhibiting cytochrome P4…

Kategori:
Acids, AcyclicAnti-HIV AgentsAnti-Infective Agents +29
Target Protein:
Cytochrome P450 3A4Cytochrome P450 3A5Cytochrome P450 3A7
Waktu ParuhThe terminal plasma…
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Cobimetinib Approved DB05239
small molecule | CAS: 934660-93-2

Cobimetinib is an orally active, potent and highly selective small molecule inhibiting mitogen-activated protein kinase kinase 1 (MAP2K1 or MEK1), and central components of the RAS/RAF/MEK/ERK signal transduction pathway. It has been approved in Switzerland a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2D6 Inhibitors +22
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe estimated appar…
KlirensFollowing oral admi…
Genetik -
Cobiprostone DB05514
small molecule | CAS: 333963-42-1

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +4
Target Protein:
Chloride channel protein 2
Waktu Paruh-
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Cobitolimod DB14819
biotech | CAS: 1226822-98-5

Cobitolimod is under investigation in clinical trial NCT03178669 (The Efficacy of Cobitolimod in Patients With Moderate to Severe Active Ulcerative Colitis).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
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Coblopasvir DB15315
small molecule | CAS: 1312608-46-0

Coblopasvir is under investigation in clinical trial NCT03416491 (Safety and Efficacy of KW-136 and Sofosbuvir for Treatment of Chronic Hepatitis C).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +2
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biotech | CAS: 2364477-18-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Cobolimab DB16372
biotech | CAS: 2022215-65-0

Cobolimab is under investigation in clinical trial NCT04655976 (Study of Cobolimab in Combination With Dostarlimab and Docetaxel in Advanced NSCLC Participants).

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Cobomarsen DB14931
biotech | CAS: 1848257-52-2

Cobomarsen is under investigation in clinical trial NCT02580552 (Safety, Tolerability and Pharmacokinetics of MRG-106 in Patients With Mycosis Fungoides (MF), CLL, DLBCL or ATLL).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
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Cocaine Approved DB00907
small molecule | CAS: 50-36-2

An alkaloid ester extracted from the leaves of plants including coca. It is a local anesthetic and vasoconstrictor and is clinically used for that purpose, particularly in the eye, ear, nose, and throat. It also has powerful central nervous system effects sim…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlkaloids +36
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium channel protein +5
Waktu Paruh1 hour
Vol. Distribusi-
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biotech

RBP-8000 is under investigation in clinical trials (A Randomized, 4-sequence, 2-period, Double-blind, Placebo Controlled Study With a DSM-IV-TR Diagnosis of Cocaine Abuse) for the treatment of Cocaine Abuse.

Kategori:
Amino Acids, Peptides, and ProteinsEnzymesEnzymes and Coenzymes +3
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biotech

Coccidioides immitis spherule is a skin test antigen indicated to detect delayed-type hypersensitivity to Coccidioides immitis in individuals with a history of pulmonary coccidioidomycosis.

Kategori:
Cell-mediated ImmunitySkin Test Antigen
Target Protein:
HLA-DRHLA class I histocompatibility antigen, A-3 alpha chainHLA class I histocompatibility antigen, B-27 alpha chain
Waktu Paruh-
Vol. DistribusiNot absorbed system…
Klirens-
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small molecule | CAS: 61791-31-9

Deskripsi belum tersedia.

Kategori:
AlcoholsAllergensAmines +3
Waktu Paruh-
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Cocoa butter Approved DB11086
biotech | CAS: 8002-31-1

Cocoa butter is an edible natural fat obtained from the _Theobroma cocoa_ seeds that is predominantly found in dark chocolate [A33033]. It is a rich source of monounsaturated and saturated fatty acids [A33040] that mainly contains approximately 33% [DB04224],…

Kategori:
Antipruritics and Local AnestheticsDiet, Food, and NutritionFats +3
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Coconut Approved DB10523
biotech

Coconut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Coconut oil DB14322
biotech | CAS: 8001-31-8

Coconut oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsDietary FatsFats +4
Waktu Paruh-
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Cod liver oil DB11321
small molecule | CAS: 8001-69-2

Cod liver oil is extracted from the liver of cod fish and mainly consists of omega-3 fatty acids, eicosapentaenoic acid (EPA) and docosahexaenoic acid (DHA). Also being a rich source of vitamin A and D, cod liver oil can be taken orally as daily supplements. …

Kategori:
Diet, Food, and NutritionDietary FatsDietary Fats, Unsaturated +8
Waktu ParuhAs cod liver oil co…
Vol. DistribusiAs cod liver oil co…
KlirensAs cod liver oil co…
Genetik -
CODA-001 DB14915
biotech | CAS: 1605326-11-1

CODA-001 is under investigation in clinical trial NCT01165450 (Efficacy and Safety Study of Nexagon for Persistent Corneal Epithelial Defects).

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Codeine Approved DB00318
small molecule | CAS: 76-57-3

The relief of pain (analgesia) is a primary goal for enhancing the quality of life of patients and for increasing the ability of patients to engage in day to day activities. Codeine, an opioid analgesic, was originally approved in the US in 1950 and is a drug…

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +26
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhPlasma half-lives o…
Vol. DistribusiApparent volume of …
KlirensRenal clearance of …
Genetik 9 Varian
small molecule | CAS: 125-27-9

Deskripsi belum tersedia.

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Codrituzumab DB14843
biotech | CAS: 1365267-33-9

Codrituzumab is under investigation in clinical trial NCT01507168 (A Study of RO5137382 (GC33) in Patients With Advanced or Metastatic Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Coenzyme A DB01992
small molecule | CAS: 85-61-0

Coenzyme A (CoA, CoASH, or HSCoA) is a coenzyme, well known for it's role in the synthesis and oxidation of fatty acids, and the oxidation of pyruvate in the citric acid cycle. All genomes sequenced to date encode enzymes that use coenzyme A as a substrate, a…

Kategori:
Adenine NucleotidesCoenzyme A, biosynthesisCoenzymes +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseCarnitine O-acetyltransferaseGalactoside O-acetyltransferase +42
Waktu Paruh-
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small molecule | CAS: 81918-99-2

Coenzyme A persulfide is a possible in vivo inhibitor of mammalian short chain acyl-CoA dehydrogenase.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isovaleryl-CoA dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme F420 DB03913
small molecule | CAS: 64885-97-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Coenzyme M Approved DB09110
small molecule | CAS: 3375-50-6

Coenzyme M (commonly known by its salt form, Mesna) is a synthetic sulfhydryl (thiol) compound and is used for prophylaxis of Ifosfamide and cyclophosphamide induced hemorrhagic cystitis.[A18572]

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +12
Waktu ParuhThe elimination hal…
Vol. DistribusiVd = 0.652 ± 0.242 …
KlirensPlasma clearance of…
Genetik -
Coffee bean Approved DB10525
biotech

Coffee bean allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Cofirasersen DB19037
biotech | CAS: 2247669-96-9

Cofirasersen is under investigation in clinical trial NCT04441788 (A Study to Assess the Safety, Tolerability, and Efficacy of ION-827359 in Participants With Mild to Moderate Chronic Obstructive Pulmonary Disease (COPD) With Chronic Bronchitis (CB)).

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Col-118 DB05778
small molecule

COL-118, a topical compound based on the SansRosa technology, for the treatment of redness associated with rosacea and other skin disorders. It is a believed to reduce erythema by constricting enlarged blood vessels in facial tissue. Col-118 is a unique formu…

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Vol. Distribusi-
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Col-Treg DB18451
biotech

Col-Treg is an autologous T-cell therapy comprising type I regulatory T-cells specific for human type II collagen.[A261635]

Waktu Paruh-
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Colchiceine Approved DB15534
small molecule | CAS: 477-27-0

Colchiceine is one of several metabolites of the anti-gout medication [colchicine].[A192714]

Kategori:
AlkaloidsColchicine DerivativesTubulin Inhibiting Agent
Target Protein:
Tubulin beta chainTubulin alpha-1A chain
Waktu Paruh-
Vol. Distribusi-
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Colchicine Approved DB01394
small molecule | CAS: 64-86-8

Colchicine is an alkaloid drug derived from a plant belonging to the Lily family, known as _Colchicum autumnale_, or "autumn crocus."[A183611] Its use was first approved by the FDA in 1961.[L8192] Colchicine is used in the treatment of gout flares and Familia…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntigout Preparations +23
Target Protein:
Tubulin beta chain
Waktu ParuhAfter several doses…
Vol. DistribusiThe mean apparent v…
KlirensIn one pharmacokine…
Genetik -
Coleneuramide DB14932
small molecule | CAS: 204200-47-5

Coleneuramide is under investigation in clinical trial NCT00307749 (Safety and Efficacy of MCC-257 in the Treatment of Diabetic Polyneuropathy).

Kategori:
Acids, AcyclicAmino SugarsCarbohydrates +3
Waktu Paruh-
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Colesevelam Approved DB00930
small molecule | CAS: 182815-43-6

Colesevelam is a bile acid sequestrant. Colesevelam is used with exercise and diet changes (restriction of cholesterol and fat intake) to reduce the amount of cholesterol and certain fatty substances in the blood. It works by binding bile acids in the intesti…

Kategori:
AlkenesAllyl CompoundsAllylamine +11
Target Protein:
Bile acids
Waktu Paruh-
Vol. Distribusi-
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Colestilan chloride Approved DB11634
small molecule | CAS: 95522-45-5

Colestilan is an ingredient in the EMA-withdrawn product BindRen.

Kategori:
Drugs for Treatment of Hyperkalemia and HyperphosphatemiaFused-Ring CompoundsSteroids
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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