Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 94 / 236
Elebsiran DB19018
biotech | CAS: 2648009-64-5

Elebsiran is under investigation in clinical trial NCT05461170 (SOLSTICE: Combination Therapy for the Treatment of Chronic Hepatitis D Infection.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eleclazine DB12394
small molecule | CAS: 1443211-72-0

Eleclazine has been used in trials studying the treatment of LQT2 Syndrome, Long QT Syndrome, Ischemic Heart Disease, Ventricular Arrhythmia, and Long QT Syndrome Type 3, among others.

Kategori:
Azepines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elenestinib DB18489
small molecule | CAS: 2505078-08-8

Elenestinib is a selective KIT inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elesclomol DB05719
small molecule | CAS: 488832-69-5

Elesclomol is a novel, injectable, drug candidate that kills cancer cells by elevating oxidative stress levels beyond a breaking point, triggering programmed cell death. In preclinical models elesclomol showed potent killing of a broad range of cancer cell ty…

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elexacaftor Approved DB15444
small molecule | CAS: 2216712-66-0

Elexacaftor (previously VX-445) is a small molecule, next-generation corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) protein.[A187361] It received FDA approval in October 2019 in combination with [tezacaftor] and [ivacaftor] as the…

Kategori:
Cystic Fibrosis Transmembrane Conductance Regulator CorrectorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Elezanumab DB15240
biotech | CAS: 1791416-49-3

Elezanumab is under investigation in clinical trial NCT03737812 (A Study to Assess the Safety and Efficacy of Elezanumab When Added to Standard of Care in Progressive Forms of Multiple Sclerosis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elgemtumab DB15430
biotech | CAS: 1512559-37-3

Elgemtumab is under investigation in clinical trial NCT02167854 (Open-Label Study Evaluating the Safety and Tolerability of LJM716, BYL719 and Trastuzumab in Patients With Metastatic HER2+ Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eliglustat Approved DB09039
small molecule | CAS: 491833-29-5

Eliglustat is a glucosylceramide synthase inhibitor used for the long-term treatment of type 1 Gaucher disease.[A3752,L41404] Gaucher disease is a rare genetic disorder characterized by the deficiency of acid ?-glucosidase, an enzyme that converts glucosylcer…

Kategori:
Alimentary Tract and MetabolismCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +15
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhEliglustat has a te…
Vol. DistribusiIn CYP2D6 extensive…
KlirensIn healthy CYP2D6 e…
Genetik -
Elimusertib DB19041
small molecule | CAS: 1876467-74-1

Elimusertib is under investigation in clinical trial NCT05071209 (Elimusertib for the Treatment of Relapsed or Refractory Solid Tumors).

Target Protein:
Serine/threonine-protein kinase ATR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elinzanetant DB18968
small molecule | CAS: 929046-33-3

Elinzanetant is under investigation in clinical trial NCT05099159 (A Study to Learn More About How Well Elinzanetant Works and How Safe It Is for the Treatment of Vasomotor Symptoms (Hot Flashes) That Are Caused by Hormonal Changes Over 26 Weeks in Women Who …

Target Protein:
Neuromedin-K receptorSubstance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elismetrep DB15287
small molecule | CAS: 1400699-64-0

Elismetrep is under investigation in clinical trial NCT02429102 (A Study to Investigate the Safety, Tolerability and Pharmacokinetics of MT-8554 in Healthy Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elivaldogene autotemcel Approved DB16746
biotech

Elivaldogene autotemcel is a gene therapy consisting of genetically modified autologous cells. It is used to provide functional copies of human adrenoleukodystrophy protein (ALDP) in patients with adrenoleukodystrophy,[L39491] an X-linked genetic disorder cha…

Kategori:
Alimentary Tract and MetabolismCellular and Gene TherapyVarious Alimentary Tract and Metabolism Products
Waktu ParuhAs elivaldogene aut…
Vol. DistribusiAs elivaldogene aut…
KlirensAs elivaldogene aut…
Genetik -
biotech | CAS: 1905397-73-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ellagic acid DB08846
small molecule | CAS: 476-66-4

Ellagic acid is present in several fruits such as cranberries, strawberries, raspberries, and pomegranates. In pomegranates, there are several therapeutic compounds but ellagic acid is the most active and abundant. Ellagic acid is also present in vegetables. …

Kategori:
BenzopyransCytochrome P-450 CYP2E1 InhibitorsCytochrome P-450 CYP2E1 Inhibitors (strength unknown) +6
Target Protein:
Heat shock 70 kDa protein 1AHeat shock 70 kDa protein 1BGlycogen synthase kinase-3 beta +17
Waktu Paruh-
Vol. Distribusi-
KlirensEllagic acid is eli…
Genetik -
Ellipticine DB17026
small molecule | CAS: 519-23-3

Ellipticine is a potent antineoplastic agent.[A252992]

Kategori:
AlkaloidsAntineoplastic AgentsCarbazoles +8
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elobixibat DB12486
small molecule | CAS: 439087-18-0

Elobixibat has been used in trials studying the treatment and basic science of Dyslipidemia, Constipation, Chronic Constipation, Functional Constipation, and Chronic Idiopathic Constipation.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAzepines +5
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elocalcitol DB06194
small molecule | CAS: 199798-84-0

Elocalcitol is a calcitriol analog for inhibition of prostate cell growth; in phase II clinical trial in patients with benign prostate hyperplasia (4/2004).

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elotuzumab Approved DB06317
biotech | CAS: 915296-00-3

Elotuzumab is a humanized IgG1 (Immunoglobulin G) monoclonal antibody indicated in combination with lenalidomide and dexamethasone for the treatment of patients with multiple myeloma who have received one to three prior therapies. Elotuzumab targets SLAMF7, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
SLAM family member 7
Waktu Paruh-
Vol. Distribusi-
KlirensThe clearance of el…
Genetik -
Elraglusib DB16047
small molecule | CAS: 1034895-42-5

Elraglusib is under investigation in clinical trial NCT04218071 (Actuate 1901: 9-ING-41 in Myelofibrosis).

Target Protein:
Glycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elranatamab Approved DB15395
biotech | CAS: 2408850-14-4

Elranatamab is a bispecific B-cell maturation antigen (BCMA)-directed CD3 T-cell engager. It is a humanized immunoglobulin 2-alanine kappa antibody derived from two monoclonal antibodies (mAbs), an anti-BCMA mAb and an anti-CD3 mAb,[A261060] each of which con…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific B-cell maturation antigen (BCMA)-directed CD3 T-cell engager +5
Target Protein:
Tumor necrosis factor receptor superfamily member 17T-cell surface glycoprotein CD3
Waktu ParuhThe mean (CV%) half…
Vol. DistribusiThe mean (CV%) stea…
KlirensThe mean (CV%) clea…
Genetik -
Elsamitrucin DB05129
small molecule | CAS: 97068-30-9

The cytostatic agent Elsamitrucin is a new fermentation product active in a variety of in vivo tumor models of murine and human origin. (PMID: 8150873)

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsCarbohydrates +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA +1
Waktu Paruh36–60 h
Vol. Distribusi-
Klirens-
Genetik -
Elsubrutinib DB18850
small molecule | CAS: 1643570-24-4

Elsubrutinib is under investigation in clinical trial NCT04451772 (A Study of the Safety of Oral Elsubrutinib Capsules and Oral Upadacitinib Tablets Given Alone or in Combination (ABBV-599) for Adult Participants With Moderately to Severely Active Systemic Lu…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elsulfavirine DB14929
small molecule | CAS: 868046-19-9

Elsulfavirine is under investigation in clinical trial NCT03706898 (Study to Evaluate the Safety and PK of Elpida® in Healthy Subjects and Patients With Hepatic Impairment and to Assess the Impact of Food Intake and Drug-Drug Interactions With Other Antiviral…

Kategori:
AmidesAminesAniline Compounds +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltanexor DB16153
small molecule | CAS: 1642300-52-4

Eltanexor is under investigation in clinical trial NCT02649790 (Study of the Safety, Tolerability and Efficacy of KPT-8602 in Patients With Relapsed/refractory Cancer Indications).

Target Protein:
Exportin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltrekibart DB19017
biotech | CAS: 2484883-56-7

Eltrekibart is under investigation in clinical trial NCT06046729 (A Study of Eltrekibart (LY3041658) in Adult Participants With Moderate to Severe Hidradenitis Suppurativa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltrombopag Approved DB06210
small molecule | CAS: 496775-61-2

Eltrombopag is used to treat low blood platelet counts in adults with chronic immune (idiopathic) thrombocytopenia (ITP), when certain other medicines, or surgery to remove the spleen, have not worked well enough. ITP is a condition that may cause unusual bru…

Kategori:
Acids, CarbocyclicBCRP/ABCG2 InhibitorsBenzene Derivatives +25
Target Protein:
Thrombopoietin receptor
Gen Terkait:
F5 SERPINC1
Waktu ParuhAbout 21-32 hours i…
Vol. DistribusiBased on a radiolab…
Klirens-
Genetik 2 Varian
Elubrixin DB12135
small molecule | CAS: 688763-64-6

Elubrixin has been used in trials studying the treatment of Cystic Fibrosis, Colitis, Ulcerative, and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AmidesBenzene DerivativesReceptors, Interleukin-8B, antagonists & inhibitors +2
Target Protein:
C-X-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluforsen DB16154
biotech | CAS: 2101868-82-8

Eluforsen is under investigation in clinical trial NCT02532764 (Dose Escalation Study of QR-010 in Homozygous ?F508 Cystic Fibrosis Patients).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluvixtamab DB17252
biotech | CAS: 1679391-73-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluxadoline Approved DB09272
small molecule | CAS: 864821-90-9

Eluxadoline is a mixed mu-opioid receptor agonist, kappa-opioid receptor agonist, and a-delta opioid receptor antagonist indicated for use in diarrhea-predominant irritable bowel syndrome (IBS-D). The mu-, kappa-, and delta-opioid receptors mediate endogenous…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +15
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhThe mean plasma eli…
Vol. Distribusi-
Klirens-
Genetik -
Elvitegravir Approved DB09101
small molecule | CAS: 697761-98-1

Elvitegravir is a human immunodeficiency virus type 1 (HIV-1) integrase strand transfer inhibitor (INSTI) used for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults. Because integrase is necessary for viral replication, inhibitio…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +22
Target Protein:
IntegraseGag-Pol polyprotein
Waktu ParuhThe median terminal…
Vol. Distribusi-
Klirens-
Genetik -
Elvucitabine DB06236
small molecule | CAS: 181785-84-2

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +13
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ELX-02 DB15080
small molecule | CAS: 1375073-95-2

ELX-02 is under investigation in clinical trial NCT03309605 (Phase 1 Study of ELX-02 in Healthy Adult Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elzasonan DB18969
small molecule | CAS: 361343-19-3

Elzasonan is under investigation in clinical trial NCT00275197 (A Research Study to Compare the Treatments of a Combination of Elzasonan With Zoloft, to Zoloft Alone, or Placebo in People With Major Depressive Disorder (MDD)).

Kategori:
Oxazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elzovantinib DB18918
small molecule | CAS: 2271119-26-5

Elzovantinib is under investigation in clinical trial NCT03993873 (Study of TPX-0022 in Patients With Advanced NSCLC, Gastric Cancer or Solid Tumors Harboring Genetic Alterations in MET).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EM-1745 DB02323
small molecule

Deskripsi belum tersedia.

Kategori:
17-Hydroxysteroid Dehydrogenases, antagonists & inhibitorsEstradiol CongenersEstranes +7
Target Protein:
17-beta-hydroxysteroid dehydrogenase type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emactuzumab DB14905
biotech | CAS: 1448221-67-7

Emactuzumab is under investigation in clinical trial NCT01494688 (A Study of RO5509554 as Monotherapy and in Combination With Paclitaxel in Participants With Advanced Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emapalumab Approved DB14724
biotech | CAS: 1709815-23-5

Emapalumab, also known as NI-0501, is a fully human monoclonal antibody that targets interferon gamma. Emapalumab development was sponsored by NovImmune SA, further developed by Sobi and FDA approved on November 20, 2018.[A38676, L4840] The approval of emapal…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +14
Target Protein:
Interferon gamma
Waktu ParuhEmapalumab eliminat…
Vol. DistribusiThe central and per…
KlirensEmapalumab clearanc…
Genetik -
Emapunil DB12666
small molecule | CAS: 226954-04-7

Emapunil has been used in trials studying the basic science and diagnostic of Baseline, Blocking Receptor Binding, and Neurodegenerative Disorders.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EMB-01 DB16091
biotech

EMB-01 is under investigation in clinical trial NCT03797391 (A Dose Escalation Study of EMB-01 in Participants With Advanced/metastatic Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Embutramide DB01487
small molecule | CAS: 15687-14-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminesAminobenzoates +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EMD-1201081 DB06181
biotech | CAS: 847484-35-9

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emedastine Approved DB01084
small molecule | CAS: 87233-61-2

Emedastine is an antihistamine used in eye drops to treat allergic conjunctivitis.

Kategori:
Anti-Allergic AgentsDecongestants and AntiallergicsHeterocyclic Compounds, Fused-Ring +9
Target Protein:
Histamine H1 receptor
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Emepronium DB13505
small molecule | CAS: 27892-33-7

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +19
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emerfetamab DB18474
biotech | CAS: 2250261-27-7

Emerfetamab is a bispecific T cell engager antibody construct with a half-life extension Fc moiety capable of binding to the neonatal Fc receptor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 5982-52-5

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emfilermin DB06562
small molecule | CAS: 159075-60-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EMI-137 DB19174
biotech

EMI-137 is under investigation in clinical trial NCT03360461 (EMI-137 in Laparoscopic Colonic Resections).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Emibetuzumab DB11849
biotech | CAS: 1365287-97-3

Emibetuzumab has been used in trials studying the treatment of Advanced Cancer, Renal Cell Carcinoma, Hepatocellular Cancer, Gastric Adenocarcinoma, and Non-Small Cell Lung Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4651–4700 dari 11778
Sebelumnya Halaman 94 / 236 Berikutnya