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11793

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8607 (73.0%)
Target
6418 (54.4%)
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102 (0.9%)
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11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 94 / 236
biotech | CAS: 2567881-77-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enibarcimab DB16730
biotech | CAS: 2305638-98-4

Enibarcimab is under investigation in clinical trial NCT03989531 (Adrecizumab in Cardiogenic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eniluracil DB03516
small molecule | CAS: 59989-18-3

Eniluracil, which was previously under development by GlaxoSmithKline (GSK), is being developed by Adherex to enhance the therapeutic value and effectiveness of 5-fluorouracil (5-FU), one of the world’s most widely-used oncology agents. 5-FU is widely used i…

Kategori:
Enzyme InhibitorsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Aldehyde oxidaseXanthine dehydrogenase/oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enitociclib DB17297
small molecule | CAS: 1610408-97-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-1198 DB05959
small molecule | CAS: 864668-87-1

Deskripsi belum tersedia.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Hypoxia-inducible factor 1-alphaTumor necrosis factor receptor superfamily member 11ASignal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-981693 DB16891
small molecule | CAS: 934353-76-1

Deskripsi belum tersedia.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Enoxacin Approved DB00467
small molecule | CAS: 74011-58-8

A broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Enoxaparin Approved DB01225
small molecule | CAS: 9005-49-6

Enoxaparin is a common low-molecular-weight heparin (LMWH) used in the prevention and management of various thromboembolic disorders. Initially approved by the FDA in 1993, it is administered by a subcutaneous or intravenous injection and marketed by several …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +7
Target Protein:
Antithrombin-IIICoagulation factor XProthrombin
Waktu ParuhThe half-life of en…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Enoximone Approved DB04880
small molecule | CAS: 77671-31-9

Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. It is used in patients with congestive heart failure. Trials were halted in the U.S., but the …

Kategori:
Cardiac Stimulants Excl. Cardiac GlycosidesCardiac TherapyCardiotonic Agents +10
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu Paruh4-10 hours
Vol. Distribusi-
Klirens-
Genetik -
Enpatoran DB16501
small molecule | CAS: 2101938-42-3

Enpatoran (M5049) was under investigation in clinical trials for various conditions. It was investigated for systemic lupus erythematosus and cutaneous lupus erythematosus in completed trials (NCT04647708 and NCT05162586) and in a recruiting trial (NCT0554032…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enprofylline Approved DB00824
small molecule | CAS: 41078-02-8

Enprofylline is a derivative of theophylline which shares bronchodilator properties. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of cerebrovascular insufficiency, sickle cell disease, and diabetic neuropathy. L…

Kategori:
Adenosine A2 Receptor AntagonistsAlkaloidsAnti-Asthmatic Agents +11
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidaseAdenosine receptor A2b +4
Waktu Paruh1.9 hours
Vol. Distribusi-
Klirens-
Genetik -
Enprostil DB13824
small molecule | CAS: 73121-56-9

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsAutacoids +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enrasentan DB06460
small molecule | CAS: 167256-08-8

Deskripsi belum tersedia.

Kategori:
Endothelin Receptor AntagonistsIndenes
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enrofloxacin DB11404
small molecule | CAS: 93106-60-6

Enrofloxacin is an antibiotic agent from the fluoroquinolone family produced by the Bayer Corporation. Enrofloxacin is approved by the FDA for its veterinary use. Due to the identification of fluoroquinolone-resistant strains of _Campylobacter_, in September …

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensartinib DB14860
small molecule | CAS: 1370651-20-9

Ensartinib is under investigation in clinical trial NCT03420508 (Treating Patients With Melanoma and ALK Alterations With Ensartinib).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
ALK tyrosine kinase receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensifentrine Approved DB16157
small molecule | CAS: 1884461-72-6

Ensifentrine is a first-in-class, selective dual inhibitor of the phosphodiesterase 3 (PDE3) and phosphodiesterase 4 (PDE4) enzymes.[L50903] On June 26, 2024, the FDA announced the approval of an inhaled product of ensifentrine for the treatment of chronic o…

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP2D6 Substrates +6
Target Protein:
Phosphodiesterase 3Phosphodiesterase 4
Waktu ParuhFollowing twice-dai…
Vol. DistribusiApparent central an…
Klirens-
Genetik -
Ensitrelvir DB18834
small molecule | CAS: 2647530-73-0

Ensitrelvir is under investigation in clinical trial NCT05605093 (Strategies and Treatments for Respiratory Infections & Viral Emergencies (STRIVE): Shionogi Protease Inhibitor (Ensitrelvir)).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensituximab DB12342
biotech | CAS: 1092658-06-4

Ensituximab has been used in trials studying the treatment of Pancreatic Cancer, Adult, Metastatic Colorectal Cancer, and Metastatic Pancreatic Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensovibep DB19078
biotech | CAS: 2451126-06-8

Ensovibep is under investigation in clinical trial NCT04501978 (ACTIV-3: Therapeutics for Inpatients With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entacapone Approved DB00494
small molecule | CAS: 130929-57-6

Entacapone is a selective, reversible catechol-O-methyl transferase (COMT) inhibitor for the treatment of Parkinson's disease. It is a member of the class of nitrocatechols. When administered concomittantly with levodopa and a decarboxylase inhibitor (e.g., c…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBenzene Derivatives +11
Target Protein:
Catechol O-methyltransferase
Waktu Paruh0.4-0.7 hour
Vol. Distribusi* 20 L
Klirens* 850 mL/min
Genetik -
biotech | CAS: 2247971-01-1

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entecavir Approved DB00442
small molecule | CAS: 142217-69-4

Entecavir is an oral antiviral drug used in the treatment of hepatitis B infection. It is marketed under the trade name Baraclude (BMS). Entecavir is a guanine analogue that inhibits all three steps in the viral replication process, and the manufacturer cl…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
DNA
Waktu ParuhAfter reaching peak…
Vol. Distribusi-
Klirens* renal cl=383.2 +/…
Genetik -
Entolimod DB12304
biotech | CAS: 951628-22-1

Entolimod has been used in trials studying the treatment of Mucositis, Tongue Cancer, Colorectal Cancer, Stage IVA Verrucous Carcinoma of the Larynx, and Stage IVB Verrucous Carcinoma of the Larynx, among others.

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENTR-601-44 DB17836
biotech

ENTR-601-44 is an exon 44 skipping phosphorodiamidate morpholino oligonucleotide (PMO). Developed by Entrada Therapeutics, it was investigated for the treatment of Duchenne muscular dystrophy.[L46641]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entrectinib Approved DB11986
small molecule | CAS: 1108743-60-7

Entrectinib is a tropomyosin receptor tyrosine kinase (TRK) TRKA, TRKB, TRKC, proto-oncogene tyrosine-protein kinase ROS1, and anaplastic lymphoma kinase (ALK) inhibitor.[L8081] It was approved by the FDA in August 2019 for use in the treatment of ROS1-positi…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
ALK tyrosine kinase receptorHigh affinity nerve growth factor receptorNT-3 growth factor receptor +4
Waktu ParuhEntrectinib has a h…
Vol. DistribusiEntrectinib has an …
KlirensThe apparent cleara…
Genetik -
Envafolimab DB15769
biotech | CAS: 2102192-68-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enzacamene Approved DB11219
small molecule | CAS: 36861-47-9

Commonly known as 4-methylbenzylidene-camphor (4-MBC), enzacamene is a camphor derivative and an organic chemical UV-B filter. It is used in cosmetic products such as sunscreen to provide skin protection against UV rays. While its effects on the human reprodu…

Kategori:
Bicyclic MonoterpenesBornanesBridged-Ring Compounds +5
Target Protein:
Progesterone receptorAndrogen receptorEstrogen receptor beta +1
Waktu ParuhThe half life of en…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Enzalutamide Approved DB08899
small molecule | CAS: 915087-33-1

Enzalutamide is an androgen receptor (AR) inhibitor for the treatment of castration-resistant prostate cancer (CRPC), both metastatic and non-metastatic.[L40639] It is a second-generation antiandrogen agent that the FDA approved on August 31, 2012.[L40639, A2…

Kategori:
AmidesAndrogen Receptor AntagonistsAndrogen Receptor Inhibitors +35
Target Protein:
Androgen receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean apparent c…
Genetik -
Enzastaurin DB06486
small molecule | CAS: 170364-57-5

Enzastaurin, an investigational, targeted, oral agent, will be evaluated at more than 100 sites worldwide for the treatment of relapsed glioblastoma multiforme (GBM), an aggressive and malignant form of brain cancer.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C beta typePhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformRAC-alpha serine/threonine-protein kinase +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eosin DB13706
small molecule | CAS: 17372-87-1

Deskripsi belum tersedia.

Kategori:
Antiseptics and DisinfectantsColoring AgentsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EP-0042 DB18120
small molecule | CAS: 1402709-93-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EP-1043 DB06118
biotech

EP-1043 is an epitope-based recombinant protein vaccine designed to induce HIV-1 specific helper T-lymphocyte (HTL) responses. The vaccine consists of a string of 18 HIV-derived major histocompatibility complex (MHC) Class II restricted epitopes, each separat…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EP-2104R DB05675
biotech

EP-2104R is an imaging pharmaceutical under development for the detection of blood clots. It is the first targeted high-resolution technique designed to visualize blood clots directly. It is being developed by EPIX Pharmaceuticals, Inc.

Kategori:
Amino Acids, Peptides, and ProteinsContrast MediaElements +3
Target Protein:
Fibrinogen alpha chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EP-217609 DB18393
small molecule | CAS: 894494-99-6

Deskripsi belum tersedia.

Kategori:
CarbohydratesCoenzymesEnzymes and Coenzymes +2
Target Protein:
Coagulation factor XProthrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epacadostat DB11717
small molecule | CAS: 1204669-58-8

Epacadostat has been used in trials studying the treatment of HL, Melanoma, Glioblastoma, Mucosal Melanoma, and Ovarian Carcinoma, among others.

Kategori:
AmidesAminesAntineoplastic Agents +4
Target Protein:
Indoleamine 2,3-dioxygenase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epafipase DB16158
biotech | CAS: 208576-22-1

Epafipase is under investigation in clinical trial NCT00037687 (Safety and Efficacy of Recombinant Human Platelet-activating Factor Acetylhydrolase for the Treatment of Severe Sepsis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epanolol DB13757
small molecule | CAS: 86880-51-5

Epanolol is an beta blocker.

Kategori:
AcetamidesAdrenergic AgentsAdrenergic Antagonists +18
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epcoritamab Approved DB16672
biotech | CAS: 2134641-34-0

Epcoritamab is an IgG1-bispecific antibody that simultaneously binds to CD3 on T-cells and CD20 on B-cells.[A259736,A258488,A259761,L46516] Epcoritamab promotes the activation and expansion of T-cells and, by being able to bind to both CD20 and CD3, it leads …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +13
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhA full dose of epco…
Vol. DistribusiEpcoritamab has an …
KlirensA full dose of epco…
Genetik -
Epeleuton DB18100
small molecule | CAS: 1667760-39-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eperisone DB08992
small molecule | CAS: 64840-90-0

Eperisone is an antispasmodic drug which relaxes both skeletal muscles and vascular smooth muscles, and demonstrates a variety of effects such as reduction of myotonia, improvement of circulation, and suppression of the pain reflex. It is not approved for use…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAutonomic Agents +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epetraborole DB11744
small molecule | CAS: 1093643-37-8

Epetraborole has been used in trials studying the treatment of Infections, Bacterial, Infections, Intestinal, Infections, Urinary Tract, and Community-acquired Infection.

Kategori:
Anti-Bacterial AgentsLeucine-tRNA Ligase, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Ephedra is an alkaloid chemical compound traditionally obtained from the plant _Ephedra sinica_. The sale of ephedra-containing supplements intended to increase muscle weight or promote weight loss was banned in the United States in 2004 due to the risk for a…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +22
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterAlpha-2A adrenergic receptor +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ephedrine Approved DB01364
small molecule | CAS: 299-42-3

Ephedrine was first described in western literature in 1888, as a naturally occurring component of the ephedra plant, along with [pseudoephedrine].[A193698] Ephedrine acts as both a direct and indirect sympathomimetic. It is an alpha- and beta-adrenergic rece…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +39
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorBeta-1 adrenergic receptor +2
Waktu ParuhOral ephedrine has …
Vol. DistribusiOral ephedrine has …
KlirensOral ephedrine has …
Genetik -
small molecule | CAS: 1082659-36-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EPI-589 DB16041
small molecule | CAS: 1147883-03-1

EPI-589 is under investigation in clinical trial NCT02460679 (Safety and Biomarker Study of EPI-589 in Participants With Amyotrophic Lateral Sclerosis (ALS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epicaptopril DB02032
small molecule | CAS: 63250-36-2

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAmino AcidsAmino Acids, Cyclic +6
Target Protein:
Metallo-beta-lactamase L1Beta-lactamaseOrganic hydroperoxide resistance protein, putative +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epicatechin DB12039
small molecule | CAS: 490-46-0

Epicatechin has been used in trials studying the treatment of Pre-diabetes.

Kategori:
BenzopyransCatechinChromans +4
Target Protein:
Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epicillin DB13300
small molecule | CAS: 26774-90-3

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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