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14361

Total database: 17430
Struktur (SMILES)
9916 (69.0%)
Target
7893 (55.0%)
Genomik
112 (0.8%)
Referensi
14361 (100.0%)

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Hasil Pencarian (14361)

Halaman 93 / 288
Clorotepine DB15971
small molecule | CAS: 13448-22-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur CompoundsThiepins
Target Protein:
5-hydroxytryptamine receptor 2CHistamine H1 receptorAlpha-1B adrenergic receptor +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
biotech

Clostridium tetani toxoid antigen (formaldehyde inactivated) is a vaccine for intramuscular injection. It is used for active immunization of children 7 years of age or older, and adults, for prevention of tetanus. The toxoid in the Clostridium tetani culture …

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBacterial Vaccines +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Clothiapine Approved DB13256
small molecule | CAS: 2058-52-8

Clothiapine has been approved in European countries and is an atypical antipsychotic, shown to be useful in some treatment-resistant patients.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clotiazepam Approved DB01559
small molecule | CAS: 33671-46-4

Clotiazepam is a thienodiazepine, not approved for sale in the U.S. or Canada, but has been approved in the U.K. It is a schedule IV drug in Canada.

Kategori:
Anti-Anxiety AgentsBenzodiazepines and benzodiazepine derivativesCentral Nervous System Depressants +8
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Clotrimazole Approved DB00257
small molecule | CAS: 23593-75-1

This drug is a broad spectrum antimycotic or antifungal agent. Clotrimazole's antimycotic properties were discovered in the late 1960s [A174094]. Clotrimazole falls under the _imidazole_ category of _azole_ antifungals, possessing broad-spectrum antimycotic a…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntifungal Agents +54
Target Protein:
C-X-C chemokine receptor type 2Lanosterol 14-alpha demethylaseIntermediate conductance calcium-activated potassium channel protein 4 +3
Waktu Paruh-
Vol. DistribusiThe topical form is…
Klirens-
Genetik -
Clove Approved DB10672
biotech | CAS: 84961-50-2

Clove allergenic extract is used in allergenic testing.

Kategori:
AngiospermsBiological ProductsCell-mediated Immunity +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clove oil Approved DB11338
biotech | CAS: 8000-34-8

Clove oil is obtained by extraction from the dried flower buds of the clove plant. Traditionally, it has been used as a flavouring spice in foods, or as a fragrance. It is also found in topical analgesics. Clove oil has shown to exert some antimicrobial activ…

Kategori:
Biological ProductsComplex MixturesDrugs that are Mainly Renally Excreted +3
Target Protein:
Vascular cell adhesion protein 1C-X-C motif chemokine 10Collagen alpha-1(I) chain +1
Waktu ParuhIn a pharmacokineti…
Vol. Distribusi-
Klirens-
Genetik -
Cloxacillin Approved DB01147
small molecule | CAS: 61-72-3

A semi-synthetic penicillin antibiotic which is a chlorinated derivative of [oxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacAPenicillin-binding protein 2XPenicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloxazolam DB01553
small molecule | CAS: 24166-13-0

Cloxazolam is a benzodiazepine with anxiolytic, sedative/hypnotic, muscle relaxant, and antiepileptic effects. It is marketed in the Argentina, Australia, Portugal, Belgium, Switzerland, Luxembourg, Germany, Taiwan and Japan -- mainly for anti-anxiety. The us…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +4
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh65 hours
Vol. Distribusi-
Klirens-
Genetik -
Clozapine Approved DB00363
small molecule | CAS: 5786-21-0

Clozapine is a tricyclic dibenzodiazepine, classified as an atypical antipsychotic agent.[A256708] Clozapine displays affinity to various neuroreceptors with a particularly low affinity to the dopamine receptors, thus breaking the mold of first-generation ant…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +65
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AD(1A) dopamine receptor +30
Gen Terkait:
GNB3
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe median volume o…
KlirensThe median clearanc…
Genetik 1 Varian
CLX-0921 DB05854
small molecule

CLX-0921 is investigated for use/treatment in diabetes mellitus type 2. CLX-0921 is a solid. CLX-0921 has a spectrum of activity that differs from commercially available thiazolidinediones. This substance targets the protein peroxisome proliferator-activated …

Kategori:
Sulfur Compounds
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CLZ-2002 DB18638
biotech

CLZ-2002 consists of allogeneic mesenchymal stem cells derived neuronal regeneration-promoting cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CM4620 DB16466
small molecule | CAS: 1713240-67-5

CM4620 (Zegocractin), is under investigation in multiple clinical trials, including NCT04195347 (pancreatitis due to asparaginase), NCT03709342 (PK/PD study in acute pancreatitis), NCT03401190 and NCT04681066 (pancreatitis and SIRS), and NCT04661540 (critical…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMC 001 DB05353
small molecule

CMC 001 is an orally administered MRI contrast agent in development for enhancement of the liver, bile ducts and gastrointestinal tract.

Waktu Paruh-
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Genetik -
CMG901 DB18619
biotech

CMG901 is an anti-Claudin 18.2 monoclonal antibody conjugated with MMAE payload.

Waktu Paruh-
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Genetik -
CMLVAX100 DB05164
biotech

CMLVAX100 is a vaccine targeting the BCR-ABL-derived p210 fusion protein which reduces residual disease in some patients with chronic myeloid leukemia. It is developed by Breakthrough Therapeutics and has completed phase I of its clinical trial.

Target Protein:
BCR/ABL p210 fusion protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
3-deoxy-manno-octulosonate cytidylyltransferase3-deoxy-manno-octulosonate cytidylyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMX-2043 DB12795
small molecule | CAS: 910627-26-8

CMX-2043 has been used in trials studying the treatment and prevention of Non STEMI, Unstable Angina, Stable Coronary Artery Disease, and Percutaneous Coronary Intervention.

Kategori:
Amino Acids, Peptides, and ProteinsCoenzymesEnzymes and Coenzymes +6
Target Protein:
RAC-alpha serine/threonine-protein kinaseHepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CN-105 DB18345
small molecule | CAS: 1632243-07-2

CN-105 is a neuroprotective pentapeptide with the sequence Acetyl-Valine-Serine-Arginine-Arginine-Arginine-NH2 (Ac-VSRRR- NH2).

Waktu Paruh-
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Genetik -
CN-201 DB18726
biotech

CN-201 is a humanized anti-CD3/CD19 bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNDO-109 DB17290
biotech

CNDO-109 are CNDO-109-activated allogeneic natural killer cells.

Waktu Paruh-
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Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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CNS-5161 DB05824
small molecule

CNS 5161 is a blocker of the NMDA ion channel and has completed Phase IIa proof of concept clinical trials as a novel compound for the treatment of neuropathic pain.

Target Protein:
Glutamate receptor ionotropic, NMDA 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNV-2197944 DB15229
small molecule | CAS: 1204535-44-3

CNV-2197944 is under investigation in clinical trial NCT01893125 (Efficacy and Safety of CNV2197944 Versus Placebo in Patients With Diabetic Peripheral Neuropathy).

Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serotonin N-acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serotonin N-acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serotonin N-acetyltransferase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 181054-95-5

Recombinant Coagulation Factor IX is a purified Factor IX glycoprotein produced by recombinant DNA technology. It has a primary amino acid sequence that is identical to the Ala148 allelic form of human factor IX, and has structural and functional characterist…

Kategori:
Blood Coagulation FactorsHemostaticsIncreased Coagulation Activity
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours
Vol. Distribusi-
Klirens8.62 ± 1.7
Genetik -
Coagulation Factor IX Human Approved DB13152
biotech | CAS: 181054-95-5

Factor IX (or Christmas factor) is one of the serine proteases of the coagulation system; it belongs to peptidase family S1. Deficiency of this protein causes hemophilia B.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours.
Vol. Distribusi-
Klirens8.62 ± 1.7.
Genetik -
Coagulation factor VII human Approved DB13150
biotech

Coagulation factor VII is human serine protease type enzyme that is involved in the extrinsic coagulation cascade which results in blood clotting.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Tissue factorCoagulation factor XCoagulation factor IX
Waktu Paruh5 h
Vol. Distribusi45 ml/kg
Klirens7.4 ml/kgh
Genetik -
biotech | CAS: 102786-61-8

Recombinant human coagulation Factor VIIa (rFVIIa), intended for promoting hemostasis by activating the extrinsic pathway of the coagulation cascade. NovoSeven is a vitamin K-dependent glycoprotein consisting of 406 amino acid residues. Cloned and expressed i…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +15
Target Protein:
Coagulation factor XTissue factor
Waktu Paruh-
Vol. Distribusi* 121 ± 30 mL/kg [a…
Klirens* 33 - 37 mL/h x kg…
Genetik -
Coagulation factor X human Approved DB13148
biotech

Coagulation Factor X (Human), is a plasma-derived human blood coagulation factor is used by adults and children (aged 12 years and above) with hereditary Factor X deficiency. However its use is limited in the perioperative setting for the management of bleedi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
biotech | CAS: 9013-55-2

Coagulation factor XIa is under investigation in clinical trial NCT01701947 (HEMOLEVEN® Expanded Access Program Prevention of Surgical/Postpartum Hemorrhage Severe Inherited Factor XI Deficiency).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coagulin-B DB17703
biotech

Coagulin-B is an adeno-associated viral vector expressing human blood-coagulation Factor IX.[A259038, A259043] It was previously investigated for the treatment of hemophilia; however, the manufacturing company discontinued the Phase I trial in 2004, halting i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coal tar Approved DB11082
small molecule | CAS: 8007-45-2

Coal tar is a brown or black liquid of extremely high viscosity. Coal tar is among the by-products when coal is carbonized to make coke or gasified to make coal gas. Coal tars are complex and variable mixtures of phenols, polycyclic aromatic hydrocarbons (PAH…

Kategori:
Complex MixturesDermatologicalsKeratolytic Agents +2
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Cobalt Approved DB14574
small molecule | CAS: 7440-48-4

A trace element that is a component of vitamin B12. It has the atomic symbol Co, atomic number 27, and atomic weight 58.93. It is used in nuclear weapons, alloys, and pigments. Deficiency in animals leads to anemia; its excess in humans can lead to erythrocyt…

Kategori:
Cell-mediated ImmunityDiet, Food, and NutritionElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobalt Co-60 DB15374
small molecule | CAS: 10198-40-0

Cobalt Co-60 is under investigation in clinical trial NCT02891083 (Adjuvant Therapies or Surgery Alone for High Risk pN0 Esophageal Cancer).

Kategori:
Cobalt IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobamamide DB11191
small molecule | CAS: 13870-90-1

Cobamamide is one of the active forms of vitamin B12 that is also known as _adenosylcobalamin_ or _dibencozide_. This drug is available as a nutritional supplement to prevent vitamin B12 deficiency. Vitamin B12 is a collective term for these variously subs…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCoenzymes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobicistat Approved DB09065
small molecule | CAS: 1004316-88-4

Cobicistat, marketed under the name Tybost (formerly GS-9350), indicated for treating infection with human immunodeficiency virus (HIV). Although it does not have any anti-HIV activity, cobicistat acts as a pharmacokinetic enhancer by inhibiting cytochrome P4…

Kategori:
Acids, AcyclicAnti-HIV AgentsAnti-Infective Agents +29
Target Protein:
Cytochrome P450 3A4Cytochrome P450 3A5Cytochrome P450 3A7
Waktu ParuhThe terminal plasma…
Vol. Distribusi-
Klirens-
Genetik -
Cobimetinib Approved DB05239
small molecule | CAS: 934660-93-2

Cobimetinib is an orally active, potent and highly selective small molecule inhibiting mitogen-activated protein kinase kinase 1 (MAP2K1 or MEK1), and central components of the RAS/RAF/MEK/ERK signal transduction pathway. It has been approved in Switzerland a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2D6 Inhibitors +22
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe estimated appar…
KlirensFollowing oral admi…
Genetik -
Cobiprostone DB05514
small molecule | CAS: 333963-42-1

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +4
Target Protein:
Chloride channel protein 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobitolimod DB14819
biotech | CAS: 1226822-98-5

Cobitolimod is under investigation in clinical trial NCT03178669 (The Efficacy of Cobitolimod in Patients With Moderate to Severe Active Ulcerative Colitis).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coblopasvir DB15315
small molecule | CAS: 1312608-46-0

Coblopasvir is under investigation in clinical trial NCT03416491 (Safety and Efficacy of KW-136 and Sofosbuvir for Treatment of Chronic Hepatitis C).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2364477-18-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobolimab DB16372
biotech | CAS: 2022215-65-0

Cobolimab is under investigation in clinical trial NCT04655976 (Study of Cobolimab in Combination With Dostarlimab and Docetaxel in Advanced NSCLC Participants).

Waktu Paruh-
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Genetik -
Cobomarsen DB14931
biotech | CAS: 1848257-52-2

Cobomarsen is under investigation in clinical trial NCT02580552 (Safety, Tolerability and Pharmacokinetics of MRG-106 in Patients With Mycosis Fungoides (MF), CLL, DLBCL or ATLL).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocaine Approved DB00907
small molecule | CAS: 50-36-2

An alkaloid ester extracted from the leaves of plants including coca. It is a local anesthetic and vasoconstrictor and is clinically used for that purpose, particularly in the eye, ear, nose, and throat. It also has powerful central nervous system effects sim…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlkaloids +36
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium channel protein +5
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
biotech

RBP-8000 is under investigation in clinical trials (A Randomized, 4-sequence, 2-period, Double-blind, Placebo Controlled Study With a DSM-IV-TR Diagnosis of Cocaine Abuse) for the treatment of Cocaine Abuse.

Kategori:
Amino Acids, Peptides, and ProteinsEnzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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