Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 93 / 134
Nogapendekin alfa Approved DB18740
biotech | CAS: 1622189-43-8

Nogapendekin alfa is a human IL-15N72D variant. It is one of the active ingredients in Anktiva, a combination product also containing [inbakicept], where a single inbakicept is complexed with two nogapendekin alfa components.[L50592] This combination product …

Kategori:
Amino Acids, Peptides, and ProteinsInterleukin-15Proteins +2
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, muscle formLactase-like proteinLactase/phlorizin hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nolatrexed DB12912
small molecule | CAS: 147149-76-6

Nolatrexed is under investigation in clinical trial NCT00012324 (Nolatrexed Dihydrochloride Compared With Doxorubicin in Treating Patients With Recurrent or Unresectable Liver Cancer).

Kategori:
AntimetabolitesAntineoplastic AgentsEnzyme Inhibitors +5
Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomifensine Approved DB04821
small molecule | CAS: 24526-64-5

Nomifensine, formerly marketed as Merital capsules, was associated with an increased incidence of hemolytic anemia. The approved application holder removed Merital capsules from the market on January 23, 1986. FDA published a notice of its determination that …

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsDopamine Agents +8
Target Protein:
D(2) dopamine receptorSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nonivamide DB11324
small molecule | CAS: 2444-46-4

Nonivamide is found in herbs and spices. It is an alkaloid from the Capsicum species. The structures of [DB06774] and nonivamide differ only slightly with respect to the fatty acid moiety of the side chain (8-methyl nonenoic acid versus nonanoic acid) [F31]. …

Kategori:
Acids, CarbocyclicAlkaloidsAlkenes +20
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhAbout 7 minutes [F3…
Vol. Distribusi-
Klirens-
Genetik -
Nonoxynol-9 Approved DB06804
small molecule | CAS: 26027-38-3

Nonoxynol-9 (N-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives. When present in the vagina during intercourse, they immobilize/inactivate/damage and/or kill sperms without eliciting systemic …

Kategori:
Adrenal Cortex HormonesAlcoholsAntispermatogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NOP-1A DB15208
small molecule | CAS: 1283095-70-4

NOP-1A is under investigation in clinical trial NCT01198197 (PET Brain and Whole Body Distribution Studies for Nociceptin/Orphanin FQ Peptide (NOP) Receptor Using [11C]NOP-1A).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
nor-NOHA DB02381
small molecule | CAS: 189302-40-7

N-Hydroxy-nor-L-arginine (nor-NOHA) is under investigation in clinical trial NCT02009527 (Arginase Inhibition in Ischemia-reperfusion Injury).

Target Protein:
Arginase-2, mitochondrialArginase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nordazepam DB14028
small molecule | CAS: 1088-11-5

An intermediate in the metabolism of DIAZEPAM to OXAZEPAM. It may have actions similar to those of diazepam.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +15
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norepinephrine Approved DB00368
small molecule | CAS: 51-41-2

Precursor of epinephrine that is secreted by the adrenal medulla and is a widespread central and autonomic neurotransmitter. Norepinephrine is the principal transmitter of most postganglionic sympathetic fibers and of the diffuse projection system in the brai…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +34
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norethisterone Approved DB00717
small molecule | CAS: 68-22-4

Norethisterone, also known as norethindrone, is a synthetic progestational hormone belonging to the 19-nortestosterone-derived class of progestins.[A10367] It is further classified as a second-generation progestin, along with [levonorgestrel] and its derivati…

Kategori:
Adrenal Cortex HormonesAnti-Gonadotropin-Releasing HormonesCombination Contraceptives (with Estrogen and derivatives) +34
Target Protein:
Progesterone receptorAndrogen receptorGlucocorticoid receptor
Waktu ParuhThe half-life of no…
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Norfloxacin Approved DB01059
small molecule | CAS: 70458-96-7

A synthetic fluoroquinolone (fluoroquinolones) with broad-spectrum antibacterial activity against most gram-negative and gram-positive bacteria. Norfloxacin inhibits bacterial DNA gyrase.

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +24
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A +4
Waktu Paruh3-4 hours
Vol. Distribusi-
Klirens-
Genetik -
Norflurane Approved DB13116
small molecule | CAS: 811-97-2

Norflurane is under investigation in clinical trial NCT01673061 (Vapocoolant Spray for Numbing Small Boils Before Incision and Drainage).

Kategori:
Aerosol PropellantsAerosolsAlkanes +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norgestomet DB11440
small molecule | CAS: 25092-41-5

Norgestomet, also known as 11?-methyl-17-hydroxy-19-norprogesterone acetate, is a steroidal progestin used in veterinary medicine to control estrus and ovulation in cattle.

Kategori:
Fused-Ring CompoundsPregnanesPregnenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norleucine DB15458
small molecule | CAS: 327-57-1

Norleucine is under investigation in clinical trial NCT00081952 (Amino Acid Therapy for Hot Flashes in Postmenopausal Women).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAminocaproates
Target Protein:
Hepatocyte nuclear factor 1-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Methionine aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 99697-24-2

norUrsodeoxycholic acid is under investigation in clinical trial NCT03872921 (Norursodeoxycholic Acid vs Placebo in PSC).

Kategori:
Bile Acids and SaltsCholanesCholic Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norvaline DB04185
small molecule | CAS: 6600-40-4

Norvaline is an isomer of the more common amino acid valine.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins
Target Protein:
Glycine amidinotransferase, mitochondrialOrnithine transcarbamylase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Novobiocin Approved DB01051
small molecule | CAS: 303-81-1

Novobiocin is an antibiotic compound derived from _Streptomyces niveus_. It has a chemical structure similar to coumarin. Novobiocin binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. (From Reynolds, Martindale The Extra Pharmacopoeia,…

Kategori:
AminocoumarinsAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh6 hours
Vol. Distribusi-
Klirens-
Genetik -
Novolimus DB19085
small molecule | CAS: 151519-50-5

Novolimus is under investigation in clinical trial NCT04483791 (Dynamx Bioadaptor Hong Kong Registry).

Kategori:
LactonesPolyketides
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NP-51 DB16995
small molecule | CAS: 66611-38-9

Deskripsi belum tersedia.

Kategori:
AminesEnzyme InhibitorsHydroxylamines
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NP-6A4 DB17599
biotech

NP-6A4 is a peptide designed to specifically bind and activate angiotensin II receptor type 2 (AT2R). It has an Orphan Drug designation from the FDA for pediatric cardiomyopathy.[A258523]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-2359 DB05805
small molecule | CAS: 195875-68-4

NS2359 is a triple monoamine re-uptake inhibitor with a new, unique drug profile expected to yield important benefits compared to existing treatments of depression. Enhancing the function of the three neurotransmitters serotonin, noradrenalin and dopamine, NS…

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds +1
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NSI-566 DB17954
biotech

NSI-566 is a stem cell therapy consisting of human spinal cord-derived neural stem cells. Developed by Seneca Biopharma, it is being investigated for the treatment of amyotrophic lateral sclerosis (ALS), stroke, and chronic spinal cord injury (cSCI).[L47097]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NUC-7738 DB19148
small molecule | CAS: 2348493-39-8

NUC-7738 is under investigation in clinical trial NCT03829254 (A Safety, Pharmacokinetic and Clinical Activity Study of NUC-7738 in Patients With Advanced Solid Tumours and Lymphoma).

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-18 DB05886
small molecule

NV-18 is a product of the Novogen diphenolic synthetic analogue program that is creating drugs with diverse activities against specific types of cancer. Like phenoxodiol, NV-18 is broadly effective in the laboratory against almost all human cancer types, but …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-354 DB18392
small molecule | CAS: 866465-21-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-5138 DB19180
small molecule | CAS: 2095886-80-7

NV-5138 is under investigation in clinical trial NCT06235905 (Open-label of SPN-820 in Adults With Major Depressive Disorder).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NVP-LEQ-506 DB12857
small molecule | CAS: 1204975-42-7

LEQ506 has been used in trials studying the treatment of Advanced Solid Tumors, Recurrent or Refractory Medulloblastoma, and Locally Advanced or Metastatic Basal Cell Carcinoma.

Target Protein:
Protein smoothened
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NX-210c DB18209
biotech | CAS: 216682-41-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

NY-ESO-1 peptide vaccine is an investigational cancer immunotherapy. It contains a peptide derived from the cancer-testis antigen (NY-ESO-1).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nylidrin Approved DB06152
small molecule | CAS: 447-41-6

Nylidrin, also known as _buphenine_ belongs to the category of drugs called _vasodilators_, which relax blood vessels and increase blood flow. Nylidrin is a peripheral vasodilator. Some studies show the evidence of improving cognitive impairment in selected i…

Kategori:
2-Amino-1-Phenylethanol DerivativesAdrenergic AgentsAdrenergic Agonists +29
Target Protein:
Interferon alpha/beta receptor 2Voltage-dependent T-type calcium channel subunit alpha-1I
Waktu ParuhDuration of action …
Vol. Distribusi-
Klirens-
Genetik -
Nystatin Approved DB00646
small molecule | CAS: 1400-61-9

Nystatin is a polyene antifungal drug that has broad-spectrum fungicidal and fungistatic activity against a number of yeasts and fungi, most notably _Candida_ species.[L10686] It is one of the most effective antifungal agents synthesized by bacteria, in this …

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +17
Target Protein:
Ergosterol
Waktu Paruh-
Vol. DistribusiNystatin is not abs…
Klirens-
Genetik -
NYX-2925 DB19149
small molecule | CAS: 2012536-16-0

NYX-2925 is under investigation in clinical trial NCT04146896 (Efficacy and Safety of NYX-2925 in Subjects With Neuropathic Pain Associated With Diabetic Peripheral Neuropathy (DPN)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1Exotoxin AElongation factor 2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Stromelysin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
N-succinylarginine dihydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ATP-dependent Clp protease proteolytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxypeptidase A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27415-09-4

Deskripsi belum tersedia.

Kategori:
Acids, Carbocyclic
Target Protein:
o-succinylbenzoate synthaseo-succinylbenzoate synthaseo-succinylbenzoate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Fibroblast growth factor 1Hepatocyte growth factorHeparan sulfate glucosamine 3-O-sulfotransferase 3A1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OAV201 DB17842
biotech

OAV201 is a non-replicating, recombinant adeno-associated virus serotype 9 (AAV9) containing the human Methyl CpG Binding Protein 2B (MECP2B) cDNA under the control of a segment of the murine MECP2 promoter. It was first developed by Novartis and investigated…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obeticholic acid Approved DB05990
small molecule | CAS: 459789-99-2

Primary biliary cirrhosis, or PBC, is a progressive and chronic condition that leads to hepatic injury often resulting in end-stage liver failure that requires liver transplantation.[A192786] Obeticholic acid is a farnesoid-X receptor (FXR) agonist used to…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +14
Target Protein:
Bile acid receptor
Waktu ParuhThe biological half…
Vol. DistribusiThe volume of distr…
KlirensClearance informati…
Genetik -
OBI-3424 DB16057
small molecule | CAS: 2097713-68-1

OBI-3424 is under investigation in clinical trial NCT04315324 (Study to Test Akr1c3-activated Prodrug OBI-3424 (OBI-3424) in Patients With Relapsed/refractory T-cell Acute Lymphoblastic Leukemia (T-ALL)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OBI-833 DB19270
biotech | CAS: 2142641-90-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obiltoxaximab Approved DB05336
biotech | CAS: 1351337-07-9

Obiltoxaximab, an affinity-enhanced monoclonal antibody (Mab), is used for prevention and treatment of infection and death caused by anthrax toxin. Obiltoxaximab is a chimeric IgG1 kappa monoclonal antibody (mAb) that binds the PA component of B. anthracis to…

Kategori:
Amino Acids, Peptides, and ProteinsAnthrax Protective Antigen-directed AntibodyAnthrax Protective Antigen-directed Antibody Interactions +15
Target Protein:
Protective antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obinutuzumab Approved DB08935
biotech | CAS: 949142-50-1

Obinutuzumab is a humanized monoclonal antibody used as a combination treatment with chlorambucil to treat patients with untreated chronic lymphocytic leukemia. It was approved by the FDA in November 2013 and is marketed under the brand name Gazyva. There is …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +20
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe half life of ob…
Vol. DistribusiObinutuzumab has a …
KlirensThe clearance of ob…
Genetik -
Ochromycinone DB15644
small molecule | CAS: 28882-53-3

Ochromycinone is under investigation in clinical trial NCT01047943 (STA-21 Topical Efficacy on Psoriasis).

Kategori:
AnthracenesQuinones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4601–4650 dari 6694
Sebelumnya Halaman 93 / 134 Berikutnya