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11778

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Halaman 93 / 236
Edoxaban Approved DB09075
small molecule | CAS: 480449-70-5

Edoxaban is a member of the Novel Oral Anti-Coagulants (NOACs) class of drugs, and is a rapidly acting, oral, selective factor Xa inhibitor. By inhibiting factor Xa, a key protein in the coagulation cascade, edoxaban prevents the stepwise amplification of pro…

Kategori:
AnticoagulantsAntithrombinsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
Klirens22 L/hr
Genetik -
Edoxudine Approved DB13421
small molecule | CAS: 15176-29-1

Edoxudine is a deoxythymidine analog with activity against herpes simplex virus. It is a potent and selective inhibitor of herpes simplex virus type 1 and 2. The obtained product is an antiviral ointment.[L2407] The activity of edoxudine against herpes simple…

Kategori:
Anti-Infective AgentsAntiviral AgentsDeoxyribonucleosides +5
Target Protein:
Thymidine kinase, cytosolicDNA polymerase
Waktu ParuhIn preclinical tria…
Vol. DistribusiThis pharmacokineti…
KlirensThe plasma clearanc…
Genetik -
EDP1815 DB16486
biotech

EDP1815, was investigated in several clinical trials (NCT05066373, NCT05439941, NCT05682222, NCT03733353, NCT04603027, NCT04488575, NCT05121480, NCT04393246) to evaluate its safety and efficacy in conditions such as gastrointestinal behavior, atopic dermatiti…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edralbrutinib DB18095
small molecule | CAS: 1858206-58-2

Edralbrutinib is an orally available small molecule inhibitor of Bruton's tyrosine kinase.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edratide DB15272
small molecule | CAS: 433922-67-9

Edratide is under investigation in clinical trial NCT00203151 (A Study to Evaluate the Tolerability, Safety and Effectiveness of Edratide in the Treatment of Lupus).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edrecolomab DB13375
biotech | CAS: 156586-89-9

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EF-022 DB17768
biotech

EF-022 is a modified version of vitamin D binding protein macrophage activator, with potential antineoplastic and anti-angiogenic activities.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efalizumab Approved DB00095
biotech | CAS: 214745-43-4

Humanized IgG1 kappa isotype monoclonal antibody that binds to human CD11a. Efalizumab has a molecular weight of approximately 150 kilodaltons and is produced in a Chinese hamster ovary mammalian cell expression system in a nutrient medium containing the anti…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-XIntegrin alpha-L
Waktu Paruh5 days
Vol. Distribusi-
Klirens-
Genetik -
Efanesoctocog alfa Approved DB16662
biotech | CAS: 2252477-42-0

Efanesoctocog alfa (BIVV001) is a recombinant factor VIII (FVIII) analogue fusion protein used for the routine prophylaxis, perioperative management of bleeding and on-demand treatment and control of bleeding episodes in patients with hemophilia A.[L45379] Th…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Target Protein:
Coagulation factor IXCoagulation factor XLow-density lipoprotein receptor-related protein 2 +1
Waktu ParuhEfanesoctocog alfa …
Vol. DistribusiEfanesoctocog alfa …
KlirensEfanesoctocog alfa …
Genetik -
Efaproxiral DB08486
small molecule | CAS: 131179-95-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAminesAntineoplastic Agents +9
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efatutazone DB11894
small molecule | CAS: 223132-37-4

Efatutazone has been used in trials studying the treatment of Lymphoma, Liposarcoma, Solid Tumors, Multiple Myeloma, and Recurrent Thyroid Cancer, among others.

Kategori:
Antineoplastic AgentsPPAR gamma, antagonists & inhibitorsSulfur Compounds +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2049067-94-7

Efavaleukin alfa is a fusion protein consisting of interleukin mutein fused to the C-terminus of an immunoglobulin G Fc domain by way of a G4S linker. It is under investigation in clinical trial NCT03422627 (Safety and Efficacy of AMG 592 in Subjects With Ste…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efbemalenograstim alfa Approved DB18704
biotech | CAS: 2200269-79-8

Efbemalenograstim alfa is a long-acting recombinant fusion protein of granulocyte-colony stimulating factor (G-CSF) due to the addition of the Fc portion of human IgG2, allowing for once-per-cycle administration.[L48852,A262167] As endogenous G-CSF mediates t…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors +2
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Efepoetin alfa DB19197
biotech | CAS: 1905452-78-9

Efepoetin alfa is under investigation in clinical trial NCT04155125 (A Study of Efepoetin Alfa in Treating Anaemia Associated With Chronic Kidney Diseases Patient).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efgartigimod alfa Approved DB15270
biotech | CAS: 1821402-21-4

Myasthenia gravis (MG) is an autoimmune disorder characterized by significant muscle weakness - particularly in the eye, throat, and extremities - caused by autoantibodies attacking the neuromuscular junction.[A243759] The production of IgG autoantibodies aga…

Kategori:
AntibodiesAntineoplastic and Immunomodulating AgentsGlobulins +6
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
biotech | CAS: 2026634-47-7

Efineptakin alfa (also known as NT-I7) is a long-acting human interleukin-7 (IL-7) fusion protein that promotes T-cell development, contributing to the immune response. Compared to endogenous IL-7, NT-I7 is more stable and potent, has a longer half-life, and …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efinopegdutide DB15077
biotech | CAS: 2055640-93-0

Efinopegdutide is under investigation in clinical trial NCT03606057 (A Study to Investigate the Effect of JNJ-64565111 on Cardiac Repolarization (Corrected QT Interval) Compared With Placebo in Healthy Adults: a Thorough ECG Study Employing Placebo, JNJ-64565…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1635395-27-5

Efizonerimod alfa is under investigation in clinical trial NCT02221960 (A Phase 1 Study to Evaluate MEDI6383 Alone and in Combination With MEDI4736 in Adult Subjects With Select Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflapegrastim Approved DB15001
biotech | CAS: 1384099-30-2

Febrile neutropenia (FN), defined as the co-occurrence of fever (temperature > 38 ?C) and severe neutropenia (ANC < 500 cells/mm<sup>3</sup>), is a potential side effect of myelosuppressive chemotherapy in which the patient develops an infection during a peri…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhIn patients with br…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ef…
Genetik -
biotech

Eflepedocokin alfa is a recombinant IL-22-Fc fusion protein manufactured in Chinese hamster ovary cells that is composed of 2 human interleukin 22 (IL-22) molecules linked to an immunoglobulin constant region (IgG2-Fc).[A225706, L27661] It is being developed …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1953227-87-6

Efmarodocokin alfa is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efmoroctocog alfa Approved DB11607
biotech | CAS: 1270012-79-7

Efmoroctocog alfa is a fully recombinant factor VIII-Fc fusion protein (rFVIIIFc) with an extended half-life compared with conventional factor VIII (FVIII) preparations, including recombinant FVIII (rFVIII) products such as [DB13999][A31551]. It is an antihem…

Kategori:
HemostaticsHuman Antihemophilic Factors
Target Protein:
von Willebrand factor
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Efonidipine DB09235
small molecule | CAS: 111011-63-3

Efonidipine is a calcium channel blocker of the _dihydropyridine class_, commercialized by Shionogi & Co. (Japan). Initially, it was marketed in 1995 under the trade name, _Landel_. The drug has been shown to block T-type in addition to L-type calcium channel…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +22
Target Protein:
Voltage gated L-type calcium channelVoltage-dependent calcium channelVoltage-dependent T-type calcium channel +4
Waktu ParuhThe peak plasma con…
Vol. Distribusi-
Klirens-
Genetik -
Efpeglenatide DB15650
biotech | CAS: 1296200-77-5

Efpeglenatide is under investigation in clinical trial NCT03713684 (Efficacy and Safety of Efpeglenatide Versus Placebo in Patients With Type 2 Diabetes Mellitus Inadequately Controlled With Basal Insulin Alone or in Combination With Oral Antidiabetic Drug(s)…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efruxifermin DB19012
biotech | CAS: 2375240-92-7

Efruxifermin is under investigation in clinical trial NCT06215716 (A Study Evaluating Efruxifermin in Subjects With Non-cirrhotic Nonalcoholic Steatohepatitis (Nash)/metabolic Dysfunction-associated Steatohepatitis (MASH) and Fibrosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1905448-17-0

Eftansomatropin alfa (GX-H9) comprises a recombinant human growth hormone fused to hyFc, a synthetic hybrid Fc fragment.[L48275] It is under investigation for the treatment of growth hormone deficiency.

Kategori:
Amino Acids, Peptides, and ProteinsGrowth HormoneHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1800476-36-1

Eftilagimod alfa is under investigation in clinical trial NCT02614833 (IMP321 (Eftilagimod Alpha) as Adjunctive to a Standard Chemotherapy Paclitaxel Metastatic Breast Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Differentiation +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eftrenonacog alfa Approved DB11608
biotech | CAS: 1270012-74-2

Eftrenonacog alfa is a long-acting recombinant fusion protein used in the treatment of hemophilia B. It is comprised of a single molecule of human factor IX (FIX) covalently linked to the constant region (Fc) domain of human IgG1 via recombinant DNA technolog…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +15
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Efungumab DB16151
biotech | CAS: 762260-74-2

Efungumab is under investigation in clinical trial NCT00217815 (Preliminary Study of Mycograb and Docetaxel in Advanced Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egaptivon pegol DB05202
biotech | CAS: 934868-74-3

Egaptivon pegol, formerly known as ARC1779, is a therapeutic aptamer antagonist of the A1 domain of von Willebrand Factor (vWF), the ligand for receptor glycoprotein 1b on platelets. Egaptivon pegol is being investigated for the treatment of thrombotic thromb…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +2
Target Protein:
von Willebrand factorPlatelet glycoprotein Ib alpha chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGT-101 DB17645
biotech

EGT-101 is an adeno-associated viral vector serotype 9 (AAV9) vector-based gene therapy consisting of the human sulfamidase (SGSH) transgene. Developed by Esteve Pharmaceuticals, it is being investigated for Sanfilippo syndrome type A.[L45919]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGT-201 DB17648
biotech

EGT-201 is an adeno-associated viral vector serotype 9 (AAV9) vector-based gene therapy consisting of the alpha-N-acetyglucosaminidase (NAGLU) transgene. Developed by Esteve Pharmaceuticals, it is being investigated for Sanfilippo syndrome type B.[L45939]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGT-301 DB17649
biotech

EGT-301 is a gene therapy being investigated for Hunter Syndrome. It consists of an adeno-associated viral vector serotype 9 (AAV9) containing the human Iduronate-2-sulfatase (I2S) transgene designed to restore I2S functional deficiency in patients with Hunte…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EHP-102 DB16933
small molecule | CAS: 1807652-43-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EI-001 DB17596
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EI-1071 DB18486
small molecule

EI-1071 is a selective Colony Stimulating Factor-1 Receptor kinase inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elacestrant Approved DB06374
small molecule | CAS: 722533-56-4

Elacestrant is a non-steroidal small molecule and an estrogen receptor (ER) antagonist.[A256838,L44918] In January 2023, it was approved by the FDA for the treatment of ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer.[L44918,L449…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiElacestrant has an …
KlirensElacestrant has an …
Genetik -
Elacridar DB04881
small molecule | CAS: 143664-11-3

Elacridar (GW120918) is an oral bioenhancer that targets multiple drug resistance in tumors. In many cases, the appearance of multidrug resistance in cancer is due to a change in expression of protein inhibitors. As of August 2007 elacridar was not listed on …

Kategori:
BCRP/ABCG2 InhibitorsBenzocycloheptenesDrug Resistance, Multiple +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eladocagene exuparvovec Approved DB16780
biotech | CAS: 2098615-91-7

Eladocagene exuparvovec is a recombinant adeno-associated virus-2 (AAV2)-based gene therapy that expresses human aromatic L-amino acid decarboxylase (AADC), and it is used to treat AADC deficiency, a fatal and rare genetic disorder that causes severe disabili…

Kategori:
Adeno-associated Viral Vector TherapiesAlimentary Tract and MetabolismEnzymes +2
Waktu ParuhNot available.
Vol. DistribusiThe biodistribution…
KlirensNot available.
Genetik -
biotech

Elaeagnus angustifolia pollen is the pollen of the Elaeagnus angustifolia plant. Elaeagnus angustifolia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elafibranor Approved DB05187
small molecule | CAS: 923978-27-2

Elafibranor is a dual peroxisome proliferator-activated receptor (PPAR) ? and ?/? agonist [A263833] that works to inhibit bile acid synthesis.[L50768] On June 10, 2024, elafibranor was granted accelerated approval by the FDA for the treatment of primary bilia…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBCRP/ABCG2 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gamma
Waktu ParuhFollowing a single …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent t…
Genetik -
Elagolix Approved DB11979
small molecule | CAS: 834153-87-6

Elagolix has been used in trials studying the basic science and treatment of Endometriosis, Folliculogenesis, Uterine Fibroids, Heavy Uterine Bleeding, and Heavy Menstrual Bleeding. As of 24 July 2018, however, the U.S. Food and Drug Administration (FDA) appr…

Kategori:
Anti-Gonadotropin-Releasing HormonesAntigonadotropins and Similar AgentsCytochrome P-450 CYP2C19 Inhibitors +16
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe terminal phase …
Vol. DistribusiThe apparent volume…
KlirensThe oral clearance …
Genetik -
Elaidamide DB03784
small molecule | CAS: 4303-70-2

Deskripsi belum tersedia.

Target Protein:
Phospholipase A2, membrane associated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elamipretide DB11981
small molecule | CAS: 736992-21-5

Elamipretide has been used in trials studying the treatment of Leber's Hereditary Optic Neuropathy.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elapegademase Approved DB14712
biotech | CAS: 1709806-75-6

Elapegademase is a PEGylated recombinant adenosine deaminase. It can be defined molecularly as a genetically modified bovine adenosine deaminase with a modification in cysteine 74 for serine and with about 13 methoxy polyethylene glycol chains bound via carbo…

Kategori:
Adenosine Deaminase InhibitorsAdjuvants, ImmunologicAmino Acids, Peptides, and Proteins +12
Target Protein:
Adenosine
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Elastin (human) DB15364
biotech | CAS: 9007-58-3

Elastin (human) is under investigation in clinical trial NCT01466413 (Two Formulations of ELAPR Compared to Restylane® Vital Light Following Repeat Implants in the Upper Arm Dermis).

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersElastin +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elbasvir Approved DB11574
small molecule | CAS: 1370468-36-2

Elbasvir is a direct-acting antiviral medication used as part of combination therapy to treat chronic hepatitis C, an infectious liver disease caused by infection with hepatitis C virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine d…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +18
Target Protein:
Nonstructural protein 5A
Waktu ParuhThe geometric mean …
Vol. DistribusiElbasvir has an est…
KlirensThe clearance of el…
Genetik -
Elcatonin DB13742
small molecule | CAS: 60731-46-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Parathyroid AgentsBone Density Conservation Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eldecalcitol DB05295
small molecule | CAS: 104121-92-8

Eldecalcitol (ED-71), a vitamin D analog, is a more potent inhibitor of bone resorption than alfacalcidol in an estrogen-deficient rat model of osteoporosis. Eldecalcitol, effectively and safely increased lumbar and hip bone mineral density (BMD) in osteopor…

Kategori:
Bone Density Conservation AgentsFused-Ring CompoundsSecosteroids +4
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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