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14494

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9687 (66.8%)
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7525 (51.9%)
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112 (0.8%)
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14494 (100.0%)

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Halaman 91 / 290
Codrituzumab DB14843
biotech | CAS: 1365267-33-9

Codrituzumab is under investigation in clinical trial NCT01507168 (A Study of RO5137382 (GC33) in Patients With Advanced or Metastatic Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coelenteramide DB04049
small molecule

Deskripsi belum tersedia.

Kategori:
AcetamidesAmidesBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme A DB01992
small molecule | CAS: 85-61-0

Coenzyme A (CoA, CoASH, or HSCoA) is a coenzyme, well known for it's role in the synthesis and oxidation of fatty acids, and the oxidation of pyruvate in the citric acid cycle. All genomes sequenced to date encode enzymes that use coenzyme A as a substrate, a…

Kategori:
Adenine NucleotidesCoenzyme A, biosynthesisCoenzymes +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseCarnitine O-acetyltransferaseGalactoside O-acetyltransferase +42
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 81918-99-2

Coenzyme A persulfide is a possible in vivo inhibitor of mammalian short chain acyl-CoA dehydrogenase.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isovaleryl-CoA dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme F420 DB03913
small molecule | CAS: 64885-97-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme M Approved DB09110
small molecule | CAS: 3375-50-6

Coenzyme M (commonly known by its salt form, Mesna) is a synthetic sulfhydryl (thiol) compound and is used for prophylaxis of Ifosfamide and cyclophosphamide induced hemorrhagic cystitis.[A18572]

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +12
Waktu ParuhThe elimination hal…
Vol. DistribusiVd = 0.652 ± 0.242 …
KlirensPlasma clearance of…
Genetik -
Coffea arabica seed, roasted Approved DB15603
biotech

Coffea arabica seed, roasted allergenic extract is used in allergenic testing.

Waktu Paruh-
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Coffee bean Approved DB10525
biotech

Coffee bean allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cofirasersen DB19037
biotech | CAS: 2247669-96-9

Cofirasersen is under investigation in clinical trial NCT04441788 (A Study to Assess the Safety, Tolerability, and Efficacy of ION-827359 in Participants With Mild to Moderate Chronic Obstructive Pulmonary Disease (COPD) With Chronic Bronchitis (CB)).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Col-118 DB05778
small molecule

COL-118, a topical compound based on the SansRosa technology, for the treatment of redness associated with rosacea and other skin disorders. It is a believed to reduce erythema by constricting enlarged blood vessels in facial tissue. Col-118 is a unique formu…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Col-Treg DB18451
biotech

Col-Treg is an autologous T-cell therapy comprising type I regulatory T-cells specific for human type II collagen.[A261635]

Waktu Paruh-
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Colchiceine Approved DB15534
small molecule | CAS: 477-27-0

Colchiceine is one of several metabolites of the anti-gout medication [colchicine].[A192714]

Kategori:
AlkaloidsColchicine DerivativesTubulin Inhibiting Agent
Target Protein:
Tubulin beta chainTubulin alpha-1A chain
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Colchicine Approved DB01394
small molecule | CAS: 64-86-8

Colchicine is an alkaloid drug derived from a plant belonging to the Lily family, known as _Colchicum autumnale_, or "autumn crocus."[A183611] Its use was first approved by the FDA in 1961.[L8192] Colchicine is used in the treatment of gout flares and Familia…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntigout Preparations +23
Target Protein:
Tubulin beta chain
Waktu ParuhAfter several doses…
Vol. DistribusiThe mean apparent v…
KlirensIn one pharmacokine…
Genetik -
Coleneuramide DB14932
small molecule | CAS: 204200-47-5

Coleneuramide is under investigation in clinical trial NCT00307749 (Safety and Efficacy of MCC-257 in the Treatment of Diabetic Polyneuropathy).

Kategori:
Acids, AcyclicAmino SugarsCarbohydrates +3
Waktu Paruh-
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Colesevelam Approved DB00930
small molecule | CAS: 182815-43-6

Colesevelam is a bile acid sequestrant. Colesevelam is used with exercise and diet changes (restriction of cholesterol and fat intake) to reduce the amount of cholesterol and certain fatty substances in the blood. It works by binding bile acids in the intesti…

Kategori:
AlkenesAllyl CompoundsAllylamine +11
Target Protein:
Bile acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Colestilan chloride Approved DB11634
small molecule | CAS: 95522-45-5

Colestilan is an ingredient in the EMA-withdrawn product BindRen.

Kategori:
Drugs for Treatment of Hyperkalemia and HyperphosphatemiaFused-Ring CompoundsSteroids
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Colestipol Approved DB00375
small molecule | CAS: 26658-42-4

Bile acid sequestrants like colestipol have been in use since the 1970s.[FDA Label, F4555, F4567, L6262] And even though such an agent may very well be useful in reducing elevated cholesterol levels and decreasing the risk for atherosclerotic vascular disease…

Kategori:
AminesAnion Exchange ResinsBile Acid Sequestrants +12
Target Protein:
Bile acids
Waktu ParuhColestipol is not a…
Vol. DistribusiColestipol is not a…
KlirensColestipol is not a…
Genetik -
Colforsin DB02587
small molecule | CAS: 66575-29-9

Potent activator of the adenylate cyclase system and the biosynthesis of cyclic AMP. From the plant Coleus forskohlii. Has antihypertensive, positive inotropic, platelet aggregation inhibitory, and smooth muscle relaxant activities; also lowers intraocular pr…

Kategori:
Adjuvants, ImmunologicAnti-Asthmatic AgentsAutonomic Agents +12
Target Protein:
Adenylate cyclaseAdenylate cyclase type 2Guanine nucleotide-binding protein G(s) subunit alpha isoforms short +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Colfosceril palmitate Approved DB09114
small molecule | CAS: 63-89-8

Colfosceril palmitate is a synthetic pulmonary surfactant administered in infants with respiratory distress syndrome.[A31510] It was part of the first generation of commercially available artificial surfactants.[T70] It was developed by Burroughs Wellcome and…

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +6
Waktu ParuhThe half-life of co…
Vol. DistribusiColfosceril palmita…
KlirensAfter 5 days of dru…
Genetik -
Colistimethate Approved DB01111
small molecule | CAS: 12705-41-8

Colistimethate is an antibiotic that has been shown to have bactericidal activity against aerobic gram-negative microorganisms. Colistimethate is particularly indicated when the infection is caused by sensitive strains of Pseudomonas aeruginosa.

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAntimicrobial Cationic Peptides +11
Target Protein:
Dihydropteroate synthaseBacterial outer membrane
Waktu Paruh2-3 hours following…
Vol. Distribusi-
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Genetik -
Colistin Approved DB00803
biotech | CAS: 1066-17-7

Cyclic polypeptide antibiotic from Bacillus colistinus. It is composed of Polymyxins E1 and E2 (or Colistins A, B, and C) which act as detergents on cell membranes. Colistin is less toxic than Polymyxin B, but otherwise similar; the methanesulfonate is used o…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +21
Target Protein:
Dihydropteroate synthaseBacterial outer membrane
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Collagen-polyvinylpyrrolidone is a copolymer generated from a mixture of type I collagen and low-molecular-weight PVP that has undergone ? irradiation[A227733]. It is characterized by antifibrotic, fibrolytic, and immunomodulatory properties[A227733].

Kategori:
AlkenesAmino Acids, Peptides, and ProteinsBiopolymers +11
Waktu Paruh-
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Genetik -
biotech | CAS: 9001-12-1

Collagenase clostridium histolyticum is an enzyme produced by the bacterium Clostridium histolyticum. It is beneficial in the breakdown of collagen plaques for the treatment of Dupuytren's contracture and Peyronie's disease.[L14882] The topical formulation is…

Kategori:
Collagen-specific EnzymeCollagenasesDermatologicals +11
Target Protein:
Collagen alpha-1(I) chainCollagen alpha-1(II) chainCollagen alpha-1(III) chain
Waktu Paruh-
Vol. DistribusiThere is no current…
KlirensClearance informati…
Genetik -
Colletotrichum coccodes Approved DB10824
biotech

Colletotrichum coccodes is a fungus which can provoke allergic reactions. Colletotrichum coccodes extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Colloidal oatmeal Approved DB11286
biotech

Colloidal oatmeal is produced by grinding fine granules of oatmeal and boiling it to extract the colloidal material. It contains high concentrations of starches and beta-glucan that exhibits water-absorbing properties. Phenols are also contained in colloidal …

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1269764-99-9

Coltuximab ravtansine (SAR3419) targets CD19 and is being investigated for the treatment of acute lymphoblastic leukemia (ALL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +16
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Combretastatin DB12596
small molecule | CAS: 82855-09-2

Combretastatin has been investigated for the treatment of Anaplastic Thyroid Cancer.

Kategori:
Antimitotic AgentsAntineoplastic AgentsAntineoplastic Agents, Phytogenic +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117048-59-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Common carp Approved DB10614
biotech

Common carp allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Comosain DB18354
biotech

Deskripsi belum tersedia.

Kategori:
Cysteine ProteasesEndopeptidasesEnzymes +3
Waktu Paruh-
Vol. Distribusi-
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Compound 18 DB02715
small molecule | CAS: 31112-66-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Compound 19 DB02615
small molecule

Deskripsi belum tersedia.

Target Protein:
Estrogen receptorTyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Compound 4-D DB03742
small molecule

Deskripsi belum tersedia.

Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Conatumumab DB11646
biotech | CAS: 896731-82-1

Conatumumab has been used in trials studying the treatment of Sarcoma, Lymphoma, Oncology, Colon Cancer, and Rectal Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Conbercept DB12460
biotech | CAS: 1227158-72-6

Conbercept has been investigated for the basic science of Age-related Macular Degeneration.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Concanamycin A DB14062
small molecule | CAS: 80890-47-7

Concanamycin A is an H+-ATPase (vacuolar) inhibitor.

Kategori:
Anti-Infective AgentsEnzyme InhibitorsLactones +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Concizumab DB12820
biotech | CAS: 1312299-39-0

Concizumab has been used in trials studying the treatment of Haemophilia A and Congenital Bleeding Disorder.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Concord grape Approved DB10875
biotech

Concord grape allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Condoliase DB12793
biotech | CAS: 9024-13-9

Condoliase has been used in trials studying the treatment of Lumbar Disc Disease, Lumbar Vertebra Hernia, and Intervertebral Disc Disease.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Conestat alfa Approved DB09228
biotech | CAS: 80295-38-1

C1 Esterase Inhibitor (Recombinant) is a recombinant analogue of endogenous complement component-1 esterase inhibitor (rhC1INH), purified from the milk of transgenic rabbits. The primary function of endogenous C1INH is to regulate the activation of the comple…

Kategori:
Amino Acids, Peptides, and ProteinsAngioedemas, Hereditary, drug therapyBlood and Blood Forming Organs +16
Target Protein:
Complement C1r subcomponentComplement C1s subcomponentPlasma kallikrein +4
Waktu Paruh-
Vol. Distribusi-
KlirensClearance was found…
Genetik -
Conivaptan Approved DB00872
small molecule | CAS: 210101-16-9

Conivaptan is a non-peptide inhibitor of antidiuretic hormone (vasopressin). It was approved in 2004 for hyponatremia (low blood sodium levels) caused by syndrome of inappropriate antidiuretic hormone (SIADH). Conivaptan inhibits both isotypes of the vasopres…

Kategori:
Antidiuretic Hormone Receptor AntagonistsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Vasopressin V1a receptorVasopressin V2 receptor
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
Conjugated estrogens Approved DB00286
small molecule | CAS: 12126-59-9

The conjugated estrogens are noncrystalline mixtures of purified female sex hormones obtained either by its isolation from the urine of pregnant mares or by synthetic generation from vegetal material. Both of these products are later conjugated to natrium sul…

Kategori:
Agents causing angioedemaBCRP/ABCG2 SubstratesCOMT Substrates +26
Target Protein:
Estrogen receptor betaEstrogen receptor
Waktu ParuhThe median half-lif…
Vol. DistribusiThe physiological d…
KlirensThe reported normal…
Genetik -
Contulakin-G DB05950
small molecule | CAS: 229180-41-0

Contulakin-G is a broad spectrum non-opioid analgesic. It is the synthetic form of a natural peptide extracted from the venom of the Conus Geographus sea snail.

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsPeptides +1
Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copanlisib Approved DB12483
small molecule | CAS: 1032568-63-0

Copanlisib is a selective pan-Class I phosphoinositide 3-kinase (PI3K) inhibitor with preferential activity against the alpha and delta isoforms. PI3K, a lipid kinase that activates downstream signalling pathways involved in cell survival and growth, that exi…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +17
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform +1
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Copper Approved DB09130
small molecule | CAS: 7440-50-8

Copper is a transition metal and a trace element in the body. It is important to the function of many enzymes including cytochrome c oxidase, monoamine oxidase and superoxide dismutase [FDA Label]. Copper is commonly used in contraceptive intrauterine devices…

Kategori:
Copper-containing Intrauterine DeviceDecreased Embryonic ImplantationDecreased Sperm Motility +12
Target Protein:
Amyloid-beta precursor proteinAdenosylhomocysteinaseHistone H2B type 1-C/E/F/G/I +143
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper Cu-64 Approved DB13980
small molecule | CAS: 13981-25-4

Copper-64 is a radiopharmaceutical usually found in the +2 oxidation state as the complexes including the +1 state tend to be more unstable.[T604] It is used in molecular radiotherapy and positron emission tomography.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Copper gluconate Approved DB11246
small molecule | CAS: 527-09-3

Copper gluconate is a copper salt of D-gluconic acid that displays a light blue to bluish-green color. It is prepared by the reaction of gluconic acid solutions with cupric oxide or basic cupric carbonate. According to the good manufacturing or feeding practi…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper oxodotreotide Cu-64 Approved DB15873
small molecule | CAS: 1426155-87-4

Copper Cu 64 dotatate is a newly approved Cu labeled somatostatin analog and has several advantages over <sup>68</sup>Ga-labeled somatostatin analogs for positron emission tomography (PET).[A220348] Copper Cu 64 dotatate has a longer half-life and can be prod…

Kategori:
Amino Acids, Peptides, and ProteinsCopper RadioisotopesPeptides +4
Target Protein:
Somatostatin receptor type 2
Waktu ParuhThe half-life of Co…
Vol. Distribusi-
Klirens-
Genetik -
Copper usnate DB13830
small molecule

Deskripsi belum tersedia.

Kategori:
Genito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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