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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 90 / 134
small molecule

N2-[(benzyloxy)carbonyl]-n1-[(3S)-1-cyanopyrrolidin-3-yl]-l-leucinamide is a solid. This compound belongs to the n-acyl-alpha amino acids and derivatives. These are compounds containing an alpha amino acid (or a derivative thereof) which bears an acyl group a…

Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Matrilysin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
Waktu Paruh-
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Genetik -
Nabilone Approved DB00486
small molecule | CAS: 51022-71-0

Nabilone (marketed as Cesamet) is a synthetic form of delta-9-tetrahydrocannabinol (??-THC), the primary psychoactive component of cannabis (marijuana). Although structurally distinct from THC, nabilone mimics THC's structure and pharmacological activity thro…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAntiemetics +30
Target Protein:
Cannabinoid receptor 2Cannabinoid receptor 1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Nabiximols DB14011
small molecule | CAS: 56575-23-6

Nabiximols (tradename Sativex®) is a whole plant extract from the Cannabis species _Cannabis sativa L._ that has been purified into the active components CBD (cannabidiol) and THC (delta-9-tetrahydrocannabinol). For trademark purposes, purified CBD is branded…

Kategori:
Agents producing tachycardiaAnalgesicsBCRP/ABCG2 Inhibitors +24
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +41
Waktu ParuhElimination from pl…
Vol. DistribusiCannabinoids are di…
Klirens-
Genetik -
Nabumetone Approved DB00461
small molecule | CAS: 42924-53-8

Nabumetone was originally developed as a non-acidic non-steroidal anti-inflammatory drug (NSAID).[label] It was thought to avoid trapping of the drug in the stomach by making it unable to dissociate into ions which was believed to reduce GI toxicity by limiti…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +21
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh6-MNA has a mean ha…
Vol. DistribusiThe Vd of 6-MNA rep…
Klirens6-MNA has an appare…
Genetik -
Nacubactam DB15353
small molecule | CAS: 1452458-86-4

Nacubactam is under investigation in clinical trial NCT03174795 (A Study to Investigate the Pharmacokinetics of RO7079901 and Meropenem in Participants With a Complicated Urinary Tract Infection).

Kategori:
AmidesAza Compounds
Target Protein:
Beta-lactamase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nadifloxacin DB12447
small molecule | CAS: 124858-35-1

Nadifloxacin has been used in trials studying the treatment of Acne Vulgaris.

Kategori:
4-QuinolonesAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +10
Waktu Paruh-
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Nadofaragene firadenovec Approved DB17381
biotech | CAS: 1823059-12-6

Nadofaragene firadenovec (nadofaragene firadenovec-vncg) is a recombinant non-replicating adenovirus serotype 5 vector containing a transgene encoding human interferon alfa-2b (IFN?2b).[L44381] It was approved by the FDA on December 2022 for the treatment of …

Kategori:
Adeno-associated Viral Vector TherapiesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Waktu Paruh-
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Nadroparin Approved DB08813
small molecule

Nadroparin is a low molecular weight heparin (LMWH) which, when bound to antithrombin III (ATIII), accelerates the inactivation of factor II and factor Xa. Nadroparin halts the coagulation pathway by inhibiting the activation of thrombin (factor IIa) by facto…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIP-selectinProtein c-Fos +1
Waktu ParuhIn healthy patients…
Vol. Distribusi3.59L
KlirensThe clearance of na…
Genetik -
Nafamostat DB12598
small molecule | CAS: 81525-10-2

Nafamostat is a synthetic serine protease inhibitor that is commonly formulated with hydrochloric acid due to its basic properties. It has been used in trials studying the prevention of Liver Transplantation and Postreperfusion Syndrome. The use of nafamostat…

Kategori:
AmidinesAnalgesicsAnalgesics, Non-Narcotic +16
Target Protein:
Tumor necrosis factorProthrombinCoagulation factor X +4
Waktu ParuhApproximately 8 min…
Vol. Distribusi-
Klirens-
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Nafarelin Approved DB00666
small molecule | CAS: 76932-56-4

Nafarelin is a potent synthetic agonist of gonadotropin-releasing hormone with 3-(2-naphthyl)-D-alanine substitution at residue 6. Nafarelin has been used in the treatments of central precocious puberty and endometriosis.

Kategori:
Adrenal Cortex HormonesAgents Causing Muscle ToxicityAmino Acids, Peptides, and Proteins +19
Target Protein:
Gonadotropin-releasing hormone receptorPutative gonadotropin-releasing hormone II receptor
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Nafcillin Approved DB00607
small molecule | CAS: 147-52-4

A semi-synthetic antibiotic related to penicillin, Naficillin is a narrow-spectrum beta-lactam antibiotic drug. It is a beta-lactamase-resistant penicillin that is indicated for the treatment of Staphylococcal infections caused by strains that are resistant t…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +17
Target Protein:
Penicillin-binding protein 1bPenicillin-binding protein 2BPenicillin-binding protein 2a +2
Waktu ParuhThe serum half-life…
Vol. DistribusiNafcillin is report…
Klirens-
Genetik -
Nafithromycin DB16246
small molecule | CAS: 1691240-78-4

Nafithromycin is under investigation in clinical trial NCT02903836 (Phase II Study of Oral Nafithromycin in CABP).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Nalidixic acid Approved DB00779
small molecule | CAS: 389-08-2

Nalidixic acid is a synthetic 1,8-naphthyridine antimicrobial agent with a limited bacteriocidal spectrum. It is an inhibitor of the A subunit of bacterial DNA gyrase.

Kategori:
4-QuinolonesAgents that reduce seizure thresholdAnti-Bacterial Agents +19
Target Protein:
DNADNA topoisomerase 2-betaDNA topoisomerase 2-alpha
Waktu Paruh1.1 to 2.5 hours in…
Vol. Distribusi-
Klirens-
Genetik -
Naloxone Approved DB01183
small molecule | CAS: 465-65-6

Naloxone is an opioid antagonist medication used to block or reverse the effects of opioid drugs, particularly within the setting of drug overdoses which are rapidly becoming a leading cause of death worldwide.[A234594] More specifically, naloxone has a high …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnalgesics +27
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +4
Waktu ParuhThe mean half life …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of na…
Genetik -
Namodenoson DB12885
small molecule | CAS: 163042-96-4

Namodenoson has been used in trials studying the treatment of Chronic Hepatitis C and Hepatocellular Carcinoma.

Kategori:
Heterocyclic Compounds, Fused-RingNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +7
Target Protein:
Adenosine receptor A3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nanaomycin D DB01668
small molecule

Deskripsi belum tersedia.

Kategori:
BenzopyransBenzoquinonesChromans +6
Target Protein:
ActVA 6 protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nandrolone decanoate Approved DB08804
small molecule | CAS: 360-70-3

Nandrolone decanoate, also known as nandrolone caprinate, is an alkylated anabolic steroid indicated in the management of anemia of renal insufficiency and as an adjunct therapy in the treatment of senile and postmenopausal osteoporosis.[A233789,A233849,L3256…

Kategori:
Anabolic AgentsAndrogensBone Density Conservation Agents +16
Target Protein:
Androgen receptorProtein c-Fos5-hydroxytryptamine 2 receptor +3
Waktu ParuhNandrolone decanoat…
Vol. Distribusi-
Klirens50 mg, 100 mg, and …
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Nanoparticle Epirubicin is under investigation in clinical trial NCT03168061 (Dose-escalation and Expansion Trial of NC-6300 in Patients With Advanced Solid Tumors or Soft Tissue Sarcoma). It is a novel [epirubicin] drug-conjugated polymeric micelle.

Kategori:
Amino Acids, Peptides, and ProteinsAminoglycoside AntibacterialsAnthracyclines +5
Waktu Paruh-
Vol. Distribusi-
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Nanvuranlat DB18250
small molecule | CAS: 1037592-40-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Napabucasin DB12155
small molecule | CAS: 83280-65-3

Napabucasin has been investigated for the treatment of Colorectal Carcinoma.

Kategori:
Heterocyclic Compounds, Fused-RingNaphthalenesQuinones
Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
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small molecule | CAS: 581-75-9

Deskripsi belum tersedia.

Kategori:
ArylsulfonatesArylsulfonic AcidsNaphthalenes +3
Target Protein:
Bacterioferritin comigratory proteinL-lactate dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naproxcinod DB06682
small molecule | CAS: 163133-43-5

Deskripsi belum tersedia.

Kategori:
Antiinflammatory and Antirheumatic ProductsAntiinflammatory and Antirheumatic Products, Non-SteroidsCardiovascular Agents +5
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naproxen Approved DB00788
small molecule | CAS: 22204-53-1

Naproxen is classified as a nonsteroidal anti-inflammatory dug (NSAID) and was initially approved for prescription use in 1976 and then for over-the-counter (OTC) use in 1994.[A178975] It can effectively manage acute pain as well as pain related to rheumatic …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +41
Target Protein:
Pancreatic triacylglycerol lipaseProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +1
Waktu ParuhThe elimination hal…
Vol. DistribusiNaproxen has a volu…
KlirensNaproxen is cleared…
Genetik -
biotech | CAS: 676258-98-3

Naptumomab Estafenatox has been used in trials studying the treatment of Pancreatic Cancer, Renal Cell Carcinoma, and Non-Small-Cell Lung Carcinoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narasin DB11432
small molecule | CAS: 55134-13-9

Narasin is an agent with coccidiostatic and antibacterial properties.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narazaciclib DB19038
small molecule | CAS: 1357470-29-1

Narazaciclib is under investigation in clinical trial NCT06351644 (On 123300 (Narazaciclib) and Dexamethasone in Patients With Relapsed And/or Refractory Multiple Myeloma).

Waktu Paruh-
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Naronapride DB05542
small molecule | CAS: 860174-12-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +7
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narsoplimab DB16418
biotech | CAS: 2108782-45-0

Thrombotic microangiopathies (TMA), including thrombotic thrombocytopenic purpura and atypical hemolytic uremic syndrome, are associated with injury and dysregulation of microvascular endothelium and platelets.[A241030] Evidence increasingly points to a role …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mannan-binding lectin serine protease 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NasoVAX DB15859
biotech

NasoVAX contains replication-deficient adenovirus vectors in suspension. It is a vaccine administered through a nasal spray that expresses influenza hemagglutinin in nasal epithelial cells[L16313]. Created by Altimmune, Inc., NasoVAX is currently being devel…

Waktu Paruh-
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Natamycin Approved DB00826
small molecule | CAS: 7681-93-8

Amphoteric macrolide antifungal antibiotic from Streptomyces natalensis or S. chattanoogensis. It is used for a variety of fungal infections, mainly topically. [PubChem]

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
Ergosterol
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nateglinide Approved DB00731
small molecule | CAS: 105816-04-4

Nateglinide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It belongs to the meglitinide class of short-acting insulin secretagogues, which act by binding to ? cells of the pancreas to stimulate i…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +21
Target Protein:
ATP-binding cassette sub-family C member 8Peroxisome proliferator-activated receptor gamma
Waktu Paruh1.5 hours
Vol. Distribusi10 liters in health…
Klirens-
Genetik -
biotech

Natural Killer (NK) cells originate and differentiate from hematopoietic stem cells through various signalling pathways involving cytokines and interleukins. These cells arise from CD34+ lymphoid progenitors and comprise 10-15% of all lymphocytes in human per…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
NAV 1800 DB05437
biotech

RIGScan CR49, a 125I-labelled CR monoclonal antibody directed against the tumour-associated antigen TAG-72, is undergoing development with Neoprobe for the intraoperative detection of metastatic colorectal cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Navafenterol DB19195
small molecule | CAS: 1435519-06-4

Navafenterol is under investigation in clinical trial NCT02971293 (Efficacy, Pharmacokinetics (PK), Safety and Tolerability Study of Inhaled AZD8871).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Navicixizumab DB12634
biotech | CAS: 1638338-43-8

Navicixizumab is under investigation in clinical trial NCT02298387 (A Phase 1 Study of Navicixizumab in Subjects With Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Navitoclax DB12340
small molecule | CAS: 923564-51-6

Navitoclax has been used in trials studying the treatment and basic science of Solid Tumors, Non-Hodgkin's Lymphoma, EGFR Activating Mutation, Chronic Lymphoid Leukemia, and Hematological Malignancies, among others. Navitoclax is an orally bioavailable sma…

Kategori:
AmidesAminesAntineoplastic Agents +3
Target Protein:
Bcl-2-like protein 1G1/S-specific cyclin-D1Apoptosis regulator Bcl-2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Navocaftor DB19039
small molecule | CAS: 2159103-66-7

Navocaftor is under investigation in clinical trial NCT04853368 (Study to Evaluate Adverse Events and Change in Disease Activity With Oral Capsules of Galicaftor/navocaftor/abbv-119 or Galicaftor/navocaftor/abbv-576 Combination Therapies in Adult Participants…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Navtemadlin DB15299
small molecule | CAS: 1352066-68-2

Navtemadlin (AMG-232) is under investigation in clinical trial NCT03041688 (MDM2 Inhibitor AMG-232 and Decitabine in Treating Patients With Relapsed, Refractory, or Newly-Diagnosed Acute Myeloid Leukemia).

Kategori:
Acids, AcyclicAntineoplastic AgentsFatty Acids +3
Target Protein:
E3 ubiquitin-protein ligase Mdm2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naxitamab Approved DB15965
biotech | CAS: 1879925-92-4

Naxitamab (humanized 3F8, hu3F8) is an IgG1 monoclonal antibody directed against the oncofetal differentiation antigen GD2 disialoganglioside.[L24454,A224604] Normally expressed during fetal development and in mature neurons, pain fibers, and skin cells, GD2 …

Kategori:
Agents that produce hypertensionAmino Acids, Peptides, and ProteinsAntibodies +18
Target Protein:
GD2 disialoganglioside
Waktu ParuhThe mean terminal h…
Vol. Distribusi-
KlirensThe clearance of na…
Genetik -
NC-6300 DB17341
small molecule

NC-6300, also known as K-912, is a novel [epirubicin] drug-conjugated polymeric micelle.

Kategori:
Amino Acids, Peptides, and ProteinsAminoglycoside AntibacterialsAnthracyclines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NCX-1000 DB16026
small molecule | CAS: 401519-96-8

NCX-1000 is under investigation in clinical trial NCT00414869 (Preliminary Efficacy and Tolerability of NCX-1000 After Repeated Oral Doses in Patients With Elevated Portal Pressure).

Kategori:
AnionsBile Acids and SaltsCholanes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NDI-5001 DB17609
small molecule | CAS: 1365571-66-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Neamine DB04808
small molecule | CAS: 3947-65-7

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Necitumumab Approved DB09559
biotech | CAS: 906805-06-9

Necitumumab is an intravenously administered recombinant monoclonal IgG1 antibody used in the treatment of non-small cell lung cancer (NSCLC) as an EGFR antagonist. It functions by binding to epidermal growth factor receptor (EGFR) and prevents binding of its…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptor
Waktu ParuhElimination half li…
Vol. DistribusiSteady state volume…
Klirens14.1 mL/h
Genetik -
Necuparanib DB16251
small molecule | CAS: 1415139-34-2

Necuparanib is under investigation in clinical trial NCT01621243 (M402 in Combination With Nab-paclitaxel and Gemcitabine in Pancreatic Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nedaplatin Approved DB13145
small molecule | CAS: 95734-82-0

Nedaplatin is a second generation platinum analog [A20300]. It is less nephrotoxic than [DB00515] but has proven equally effective. It was approved for use in Japan in 1995.

Kategori:
Antineoplastic AgentsDrugs that are Mainly Renally ExcretedDrugs that are Mainly Renally Excreted with a Narrow Therapeutic Index +3
Target Protein:
DNAGlutathione
Waktu Paruh-
Vol. DistribusiThe volume of distr…
KlirensClearance of the fr…
Genetik -
Nedisertib DB16252
small molecule | CAS: 1637542-33-6

Nedisertib is under investigation in clinical trial NCT03770689 (Study of M3814 in Combination With Capecitabine and Radiotherapy in Rectal Cancer).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
DNA-dependent protein kinase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4451–4500 dari 6694
Sebelumnya Halaman 90 / 134 Berikutnya