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2279

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866 (38.0%)
Target
1100 (48.3%)
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Hasil Pencarian (2279)

Halaman 9 / 46
Butorphanol Approved DB00611
small molecule | CAS: 42408-82-2

A synthetic morphinan analgesic with narcotic antagonist action. It is used in the management of severe pain.

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +18
Target Protein:
Kappa-type opioid receptorDelta-type opioid receptorMu-type opioid receptor
Waktu ParuhThe elimination hal…
Vol. Distribusi* 305 to 901 L
Klirens* 99 +/- 23 L/h [Yo…
Genetik -
BW-A 58C DB06740
small molecule | CAS: 94015-46-0

BW-A 58C, also known as 2-(4-tert-butylcyclohexyl)-3-hydroxy-1,4-naphthoquinone, is an experimental naphthoquinone antimalarial drug which undergoes extensive alkyl hydroxylation to a single t-butylhydroxy metabolite in man in vivo and also in human liver mic…

Kategori:
NaphthalenesQuinones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
C-peptide DB16187
small molecule | CAS: 59112-80-0

C-peptide is under investigation in clinical trial NCT00278980 (Effect of C-peptide on Diabetic Peripheral Neuropathy).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
C134 DB18261
biotech

C134 is a genetically engineered oncolytic herpes simplex virus expressing human cytomegalovirus (HCMV) internal repeat short 1 (IRS1).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
C31G DB05398
small molecule

C31G is a potent broad spectrum antimicrobial agent, effective against gram positive and gram negative bacteria, yeast and fungi.C31G, vaginal gel is developed by Biosyn Inc. and has commenced enrollment in a phase III pivotal clinical trial for the reduction…

Kategori:
AminesFatty AcidsLipids +3
Target Protein:
Gag-Pol polyproteinCD9 antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CA4P DB05284
small molecule | CAS: 222030-63-9

CA4P has been shown in the laboratory to shut down the blood supply to tumours. It is one of the first vascular targeting drugs to be tested in patients. This drug was originally isolated from the African Bush Willow. The first studies in patients with this d…

Target Protein:
Tubulin beta chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 12321-44-7

Calcitonin is a polypeptide hormone secreted by the parafollicular cells of the thyroid gland in mammals. It inhibits bone resorption and lowers both serum and urinary calcium concentrations. Human calcitonin is available only in very small quantities but has…

Kategori:
Bone Density Conservation AgentsCalcitonin PreparationsCalcium Homeostasis +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Calcitriol Approved DB00136
small molecule | CAS: 32222-06-3

Calcitriol is an active metabolite of vitamin D with 3 hydroxyl (OH) groups and is commonly referred to as 1,25-dihydroxycholecalciferol, or 1alpha,25-dihydroxyvitamin D<sub>3</sub>, 1,25-dihydroxyvitamin D<sub>3</sub>. It is produced in the body after series…

Kategori:
Alimentary Tract and MetabolismAntipsoriaticsAntipsoriatics for Topical Use +27
Target Protein:
Vitamin D3 receptorHomeobox protein Hox-A10
Waktu ParuhAfter administratio…
Vol. DistribusiUpon intravenous ad…
KlirensThe metabolic clear…
Genetik -
Calfactant Approved DB06415
small molecule | CAS: 183325-78-2

Calfactant is a sterile, non-pyrogenic lung surfactant intended for intratracheal instillation. It is an off-white suspension of an extract of natural surfactant from calf lungs suspended in 0.9% saline. Each milliliter of calfactant contains 35mg of phosphol…

Kategori:
Alveolar Surface Tension ReductionBradycardia-Causing AgentsComplex Mixtures +6
Waktu ParuhHalf time clearance…
Vol. DistribusiNo human studies on…
KlirensNo human studies on…
Genetik -
Calmangafodipir DB18398
small molecule | CAS: 1401243-67-1

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmines +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Calpurbatug DB18734
biotech | CAS: 2635404-72-5

Calpurbatug (TRL1068) is a high-affinity and broad-spectrum human antibody that targets and disintegrates bacterial biofilm.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CALY-002 DB18378
biotech

CALY-002 is a humanized monoclonal antibody targeting interleukin-15.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CAM-101 DB18414
biotech

CAM-101 is an allogeneic human platelet lysate product depleted of fibrinogen.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CAM-GM201 DB17687
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Camoteskimab DB18876
biotech | CAS: 2492472-82-7

Camoteskimab is under investigation in clinical trial NCT06436183 (A Study of the Effects of Camoteskimab in Adults With Moderate to Severe Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CAN-106 DB18389
biotech

CAN-106 a novel, long-acting monoclonal antibody directed against human complement C5.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canagliflozin Approved DB08907
small molecule | CAS: 842133-18-0

Canagliflozin, also known as _Invokana_, is a sodium-glucose cotransporter 2 (SGLT2) inhibitor used in the management of type 2 diabetes mellitus along with lifestyle changes including diet and exercise [FDA label]. It was initially approved by the FDA in …

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +15
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhIn a clinical study…
Vol. DistribusiThis drug is extens…
KlirensIn healthy subjects…
Genetik -
Canakinumab Approved DB06168
biotech | CAS: 914613-48-2

Canakinumab is a recombinant, human anti-human-IL-1? monoclonal antibody that belongs to the IgG1/? isotype subclass. It is expressed in a murine Sp2/0-Ag14 cell line and comprised of two 447- (or 448-) residue heavy chains and two 214-residue light chains, w…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +13
Target Protein:
Interleukin-1 beta
Waktu Paruh26 days
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ca…
Genetik -
Cannabidiol Approved DB09061
small molecule | CAS: 13956-29-1

Cannabidiol, or CBD, is one of at least 85 active cannabinoids identified within the Cannabis plant. It is a major phytocannabinoid, accounting for up to 40% of the Cannabis plant's extract, that binds to a wide variety of physiological targets of the endocan…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnticonvulsants +56
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +36
Waktu ParuhThe CBD component o…
Vol. DistribusiCannabinoids are di…
Klirens-
Genetik -
Cannabidivarin DB14050
small molecule | CAS: 24274-48-4

Cannabidivarin, also known as cannabidivarol or CBDV, is a non-psychoactive cannabinoid found within [DB14009]. It is one of over 100 cannabinoids identified from the Cannabis plant that can modulate the physiological activity of cannabis, or marijuana [A3258…

Kategori:
AnticonvulsantsCentral Nervous System DepressantsTerpenes
Target Protein:
Transient receptor potential cation channel subfamily V member 1Transient receptor potential cation channel subfamily V member 2Transient receptor potential cation channel subfamily A member 1 +1
Waktu ParuhOrally administered…
Vol. DistribusiDue to its lipophil…
Klirens-
Genetik -
Canoctakin DB18195
biotech | CAS: 1019859-03-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cantharidin Approved DB12328
small molecule | CAS: 56-25-7

Cantharidin is a naturally occurring odorless, colorless fatty substance of the terpenoid class that is produced as an oral fluid in the alimentary canal of the male blister beetle.[A32891, A32892] For its natural purpose, the male blister beetle secretes and…

Kategori:
BenzofuransCompounds used in a research, industrial, or household settingEnzyme Inhibitors +4
Target Protein:
Serine/threonine-protein phosphatase PP1-alpha catalytic subunitAryl hydrocarbon receptor
Waktu ParuhLittle pharmacodyna…
Vol. DistribusiAfter oral or IP in…
KlirensLittle pharmacodyna…
Genetik -
biotech | CAS: 400010-39-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caplacizumab Approved DB06081
biotech | CAS: 915810-67-2

Caplacizumab, firstly called ALX-0081, is a humanized single-variable-domain immunoglobulin consisting of two identical humanized building blocks genetically linked by a three-alanine linker. Caplacizumab was developed by Ablynx, a Sanofi company and FDA appr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
von Willebrand factor
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensAs the elimination …
Genetik -
Capmatinib Approved DB11791
small molecule | CAS: 1029712-80-8

Capmatinib is a small molecule kinase inhibitor targeted against c-Met (a.k.a. hepatocyte growth factor receptor [HGFR]), a receptor tyrosine kinase that, in healthy humans, activates signaling cascades involved in organ regeneration and tissue repair.[A19912…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +20
Target Protein:
Hepatocyte growth factor receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Capsaicin Approved DB06774
small molecule | CAS: 404-86-4

Capsaicin is most often used as a topical analgesic and exists in many formulations of cream, liquid, and patch preparations of various strengths; however, it may also be found in some dietary supplements. Capsaicin is a naturally-occurring botanical irritant…

Kategori:
AlkaloidsAlkenesAmides +28
Target Protein:
Transient receptor potential cation channel subfamily V member 1Prohibitin-2
Waktu ParuhFollowing oral inge…
Vol. Distribusi-
Klirens-
Genetik -
Capsicum oleoresin Approved DB11131
biotech | CAS: 8023-77-6

Capsicum oleoresin is an oily organic resin derived from the fruit of plants in the Capsicum genus, such as chilli peppers. When the plants are finely ground, capsicum oleoresin is formed after the extraction process of capsaicin using oragnic solvents such a…

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Carbinoxamine Approved DB00748
small molecule | CAS: 486-16-8

Carbinoxamine is a first generation antihistamine that competes with free histamine for binding at HA-receptor sites. This antagonizes the effects of histamine on HA-receptors, leading to a reduction of the negative symptoms brought on by histamine HA-recepto…

Kategori:
Aminoalkyl EthersAntihistamines for Systemic UseCentral Nervous System Depressants +8
Target Protein:
Histamine H1 receptor
Waktu Paruh10 to 20 hours
Vol. Distribusi-
Klirens-
Genetik -
Carbocromen Approved DB13279
small molecule | CAS: 804-10-4

Carbocromen was marketed for use in Germany as a vasodilator, however, it has been discontinued due to the risk of arrhythmia development [L5635].

Kategori:
BenzopyransCardiac TherapyCardiovascular Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carbon monoxide Approved DB11588
small molecule | CAS: 630-08-0

Carbon monoxide (CO) is a colorless, odorless, and tasteless gas that has a slightly lower density than air. It is toxic to hemoglobin utilizing animals (including humans), when encountered in concentrations above about 35 ppm, although it is also formed in n…

Kategori:
Carbon Compounds, InorganicDiagnostic AgentsGases +6
Target Protein:
Myoglobin
Waktu ParuhThe half-life of ca…
Vol. Distribusi-
Klirens-
Genetik -
Cardiotrophin 1 DB18399
biotech | CAS: 1422101-11-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carfentanil DB01535
small molecule | CAS: 59708-52-0

Carfentanil or carfentanyl (Wildnil) is an analogue of the popular synthetic opioid analgesic fentanyl, and is one of the most potent opioids known (also the most potent opioid used commercially). Carfentanil was first synthesized in 1974 by a team of chemist…

Kategori:
AnalgesicsCarbon RadioisotopesCentral Nervous System Agents +9
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cariprazine Approved DB06016
small molecule | CAS: 839712-12-8

Cariprazine is an atypical antipsychotic agent and a piperazine derivative that was first developed in Hungary.[A247100] It works as a partial agonist at central dopamine D2, dopamine D3, and serotonin 5-HT<sub>1A</sub> receptors and as an antagonist at serot…

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntipsychotic Agents +48
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor5-hydroxytryptamine receptor 1A +5
Waktu ParuhCariprazine and its…
Vol. Distribusi-
Klirens-
Genetik -
Carlumab DB12718
biotech | CAS: 915404-94-3

Carlumab has been used in trials studying the treatment of Cancer and Prostate Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carotuximab DB06322
biotech | CAS: 1268714-50-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Endoglin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carphenazine DB01038
small molecule | CAS: 2622-30-2

Carphenazine is an antipsychotic drug, used in hospitalized patients in the management of chronic schizophrenic psychoses.

Kategori:
Dopamine AntagonistsDopamine D2 Receptor Antagonists
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carprofen Approved DB00821
small molecule | CAS: 53716-49-7

Carprofen is a non-steroidal anti-inflammatory drug (NSAID) that is used by veterinarians as a supportive treatment for the relief of arthritic symptoms in geriatric dogs. Carprofen was previously used in human medicine for over 10 years (1985-1995). It was g…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +15
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhApproximately 8 hou…
Vol. Distribusi-
Klirens-
Genetik -
Casdozokitug DB17513
biotech | CAS: 2643331-37-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Casimersen Approved DB14984
biotech | CAS: 1422958-19-7

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive impairment of ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albe…

Kategori:
Antisense OligonucleotidesCytochrome P-450 CYP2C19 InhibitorsCytochrome P-450 CYP2C19 inhibitors (strength unknown) +16
Target Protein:
DMD gene (exon 45 casimersen target site)
Waktu ParuhCasimersen has an e…
Vol. DistribusiCasimersen administ…
KlirensCasimersen administ…
Genetik -
Casirivimab Approved DB15941
biotech | CAS: 2415933-42-3

Casirivimab is a monoclonal antibody combined with [Imdevimab] in Regeneron's antibody cocktail known as REGN-COV2 for the treatment of COVID-19.[L23539] This drug is a combination of antibodies derived from humanized VelocImmune® mice in addition to blood s…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Castor oil Approved DB11113
biotech | CAS: 8001-79-4

Castor oil is a vegetable oil obtained by pressing the seeds of the castor oil plant (_Ricinus communis_ L.) mainly cultivated in India, South America, Africa, and China. Castor oil is a rich source of [DB02955], which represents up to 90% of the total castor…

Kategori:
Alimentary Tract and MetabolismBiological ProductsComplex Mixtures +10
Target Protein:
Prostaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP4 subtype
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Cathinone DB01560
small molecule | CAS: 71031-15-7

Cathinone is a monoamine alkaloid found in the shrub Catha edulis (Khat). Closely related to ephedrine, cathine and other amphetamines, it is probably the main contributor to the stimulant effect of Catha edulis. Cathinone differs from many other amphetamines…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCentral Nervous System Stimulants +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Catridecacog Approved DB09310
biotech | CAS: 606138-08-3

Coagulation Factor XIII A-Subunit (Recombinant), also known as catridecacog, is a recombinant form of the Factor XIII-A2 homodimer composed of two factor XIII (FXIII) A-subunits [FDA Label]. For people with congenital deficiency or mutation of Factor XIII, a …

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
Coagulation factor XIII B chain
Waktu Paruh7.1 days
Vol. Distribusi-
Klirens0.41 mL/h/kg
Genetik -
Catumaxomab Approved DB06607
biotech | CAS: 509077-98-9

Catumaxumab is a trifunctional monoclonal antibody developed for use in cancer treatment. It has affinity for T-cells, accessory immune cells, and cancer cells. Catumaxumab was initially authorized for market by the European Medicines Agency in April 2009 for…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Low affinity immunoglobulin gamma Fc region receptor II-aLow affinity immunoglobulin gamma Fc region receptor III-ALow affinity immunoglobulin gamma Fc region receptor III-B +3
Waktu ParuhCatumaxomab has an …
Vol. Distribusi-
Klirens-
Genetik -
CCR5 mAb DB05906
biotech

CCR5 mAb is a fully human monoclonal antibody that specifically recognizes and binds the chemokine receptor CCR5, which is known to be a key facilitator of infection with human immunodeficiency virus (HIV-1). It was generated by HGS using the Abgenix XenoMous…

Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDX-1135 DB17607
biotech

CDX-1135, formerly TP-10, is a soluble, recombinant human Complement Receptor Type 1 (sCR1) developed by Avant Immunotherapeutics (now Celldex). It was investigated in clinical trials for post-cardiopulmonary bypass syndrome and kidney damage.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsProteins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefamandole Approved DB01326
small molecule | CAS: 34444-01-4

Cefamandole is also known as cephamandole. It is a parenterally administered broad-spectrum cephalosporin antibiotic. It is generally formulated as a formate ester, [cefamandole nafate]. It is no longer marketed in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 2
Waktu ParuhThe half-life after…
Vol. Distribusi-
Klirens-
Genetik -
Cefamandole nafate Approved DB14725
small molecule | CAS: 57268-80-1

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefapirin Approved DB01139
small molecule | CAS: 21593-23-7

Cefapirin (INN, also spelled cephapirin), commonly marketed under the trade name Cefadyl, is a first-generation cephalosporin antibiotic that is available in injectable formulations. Production for use in humans has been discontinued in the United States. Cef…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefmetazole Approved DB00274
small molecule | CAS: 56796-20-4

A semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It has a high rate of efficacy in many types of infection and to date no severe side effects have been noted.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin binding protein 2aPenicillin-binding protein 1APenicillin-binding protein 1B +3
Waktu Paruh1.50 &plusmn;0.14 h…
Vol. Distribusi-
Klirens-
Genetik -
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